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CDK1/Cyclin A Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
StaurosporineIC501.7 [1]
Oxindole-Based Inhibitor 22IC5010.0 [1]
Oxindole-Based Inhibitor 81IC5012.0 [1]
2-(3-Hydroxy-4-methoxystyryl)-8-hydroxyquinoline-7-carboxylic acidIC5010000.0 [1]
Oxindole-Based Inhibitor 27IC5037.0 [1]
Oxindole-Based Inhibitor 31IC5041.0 [1]
Oxindole-Based Inhibitor 49IC50350.0 [1]
Oxindole-Based Inhibitor 50IC50170.0 [1]
Oxindole-Based Inhibitor 56IC502.8 [1]
Oxindole-Based Inhibitor 79IC5043.0 [1]
2-(2,4-Dihydroxybenzylcarbamoyl)-8-hydroxyquinoline-7-carboxylic acidIC5010000.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
4-(3,3-Diethyl-7-fluoro-2-methylindol-5-yl)-5-fluoro-N-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]pyrimidin-2-amineIC5096.0 [1]
CDK4/6/1 InhibitorIC502707.0 [1]
2-[4-[6-[[5-Fluoro-4-(7'-fluoro-2'-methylspiro[cyclopentane-1,3'-indole]-5'-yl)pyrimidin-2-yl]amino]pyridin-3-yl]piperazin-1-yl]ethanolIC50328.0 [1]
4-(3-Ethyl-2,3-dimethylindol-5-yl)-5-fluoro-N-(5-piperazin-1-ylpyridin-2-yl)pyrimidin-2-amineIC50142.0 [1]
5-Fluoro-4-(7-fluoro-2,3,3-trimethylindol-5-yl)-N-(5-piperazin-1-ylpyridin-2-yl)pyrimidin-2-amineIC502224.0 [1]
4-(3-Ethyl-7-fluoro-2,3-dimethylindol-5-yl)-5-fluoro-N-(5-piperazin-1-ylpyridin-2-yl)pyrimidin-2-amineIC5084.0 [1]
5-Fluoro-4-(2'-methylspiro[cyclopentane-1,3'-indole]-5'-yl)-N-(5-piperazin-1-ylpyridin-2-yl)pyrimidin-2-amineIC50234.0 [1]
4-(3,3-Diethyl-7-fluoro-2-methylindol-5-yl)-5-fluoro-N-(5-piperazin-1-ylpyridin-2-yl)pyrimidin-2-amineIC5082.0 [1]
4-(3-Ethyl-7-fluoro-2,3-dimethylindol-5-yl)-5-fluoro-N-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]pyrimidin-2-amineIC50153.0 [1]
N-[5-(4-Ethylpiperazin-1-yl)pyridin-2-yl]-5-fluoro-4-(7'-fluoro-2'-methylspiro[cyclopentane-1,3'-indole]-5'-yl)pyrimidin-2-amineIC501160.0 [1]
4-(3-Ethyl-2,3-dimethylindol-5-yl)-5-fluoro-N-(5-piperidin-4-ylpyridin-2-yl)pyrimidin-2-amineIC50166.0 [1]
4-(3-Ethyl-2,3-dimethylindol-5-yl)-5-fluoro-N-[5-(1-methylpiperidin-4-yl)pyridin-2-yl]pyrimidin-2-amineIC5054.0 [1]
N-[5-[(4-Ethylpiperazin-1-yl)methyl]pyridin-2-yl]-5-fluoro-4-(2'-methylspiro[cyclopentane-1,3'-indole]-5'-yl)pyrimidin-2-amineIC50268.0 [1]
4-(3-Ethyl-7-fluoro-2,3-dimethylindol-5-yl)-N-[5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl]-5-fluoropyrimidin-2-amineIC50966.0 [1]
N-[5-(1-Ethylpiperidin-4-yl)pyridin-2-yl]-5-fluoro-4-(7'-fluoro-2'-methylspiro[cyclopentane-1,3'-indole]-5'-yl)pyrimidin-2-amineIC501071.0 [1]
4-(3-Ethyl-7-fluoro-2,3-dimethylindol-5-yl)-N-[5-(4-ethylpiperazin-1-yl)pyridin-2-yl]-5-fluoropyrimidin-2-amineIC5065.0 [1]
N-[5-(4-Ethylpiperazin-1-yl)pyridin-2-yl]-5-fluoro-4-(2'-methylspiro[cyclopentane-1,3'-indole]-5'-yl)pyrimidin-2-amineIC50915.0 [1]
5-Fluoro-4-(2'-methylspiro[cyclopentane-1,3'-indole]-5'-yl)-N-(5-piperidin-4-ylpyridin-2-yl)pyrimidin-2-amineIC5027.0 [1]
