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CDK4/Cyclin D3 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
RibociclibIC5013.0 [1]
Abemaciclib mesylateIC508.0 [1]
FascaplysinIC50100000.0 [1]
9H-Purine-2,6-diamine, N2-(2-aminocyclohexyl)-N6-(3-chlorophenyl)-9-ethyl-, cis-IC50573.0 [1]
8-Anilino-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC5010.0 [1]
8-Anilino-N,1-dimethyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC50160.0 [1]
1-Methyl-8-(4-morpholin-4-ylanilino)-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC50280.0 [1]
Ethyl 8-anilino-1-methyl-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxylateIC503240.0 [1]
1-Methyl-8-[4-(4-methylpiperazin-1-yl)anilino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC503.0 [1]
8-Anilino-1,4,4-trimethyl-5H-pyrazolo[4,3-h]quinazoline-3-carboxamideIC5010.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
6-N-(3-Amino-5-chlorophenyl)-2-N-[(3R)-piperidin-3-yl]-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
6-N-(3-Amino-5-chlorophenyl)-2-N-[(1R,2S)-2-aminocyclohexyl]-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
N-[3-[[2-[[(1R,2S)-2-Aminocyclohexyl]amino]-9-propan-2-ylpurin-6-yl]amino]-5-chlorophenyl]acetamideIC50611.0 [1]
6-N-(3-Amino-5-chlorophenyl)-2-N-[(1S,2S)-2-aminocyclohexyl]-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
6-N-(3-Amino-5-chlorophenyl)-2-N-[(1R,2R)-2-aminocyclohexyl]-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
N-[3-[[2-[[(1S,2R)-2-Aminocyclohexyl]amino]-9-propan-2-ylpurin-6-yl]amino]-5-chlorophenyl]acetamideIC501000.0 [1]
2-N-[(1S,2R)-2-Aminocyclohexyl]-6-N-(3-chlorophenyl)-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
2-N-[(1R,2R)-2-Aminocyclohexyl]-6-N-(3-chlorophenyl)-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
2-N-[(1S,2S)-2-Aminocyclohexyl]-6-N-(3-chlorophenyl)-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
6-N-(3-Amino-5-chlorophenyl)-2-N-[(1S,2R)-2-aminocyclohexyl]-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
2-N-[(1R,2S)-2-Aminocyclohexyl]-6-N-(3-chlorophenyl)-9-propan-2-ylpurine-2,6-diamineIC50541.0 [1]
6-N-(3-Amino-5-chlorophenyl)-9-propan-2-yl-2-N-[(3S)-pyrrolidin-3-yl]purine-2,6-diamineIC501000.0 [1]
6-N-(3-Amino-5-chlorophenyl)-2-N-[(3S)-piperidin-3-yl]-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
6-N-(3-Amino-5-chlorophenyl)-9-propan-2-yl-2-N-[(3R)-pyrrolidin-3-yl]purine-2,6-diamineIC501000.0 [1]
4-[3-(1h-Benzimidazol-2-Yl)-1h-Indazol-6-Yl]-3-EthylphenolKi4.4 [1]
4-[3-(1H-Benzimidazol-2-yl)-1H-indazol-6-yl]-3-methylphenolKi3.2 [1]
6-(2-Methoxy-4-hydroxyphenyl)-3-1H-benzoimidazol-2-yl-1H-indazoleKi17.0 [1]
3-Methoxy-4-[3-[4-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]-1H-indazol-6-yl]phenolKi98.0 [1]
3-1H-Benzoimidazol-2-yl-6-(3-hydroxyphenyl)-1H-indazoleKi200.0 [1]
Cdk9-IN-8IC50142.0 [1]
2-[(E)-2-(2,6-Dichlorophenyl)ethenyl]-5,7-dihydroxy-8-[(3S,4R)-3-hydroxy-1-methylpiperidin-4-yl]chromen-4-oneIC5022.5 [1]
N-[3-[[7-Cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]-N'-hydroxyoctanediamideIC5030.0 [1]
N-[4-[[7-Cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]-N'-hydroxyheptanediamideIC5010.0 [1]
Methyl 7-[[4-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]benzoyl]amino]heptanoateIC5011.0 [1]
7-Cyclopentyl-2-[[5-[4-[8-(hydroxyamino)-8-oxooctanoyl]piperazin-1-yl]pyridin-2-yl]amino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamideIC5013.0 [1]
N-[4-[(3-Cyclopentyltriazolo[4,5-d]pyrimidin-5-yl)amino]phenyl]-N'-hydroxyoctanediamideIC501140.0 [1]
