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CDK3/Cyclin E Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
StaurosporineIC504.0 [1]
(16E)-14-Methyl-20-oxa-5,7,14,27-tetrazatetracyclo[19.3.1.12,6.18,12]heptacosa-1(25),2(27),3,5,8,10,12(26),16,21,23-decaeneIC503.0 [1]
RGB-286638 free baseIC502.0 [1]
4-[[[4-[5-Chloro-2-[[4-(2-methoxyethylamino)cyclohexyl]amino]pyridin-4-yl]-1,3-thiazol-2-yl]amino]methyl]oxane-4-carbonitrileIC5010000.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
2-[(E)-2-(2,6-Dichlorophenyl)ethenyl]-5,7-dihydroxy-8-[(3S,4R)-3-hydroxy-1-methylpiperidin-4-yl]chromen-4-oneIC501000.0 [1]
(1S,3R)-3-Acetamido-N-[4-(4-fluoro-2-methoxyphenyl)pyridin-2-yl]cyclohexane-1-carboxamideIC5094.0 [1]
(1R,3S)-3-Acetamido-N-[4-(4-fluoro-2-methoxyphenyl)pyridin-2-yl]cyclopentane-1-carboxamideIC50913.0 [1]
4-{[4-Amino-5-(2-Nitrobenzoyl)-1,3-Thiazol-2-Yl]amino}benzenesulfonamideIC5038.0 [1]
2-Chloro-N-methyl-5-[[1-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-ylcarbamoyl)cyclopropyl]amino]benzamideIC5038.0 [1]
2-(3-Hydroxyanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)acetamideIC50128.0 [1]
2-(3-Fluoroanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)acetamideIC50391.0 [1]
2-(4-Chloro-3-methoxyanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)acetamideIC50468.0 [1]
2-(4-Chloro-3-hydroxyanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)acetamideIC5028.0 [1]
2-(4-Chloroanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)acetamideIC5081.0 [1]
2-(3-Aminoanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)acetamideIC50355.0 [1]
2-[3-(Methanesulfonamido)anilino]-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)acetamideIC50410.0 [1]
2-(1H-Indazol-6-ylamino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)acetamideIC5088.0 [1]
2-(3-Acetamido-4-chloroanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)acetamideIC5050.0 [1]
2-Anilino-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]acetamideIC50380.0 [1]
2-Anilino-N-(4-methyl-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)acetamideIC50242.0 [1]
2-(3-Hydroxyanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)propanamideIC5047.0 [1]
2-(4-Chloroanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)propanamideIC5075.0 [1]
2-(3-Acetamido-4-chloroanilino)-2-phenyl-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]acetamideIC50128.0 [1]
N-[2-Chloro-5-[[2-oxo-1-phenyl-2-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]ethyl]amino]phenyl]propanamideIC50353.0 [1]
2-Methyl-2-(4-methylanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)propanamideIC50367.0 [1]
2-(4-Chloroanilino)-3-hydroxy-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)propanamideIC5029.0 [1]
1-(4-Chloroanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)cyclohexane-1-carboxamideIC50412.0 [1]
2-[4-Chloro-3-(propanoylamino)anilino]-2-methyl-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)propanamideIC50103.0 [1]
Ethyl 2-chloro-5-[[2-methyl-1-oxo-1-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-ylamino)propan-2-yl]amino]benzoateIC50157.0 [1]
N-Ethyl-2-fluoro-5-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzamideIC5047.0 [1]
3-[[2-Methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzoic acidIC50333.0 [1]
2-Chloro-N-methyl-5-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzamideIC5023.0 [1]
N-[2-Chloro-5-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]phenyl]cyclopropanecarboxamideIC50165.0 [1]
2-Chloro-N-cyclopropyl-5-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzamideIC5041.0 [1]
2-(4-Fluoroanilino)-2-methyl-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]propanamideIC50163.0 [1]
4-[[2-Chloro-5-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzoyl]amino]butanoic acidIC50180.0 [1]
2-Hydroxyethyl 2-[[3-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzoyl]amino]acetateIC5085.0 [1]
Ethyl 2-chloro-5-[[1-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-ylcarbamoyl)cyclopropyl]amino]benzoateIC50169.0 [1]
2-[4-Chloro-3-(2,3-dihydroxypropoxy)anilino]-2-methyl-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]propanamideIC508.7 [1]
2-(3-Hydroxyanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)butanediamideIC5055.0 [1]
5-Chloro-N-methoxy-N-methyl-2-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzamideIC50344.0 [1]
2-(4-Fluoroanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)acetamideIC50257.0 [1]
1-(4-Chloroanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)cyclopentane-1-carboxamideIC50217.0 [1]
2-(3-Methoxyanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)butanediamideIC50392.0 [1]
2-Anilino-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)acetamideIC50395.0 [1]
2-[4-Chloro-3-(methylcarbamoylamino)anilino]-2-methyl-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]propanamideIC5070.0 [1]
2-(3-Acetamido-4-chloroanilino)-2-methyl-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]propanamideIC5045.0 [1]