4-(3-Ethyl-7-fluoro-2,3-dimethylindol-5-yl)-5-fluoro-N-[5-(1-methylpiperidin-4-yl)pyridin-2-yl]pyrimidin-2-amineIC50131.0 [1]
5-Fluoro-4-(7'-fluoro-2'-methylspiro[cyclopentane-1,3'-indole]-5'-yl)-N-(5-piperidin-4-ylpyridin-2-yl)pyrimidin-2-amineIC50327.0 [1]
N-[5-[(4-Ethylpiperazin-1-yl)methyl]pyridin-2-yl]-5-fluoro-4-(7'-fluoro-2'-methylspiro[cyclopentane-1,3'-indole]-5'-yl)pyrimidin-2-amineIC502239.0 [1]
5-Fluoro-4-(7'-fluoro-2'-methylspiro[cyclopentane-1,3'-indole]-5'-yl)-N-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]pyrimidin-2-amineIC501444.0 [1]
5-Fluoro-4-(7'-fluoro-2'-methylspiro[cyclopentane-1,3'-indole]-5'-yl)-N-(5-piperazin-1-ylpyridin-2-yl)pyrimidin-2-amineIC50152.0 [1]
5-Fluoro-N-[5-(1-methylpiperidin-4-yl)pyridin-2-yl]-4-(2'-methylspiro[cyclopentane-1,3'-indole]-5'-yl)pyrimidin-2-amineIC5050.0 [1]
4-(3,3-Diethyl-7-fluoro-2-methylindol-5-yl)-N-[5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl]-5-fluoropyrimidin-2-amineIC50436.0 [1]
N-[5-(1-Ethylpiperidin-4-yl)pyridin-2-yl]-5-fluoro-4-(2'-methylspiro[cyclopentane-1,3'-indole]-5'-yl)pyrimidin-2-amineIC50135.0 [1]
5-Fluoro-N-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]-4-(2'-methylspiro[cyclopentane-1,3'-indole]-5'-yl)pyrimidin-2-amineIC50417.0 [1]
4-(3-Ethyl-2,3-dimethylindol-5-yl)-5-fluoro-N-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]pyrimidin-2-amineIC50112.0 [1]
4-(3-Ethyl-2,3-dimethylindol-5-yl)-N-[5-(4-ethylpiperazin-1-yl)pyridin-2-yl]-5-fluoropyrimidin-2-amineIC50101.0 [1]
4-(3-Ethyl-7-fluoro-2,3-dimethylindol-5-yl)-N-[5-(1-ethylpiperidin-4-yl)pyridin-2-yl]-5-fluoropyrimidin-2-amineIC50216.0 [1]
4-(3-Ethyl-7-fluoro-2,3-dimethylindol-5-yl)-5-fluoro-N-(5-piperidin-4-ylpyridin-2-yl)pyrimidin-2-amineIC50110.0 [1]
2-[4-[6-[[5-Fluoro-4-(7'-fluoro-2'-methylspiro[cyclopentane-1,3'-indole]-5'-yl)pyrimidin-2-yl]amino]pyridin-3-yl]piperidin-1-yl]ethanolIC50176.0 [1]
2-[(E)-2-(2,6-Dichlorophenyl)ethenyl]-5,7-dihydroxy-8-[(3S,4R)-3-hydroxy-1-methylpiperidin-4-yl]chromen-4-oneIC504.93 [1]
4-(3-Ethyl-2,3-dimethylindol-5-yl)-N-[5-(1-ethylpiperidin-4-yl)pyridin-2-yl]-5-fluoropyrimidin-2-amineIC50125.0 [1]
5-Fluoro-4-(7'-fluoro-2'-methylspiro[cyclopentane-1,3'-indole]-5'-yl)-N-[5-(4-propan-2-ylpiperazin-1-yl)pyridin-2-yl]pyrimidin-2-amineIC501056.0 [1]
4-{[4-Amino-5-(2-Nitrobenzoyl)-1,3-Thiazol-2-Yl]amino}benzenesulfonamideIC507.6 [1]
Items per page: 1 - 10 of 48
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References

This online tool may be cited as follows

MLA

"Quest Database™ CDK1/Cyclin A Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/cdk1-cyclin-a-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ CDK1/Cyclin A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cdk1-cyclin-a-inhibitors-ic50-ki.
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