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Cathepsin L2 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
Gallinamide AIC50140.0 [1], 460.0 [2]
Citrusinine IIC502200.0 [1]
Citrusinine IKi1000.0 [1]
1,3,5-Trihydroxy-2,8-bis(3-methyl-2-butenyl)-10-methylacridine-9(10H)-oneIC503900.0 [1]
1,3,5-Trihydroxy-2,8-bis(3-methyl-2-butenyl)-10-methylacridine-9(10H)-oneKi1200.0 [1]
Cathepsin inhibitor 1IC50199.53 [1]
Citrusinine IIIC5010000.0 [1]
Citrusinine IIKi4200.0 [1]
5-Tert-butyl-N-[(2S)-1-(cyanomethylamino)-3-(3-methylphenyl)-1-oxopropan-2-yl]-2-methylpyrazole-3-carboxamideIC50398.11 [1]
Glycocitrine-IVIC502200.0 [1]
Glycocitrine-IVKi1100.0 [1]
CitbrasineIC501200.0 [1]
CitbrasineKi200.0 [1]
N-[(2S)-3-(3-Chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]benzamideIC50794.33 [1]
1,3,5-Trihydroxy-4-methoxy-10-methyl-2,8-bis(3-methylbut-2-enyl)acridin-9-oneIC502500.0 [1]
1,3,5-Trihydroxy-4-methoxy-10-methyl-2,8-bis(3-methylbut-2-enyl)acridin-9-oneKi500.0 [1]
4,9-Dihydroxy-2-(2-hydroxypropan-2-yl)-11-methoxy-10-methyl-2,3-dihydrofuro[3,2-b]acridin-5-oneIC505200.0 [1]
4,9-Dihydroxy-2-(2-hydroxypropan-2-yl)-11-methoxy-10-methyl-2,3-dihydrofuro[3,2-b]acridin-5-oneKi4400.0 [1]
Glycocitrine-IIC5025000.0 [1]
Glycocitrine-IKi10000.0 [1]
3,5,8-Trihydroxy-6-methoxy-2,2,7-trimethyl-3,4-dihydropyrano[2,3-a]acridin-12-oneIC502800.0 [1]
3,5,8-Trihydroxy-6-methoxy-2,2,7-trimethyl-3,4-dihydropyrano[2,3-a]acridin-12-oneKi1700.0 [1]
2-(4-Butylphenyl)-1H-quinolin-4-oneIC505200.0 [1]
2-(4-Butylphenyl)-1H-quinolin-4-oneKi800.0 [1]
3-Phenylmethoxy-10H-acridin-9-oneIC503600.0 [1]
3-Phenylmethoxy-10H-acridin-9-oneKi1300.0 [1]
2-Nitro-7-phenylmethoxy-10H-acridin-9-oneIC501700.0 [1]
2-Nitro-7-phenylmethoxy-10H-acridin-9-oneKi400.0 [1]
3-(3-Methoxy-4-phenylmethoxyanilino)naphthalene-2-carboxylic acidIC501800.0 [1]
3-(3-Methoxy-4-phenylmethoxyanilino)naphthalene-2-carboxylic acidKi1100.0 [1]
3-(3-Nitro-4-phenylmethoxyanilino)naphthalene-2-carboxylic acidIC501000.0 [1]
3-(3-Nitro-4-phenylmethoxyanilino)naphthalene-2-carboxylic acidKi800.0 [1]
TelaprevirIC501350.0 [1]
BoceprevirIC5075.0 [1]
OdanacatibIC50762.0 [1]
2-Phenylquinolin-4-olIC504700.0 [1]
RelacatibKi0.06 [1]
(1R,21S,24S)-21-Tert-butyl-N-[(1R,2S)-1-(cyclopropylsulfonylcarbamoyl)-2-ethenylcyclopropyl]-16,16-dimethyl-3,19,22-trioxo-2,18-dioxa-4,20,23-triazatetracyclo[21.2.1.14,7.06,11]heptacosa-6(11),7,9-triene-24-carboxamideIC5010000.0 [1]
2-((4-Methoxyphenyl)amino)benzoic acidIC5050000.0 [1]
11-HydroxynoracronycineIC5048000.0 [1]
2-Undecyl-4(1H)-quinolinoneIC509900.0 [1]
Grassystatin AIC5010000.0 [1]
Cruzain-IN-1IC50239.88 [1]
9-(3,5-Difluorophenyl)-6-(ethylamino)-2-purinecarbonitrileIC5070794.58 [1]
2-(p-Methylphenyl)quinolin-4(1H)-oneIC505000.0 [1]
[(2S)-3,3-Dimethyl-1-[3-[4-(trifluoromethyl)phenyl]pyrazol-1-yl]butan-2-yl] N-[(3S)-1,2-dioxo-1-(1H-pyrazol-5-ylamino)heptan-3-yl]carbamateIC50170.0 [1]
N-[(2S)-3-Cyclohexyl-1-[2-(4-methoxyanilino)ethylamino]-1-oxopropan-2-yl]-5-[3-(trifluoromethyl)phenyl]furan-2-carboxamideKi20000.0 [1]
N-[(2S)-4-Methyl-1-oxo-1-[[(4S)-3-oxo-1-pyridin-2-ylsulfonylazepan-4-yl]amino]pentan-2-yl]-1-benzofuran-2-carboxamideKi1.8 [1]
[(3S)-4,4-Dimethyl-2-oxooxolan-3-yl] N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC5079.0 [1]