Methyl 8-[2-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]anilino]-8-oxooctanoateIC505000.0 [1]
N-[4-[[7-Cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]-N',N'-dimethyloctanediamideIC5016.0 [1]
7-Cyclopentyl-2-[4-[[7-(hydroxyamino)-7-oxoheptyl]carbamoyl]anilino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamideIC5012.0 [1]
N-[4-[[7-Cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]-N'-hydroxyoctanediamideIC508.8 [1]
Methyl 8-[2-[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]hydrazinyl]-8-oxooctanoateIC505000.0 [1]
Methyl 8-[[4-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]methylamino]-8-oxooctanoateIC5025.0 [1]
7-Cyclopentyl-2-[4-(heptanoylamino)anilino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamideIC5027.0 [1]
Methyl 8-[4-[6-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]pyridin-3-yl]piperazin-1-yl]-8-oxooctanoateIC5013.0 [1]
7-Cyclopentyl-N,N-dimethyl-2-[4-(nonanoylamino)anilino]pyrrolo[2,3-d]pyrimidine-6-carboxamideIC50123.0 [1]
Methyl 8-[4-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]anilino]-8-oxooctanoateIC5012.0 [1]
Methyl 5-[[4-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]benzoyl]amino]pentanoateIC506.3 [1]
7-Cyclopentyl-2-[4-[[5-(hydroxyamino)-5-oxopentyl]carbamoyl]anilino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamideIC5011.0 [1]
Methyl 8-[4-[(9-cyclopentylpurin-2-yl)amino]anilino]-8-oxooctanoateIC505000.0 [1]
7-Cyclopentyl-2-[4-(8-hydroxyoctanoylamino)anilino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamideIC5010.0 [1]
Methyl 8-[3-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]anilino]-8-oxooctanoateIC5026.0 [1]
N-[4-[[7-Cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]-N'-hydroxyhexanediamideIC5011.0 [1]
N-[6-[[7-Cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]pyridin-3-yl]-N'-hydroxyoctanediamideIC5093.0 [1]
N-[3-[6-[(3-Bromophenyl)methylamino]purin-9-yl]cyclobutyl]-6-methylpyridine-2-carboxamideIC50611.0 [1]
7-Cyclopentyl-2-[4-[[6-(hydroxyamino)-6-oxohexyl]carbamoylamino]anilino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamideIC508.4 [1]
Methyl 8-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]-8-oxooctanoateIC505000.0 [1]
N-[2-[[7-Cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]-N'-hydroxyoctanediamideIC505000.0 [1]
Methyl 7-[4-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]anilino]-7-oxoheptanoateIC5010.0 [1]
N-[4-[(9-Cyclopentylpurin-2-yl)amino]phenyl]-N'-hydroxyoctanediamideIC505000.0 [1]
Methyl 6-[[4-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]benzoyl]amino]hexanoateIC507.3 [1]
Methyl 6-[[4-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]carbamoylamino]hexanoateIC5023.0 [1]
7-Cyclopentyl-2-[4-(hexanoylamino)anilino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamideIC5010.0 [1]
Methyl 8-[4-[(3-cyclopentyltriazolo[4,5-d]pyrimidin-5-yl)amino]anilino]-8-oxooctanoateIC50857.0 [1]
N-[[4-[[7-Cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]methyl]-N'-hydroxyoctanediamideIC5010.0 [1]
Methyl 8-[[4-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]benzoyl]amino]octanoateIC508.2 [1]
7-Cyclopentyl-2-[4-[[6-(hydroxyamino)-6-oxohexyl]carbamoyl]anilino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamideIC509.6 [1]
Methyl 9-[4-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]anilino]-9-oxononanoateIC5024.0 [1]
8-[4-[[7-Cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]anilino]-8-oxooctanoic acidIC5018.0 [1]