N-(3-Amino-3-oxopropyl)-3-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzamideIC5021.0 [1]
1-(4-Chloroanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)cyclopropane-1-carboxamideIC5044.0 [1]
1-(3-Hydroxyanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)cyclopropane-1-carboxamideIC5063.0 [1]
2-Fluoro-5-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzamideIC5012.0 [1]
2-Methyl-2-(3-sulfamoylanilino)-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]propanamideIC505.9 [1]
2-[4-Chloro-3-(2-oxo-1H-imidazol-3-yl)anilino]-2-methyl-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]propanamideIC50279.0 [1]
2-(3-Acetamido-4-chloroanilino)-2-methyl-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)propanamideIC5061.0 [1]
2-Chloro-5-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]-N-(3-sulfamoylpropyl)benzamideIC5030.0 [1]
2-(3-Acetamido-4-fluoroanilino)-2-methyl-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]propanamideIC5055.0 [1]
2-[4-Chloro-3-(methanesulfonamido)anilino]-2-methyl-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]propanamideIC5044.0 [1]
2-(3-Hydroxyanilino)-2-methyl-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)propanamideIC5033.0 [1]
2-(4-Chloro-3-hydroxyanilino)-2-methyl-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]propanamideIC5022.0 [1]
2-[4-Chloro-3-(propanoylamino)anilino]-2-methyl-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]propanamideIC50304.0 [1]
2-(3-Hydroxyanilino)-4-methyl-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)pentanamideIC50448.0 [1]
2-Fluoro-N-methyl-5-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzamideIC5012.0 [1]
N-(2-Amino-2-oxoethyl)-5-chloro-2-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzamideIC50386.0 [1]
2-[[2-Chloro-5-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzoyl]amino]acetic acidIC50134.0 [1]
2-(3-Fluoroanilino)-2-methyl-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]propanamideIC50371.0 [1]
2-Hydroxyethyl N-[2-chloro-5-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]phenyl]carbamateIC50105.0 [1]
N-(2-Amino-2-oxoethyl)-2-chloro-5-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzamideIC500.6 [1]
2-(4-Chloroanilino)-2-methyl-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)propanamideIC5080.0 [1]
1-[4-Fluoro-3-(propanoylamino)anilino]-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)cyclopropane-1-carboxamideIC50125.0 [1]
Methyl 3-[[2-oxo-2-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-ylamino)ethyl]amino]benzoateIC50477.0 [1]
1-(3-Acetamido-4-fluoroanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)cyclopropane-1-carboxamideIC50105.0 [1]
2-Chloro-5-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]-N-phenylmethoxybenzamideIC50128.0 [1]
2-Chloro-5-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzamideIC5023.0 [1]
2-(3-Acetamido-4-chloroanilino)-2-phenyl-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)acetamideIC50427.0 [1]
1-(4-Chloroanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)cyclobutane-1-carboxamideIC50174.0 [1]
2-(3,4-Difluoroanilino)-2-methyl-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]propanamideIC50180.0 [1]
2-Chloro-5-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzoic acidIC5099.0 [1]
4-[[3-[[2-Methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzoyl]amino]butanoic acidIC50160.0 [1]
3-[[2-Chloro-5-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzoyl]amino]propanoic acidIC5070.0 [1]
1-(4-Chlorophenyl)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)pyrrolidine-2-carboxamideIC50262.0 [1]
2-Chloro-N-ethyl-5-[[2-methyl-1-oxo-1-[[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]amino]propan-2-yl]amino]benzamideIC5016.0 [1]
2-[(6-Chloropyridin-3-yl)amino]-2-methyl-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]propanamideIC50277.0 [1]
Propan-2-yl 2-chloro-5-[[2-methyl-1-oxo-1-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-ylamino)propan-2-yl]amino]benzoateIC50343.0 [1]
Propan-2-yl 2-chloro-5-[[1-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-ylcarbamoyl)cyclopropyl]amino]benzoateIC50195.0 [1]
2-[3-(Methanesulfonamido)anilino]-2-methyl-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]propanamideIC50266.0 [1]
2-[4-Fluoro-3-(propanoylamino)anilino]-2-methyl-N-[4-(trifluoromethyl)-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl]propanamideIC50124.0 [1]
2-(3-Acetamidoanilino)-N-(6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)acetamideIC50153.0 [1]
1-(4-Chloroanilino)-N-(4-methyl-6H-pyrazolo[3,4-g][1,3]benzothiazol-2-yl)cyclopropane-1-carboxamideIC50185.0 [1]
6-(Benzimidazol-1-yl)-N-[5-[2-(dimethylamino)ethoxy]pyridin-2-yl]pyrimidin-4-amineIC503500.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ CDK3/Cyclin E Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/cdk3-cyclin-e-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ CDK3/Cyclin E Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cdk3-cyclin-e-inhibitors-ic50-ki.
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