Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| 3-Benzyl-1-[4-[(5-cyanopyridin-2-yl)amino]cyclohexyl]-1-[4-(1-methylpyrazol-4-yl)phenyl]urea | IC50 | 63.0 [1], 30000.0 [2] | |
| N-[4-[(5-Cyanopyridin-2-yl)amino]cyclohexyl]-N-[4-(1-methylpyrazol-4-yl)phenyl]acetamide | IC50 | 130.0 [1], 30000.0 [2] | |
| Staurosporine | IC50 | 53.0 [1] | |
| CDK12 inhibitor 2 | IC50 | 52.0 [1] | |
| N-[4-(1-Methylpyrazol-4-yl)phenyl]-N-[4-(quinazolin-2-ylamino)cyclohexyl]acetamide | IC50 | 13.0 [1] | |
MLA | "Quest Database™ CDK12/Cyclin K Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 2 Nov. 2025, https://www.aatbio.com/data-sets/cdk12-cyclin-k-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, November 2). Quest Database™ CDK12/Cyclin K Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cdk12-cyclin-k-inhibitors-ic50-ki. | |
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