[(2R)-1-[5-(4-Fluorophenyl)-1,3,4-oxadiazol-2-yl]-3,3-dimethylbutan-2-yl] N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC5034000.0 [1]
[(2R)-3,3-Dimethyl-1-(5-phenyl-1,3,4-oxadiazol-2-yl)butan-2-yl] N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC501600.0 [1]
[(2S)-3,3-Dimethyl-1-[4-[4-(trifluoromethyl)phenyl]pyrazol-1-yl]butan-2-yl] N-[(3S)-1,2-dioxo-1-(1H-pyrazol-5-ylamino)heptan-3-yl]carbamateIC50430.0 [1]
[(2S)-3,3-Dimethyl-1-[4-[4-(trifluoromethyl)phenyl]imidazol-1-yl]butan-2-yl] N-[(3S)-1,2-dioxo-1-(1H-pyrazol-5-ylamino)heptan-3-yl]carbamateIC50130.0 [1]
[(2R)-3,3-Dimethyl-1-[5-[4-(trifluoromethyl)phenyl]-1,3,4-oxadiazol-2-yl]butan-2-yl] N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC505000.0 [1]
[(2R)-3,3-Dimethyl-1-[5-[4-(trifluoromethyl)phenyl]-1,3,4-oxadiazol-2-yl]butan-2-yl] N-[(3S)-1,2-dioxo-1-(1H-pyrazol-5-ylamino)heptan-3-yl]carbamateIC501200.0 [1]
[(2S)-3,3-Dimethyl-1-[4-[4-(trifluoromethyl)phenyl]imidazol-1-yl]butan-2-yl] N-[(3S)-1,2-dioxo-1-(1,3-thiazol-2-ylamino)heptan-3-yl]carbamateIC5036000.0 [1]
6-[4-[3-(4-Ethylpiperazin-1-yl)propoxy]-3-(trifluoromethyl)phenyl]-1-methylimidazo[4,5-c]pyridine-4-carbonitrileIC5010000.0 [1]
2-Methoxy-7-nitroacridin-9(10H)-oneIC502000.0 [1]
[(2S)-3,3-Dimethyl-1-[2-oxo-3-[4-(trifluoromethyl)phenyl]imidazolidin-1-yl]butan-2-yl] N-[(3S)-1,2-dioxo-1-(1H-pyrazol-5-ylamino)heptan-3-yl]carbamateIC501700.0 [1]
[(2R)-1-[5-(4-Fluorophenyl)-1,3,4-oxadiazol-2-yl]-3,3-dimethylbutan-2-yl] N-[(3S)-1,2-dioxo-1-(pyridin-3-ylmethylamino)heptan-3-yl]carbamateIC5014000.0 [1]
1-Methyl-6-[4-(2-piperidin-4-ylethoxy)-3-(trifluoromethyl)phenyl]imidazo[4,5-c]pyridine-4-carbonitrileIC5010000.0 [1]
6-[4-[3-(Dimethylamino)propoxy]-3-(trifluoromethyl)phenyl]-1-methylimidazo[4,5-c]pyridine-4-carbonitrileIC5010000.0 [1]
[(2R)-3,3-Dimethyl-1-[5-[4-(trifluoromethyl)phenyl]-1,3,4-oxadiazol-2-yl]butan-2-yl] N-[(3S)-1,2-dioxo-1-[(2-oxo-1,3-oxazolidin-3-yl)amino]heptan-3-yl]carbamateIC507100.0 [1]
(3S)-19-Chloro-N-(1-cyanocyclopropyl)-5-oxo-9-(trifluoromethyl)-12,17-dioxa-4-azatricyclo[16.2.2.06,11]docosa-1(20),6(11),7,9,18,21-hexaene-3-carboxamideIC501043.0 [1]
[(2S)-3,3-Dimethyl-1-[3-[4-(trifluoromethyl)phenyl]pyrazol-1-yl]butan-2-yl] N-[(3S)-1-(1,2-oxazol-5-ylmethylamino)-1,2-dioxoheptan-3-yl]carbamateIC5036000.0 [1]
[(2R)-3-Methyl-1-(5-phenyl-1,3,4-oxadiazol-2-yl)butan-2-yl] N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC505600.0 [1]
[(2R)-1-[5-(4-Fluorophenyl)-1,3,4-oxadiazol-2-yl]-3,3-dimethylbutan-2-yl] N-[(3S)-1,2-dioxo-1-(1H-pyrazol-5-ylamino)heptan-3-yl]carbamateIC50230000.0 [1]
[(2R)-3,3-Dimethyl-1-(5-phenyl-1,3,4-oxadiazol-2-yl)pentan-2-yl] N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC502800.0 [1]
[(2S)-3,3-Dimethyl-1-[3-[4-(trifluoromethyl)phenyl]pyrazol-1-yl]butan-2-yl] N-[(3S)-1,2-dioxo-1-(pyridin-2-ylamino)heptan-3-yl]carbamateIC504500.0 [1]
2-(Furan-2-yl)-1H-quinolin-4-oneIC504700.0 [1]
[(3S)-4,4-Dimethyl-2-oxopyrrolidin-3-yl] N-[(3S)-1,2-dioxo-1-[[(1R)-1-phenylethyl]amino]heptan-3-yl]carbamateIC5029.0 [1]
2-Anilino-3-methoxybenzoic acidIC5050000.0 [1]
(3R,4R)-4-(2,3-Dimethylphenoxy)piperidin-3-olIC50100000.0 [1]