Methyl 8-[[5-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]pyridin-2-yl]amino]-8-oxooctanoateIC5016.0 [1]
N-[4-[[7-Cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]-N'-hydroxynonanediamideIC508.1 [1]
N-[3-[6-[(3-Chlorophenyl)methylamino]purin-9-yl]cyclobutyl]-6-methylpyridine-2-carboxamideIC501000.0 [1]
Methyl 6-[4-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]anilino]-6-oxohexanoateIC504.8 [1]
7-Cyclopentyl-N,N-dimethyl-2-[4-(octanoylamino)anilino]pyrrolo[2,3-d]pyrimidine-6-carboxamideIC5029.0 [1]
Methyl 8-[[6-[[7-cyclopentyl-6-(dimethylcarbamoyl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]pyridin-3-yl]amino]-8-oxooctanoateIC5047.0 [1]
7-Cyclopentyl-2-[4-[[8-(hydroxyamino)-8-oxooctyl]carbamoyl]anilino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamideIC5026.0 [1]
1-Methyl-8-(3-piperazin-1-ylanilino)-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC505620.0 [1]
8-[4-(Dimethylamino)anilino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC5034.0 [1]
8-[[5-(Dimethylamino)pyridin-2-yl]amino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC50680.0 [1]
1-Methyl-8-[(5-morpholin-4-ylpyridin-2-yl)amino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC5030.0 [1]
1-Methyl-8-(3-morpholin-4-ylanilino)-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC503650.0 [1]
1-Methyl-8-(4-methylanilino)-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC50250.0 [1]
8-[[4-(Dimethylamino)pyridin-2-yl]amino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC505700.0 [1]
1-Methyl-8-[(5-piperazin-1-ylpyridin-2-yl)amino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC5029.0 [1]
8-[3-(Dimethylamino)anilino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC501850.0 [1]
Ethyl 8-anilino-1,4-dimethyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxylateIC5010000.0 [1]
1-Methyl-8-[[5-(4-methylpiperazin-1-yl)pyridin-2-yl]amino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC5010.0 [1]
1-Methyl-8-(4-piperazin-1-ylanilino)-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC508.0 [1]
8-(4-Chloroanilino)-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC5060.0 [1]
8-Anilino-N-ethyl-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC50450.0 [1]
8-Anilino-1,4-dimethyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC505260.0 [1]
Ethyl 8-anilino-1,4,4-trimethyl-5H-pyrazolo[4,3-h]quinazoline-3-carboxylateIC501000.0 [1]
N2-[(1R,2S)-2-Aminocyclohexyl]-N6-(3-chlorophenyl)-9-ethyl-9H-purine-2,6-diamineIC501000.0 [1]
8-Anilino-N,1,4,4-tetramethyl-5H-pyrazolo[4,3-h]quinazoline-3-carboxamideIC50450.0 [1]
2-N-[(1S,2S)-2-Aminocyclohexyl]-6-N-(3-chlorophenyl)-9-ethylpurine-2,6-diamineIC501000.0 [1]
2-[6-(4-Hydroxy-2-methoxyphenyl)-1H-indazol-3-yl]-N-(2-morpholin-4-ylethyl)-3H-benzimidazole-5-carboxamideKi48.0 [1]
4-[3-[4-(2-Hydroxyethylsulfanyl)-1H-benzimidazol-2-yl]-1H-indazol-6-yl]-3-methoxyphenolKi1000.0 [1]
4-[3-[(E)-2-(3,4-Dimethoxyphenyl)ethenyl]-1H-indazol-6-yl]-2-methoxyphenolKi13.0 [1]
2-Methoxy-4-[3-(3,4,5-trimethoxyphenyl)-1H-indazol-6-yl]phenolKi26000.0 [1]
3-Methoxy-4-[3-[6-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]-1H-indazol-6-yl]phenolKi15.5 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ CDK4/Cyclin D3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/cdk4-cyclin-d3-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ CDK4/Cyclin D3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cdk4-cyclin-d3-inhibitors-ic50-ki.
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