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CDK6/cyclin D1 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
AbemaciclibIC5010.0 [1]
AbemaciclibKi10.0 [1]
N-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-4-(thieno[2,3-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamideIC504.24 [1], 10.0 [2]
StaurosporineIC502.9 [1]
SeliciclibIC5023500.0 [1]
PalbociclibIC503.76 [1]
FascaplysinIC503400.0 [1]
(2S,3S)-3-((7-(Benzylamino)-3-isopropylpyrazolo[1,5-a]pyrimidin-5-yl)amino)butane-1,2,4-triolIC5035500.0 [1]
CID 56649281IC509.82 [1]
N'-(Pyrrolidino[2,1-B]isoindolin-4-ON-8-YL)-N-(pyridin-2-YL)ureaIC5071.0 [1]
2-Bromo-N-(2,5-dichlorothiophen-3-yl)sulfonyl-N-phenylacetamideIC5034900.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
4-Methyl-N-[3-(trifluoromethyl)phenyl]benzenesulfonamideIC50208800.0 [1]
2-[(E)-2-(2,6-Dichlorophenyl)ethenyl]-5,7-dihydroxy-8-[(3S,4R)-3-hydroxy-1-methylpiperidin-4-yl]chromen-4-oneIC5045.0 [1]
2,4,5-Trichloro-N-[3-(trifluoromethyl)phenyl]benzenesulfonamideIC5058800.0 [1]
N-(6-Methoxyquinolin-8-yl)-N',N'-bis(3-methylbutyl)propane-1,3-diamineIC50325000.0 [1]
(2S)-2-[Bis(2-methylpropyl)amino]-1-[(6-methoxy-2-methylquinolin-8-yl)amino]propan-2-olIC50691000.0 [1]
5-N-(2-Aminocyclohexyl)-7-N-benzyl-3-propan-2-yl-2H-pyrazolo[4,3-d]pyrimidine-5,7-diamineIC50100000.0 [1]
CID 49798457IC50110400.0 [1]
2,5-Dichloro-N-p-tolylthiophene-3-sulfonamideIC5051300.0 [1]
2,5-Dichloro-N-(4-methylphenyl)-N-(trichloromethylsulfanyl)thiophene-3-sulfonamideIC5018000.0 [1]
5-N-(4-Aminocyclohexyl)-7-N-benzyl-3-propan-2-yl-2H-pyrazolo[4,3-d]pyrimidine-5,7-diamineIC5091000.0 [1]
N-[(4-Methoxyphenyl)methyl]-[1]benzofuro[2,3-b]pyridin-4-amineIC50129000.0 [1]
4-Phenyl-[1]benzofuro[2,3-b]pyridine-3,6-diolKi773000.0 [1]
4-{[4-Amino-5-(2-Nitrobenzoyl)-1,3-Thiazol-2-Yl]amino}benzenesulfonamideIC506.6 [1]
N-[4-(Morpholin-4-ylmethyl)phenyl]-4-(thieno[2,3-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamideIC503.88 [1]
4-(Furo[2,3-d]pyrimidin-4-ylamino)-N-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]-1H-pyrazole-5-carboxamideIC505.09 [1]
CID 72195175IC501.96 [1]
N-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-4-(thieno[3,2-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamideIC504.11 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ CDK6/cyclin D1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.8 May2024https://www.aatbio.com/data-sets/cdk6-cyclin-d1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 8). Quest Database™ CDK6/cyclin D1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cdk6-cyclin-d1-inhibitors-ic50-ki.
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