(4S,5R)-4-(2,3-Dimethylphenoxy)-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC50131.0 [1]
2-(3-Benzyloxyphenylamino)benzoic acidIC502100.0 [1]
2-Anilino-5-nitrobenzoic acidIC5010000.0 [1]
(4S,5S)-4-(2,3-Dimethylphenoxy)-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC503317.0 [1]
(4S,5R)-4-Phenoxy-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC50158.0 [1]
(4S,5R)-4-Phenylmethoxy-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC501289.0 [1]
(4S,5R)-4-(2-Methylpropoxy)-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC50894.0 [1]
(4S,5S)-4-Bromo-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC5010000.0 [1]
1-[4-[4-[(1S)-1-[[(2S)-1-[[(1S)-1-Cyano-2-(4-cyano-2-fluorophenyl)ethyl]amino]-3-methyl-1-oxobutan-2-yl]amino]-2,2,2-trifluoroethyl]phenyl]phenyl]cyclopropane-1-carboxamideIC5079.0 [1]
(2S)-N-[(1S)-1-Cyano-2-(4-cyano-2-fluorophenyl)ethyl]-2-[[(1S)-1-[4-[4-[(1R)-2,2-difluoro-1-hydroxyethyl]phenyl]phenyl]-2,2,2-trifluoroethyl]amino]-3-methylbutanamideIC5069.0 [1]
(2S)-N-[(1S)-1-Cyano-2-(4-cyano-2-fluorophenyl)ethyl]-3-methyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]butanamideIC5028.0 [1]
N-[(2S)-3-(3-Chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]cyclohexanecarboxamideIC506309.57 [1]
N-[(2S)-3-(3-Chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]cyclohexene-1-carboxamideIC50398.11 [1]
N-[(2S)-3-(3-Chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]cycloheptanecarboxamideIC506309.57 [1]
N-[(2S)-3-(3-Chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]-4-methylbenzamideIC501000.0 [1]
N-[(2S)-3-(3-Chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]-3-methylbenzamideIC50794.33 [1]
N-[(2S)-3-(3-Chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]-2-methylbenzamideIC505011.87 [1]
3-Chloro-N-[(2S)-3-(3-chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]benzamideIC50199.53 [1]
N-[(2S)-3-(3-Chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]-2,5-dimethylbenzamideIC501584.89 [1]
N-[(2S)-3-(3-Chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]-2,3-dimethylbenzamideIC503981.07 [1]
N-[(2S)-3-(3-Chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]-3,5-dimethylbenzamideIC50199.53 [1]
N-[(2S)-3-(3-Chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]naphthalene-1-carboxamideIC503981.07 [1]
N-[(2S)-3-(3-Chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]-5,6,7,8-tetrahydronaphthalene-1-carboxamideIC5010000.0 [1]
N-[(2S)-3-(3-Chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]quinoline-4-carboxamideIC503162.28 [1]
N-[(2S)-3-(3-Chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]-3,7-dimethylnaphthalene-1-carboxamideIC501000.0 [1]
N-[(2S)-3-(3-Chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]-1,3-dimethylpyrazole-4-carboxamideIC501258.93 [1]
N-[(2S)-3-(3-Chlorophenyl)-1-(cyanomethylamino)-1-oxopropan-2-yl]-2,5-dimethylpyrazole-3-carboxamideIC501258.93 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Cathepsin L2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/cathepsin-l2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Cathepsin L2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cathepsin-l2-inhibitors-ic50-ki.
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