 | Abemaciclib | IC50 | 3112.0 [1] |
| Abemaciclib | Ki | 3910.0 [1] |
 | 1-[4-[4-[[5-(Oxan-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]cyclohexyl]piperazin-1-yl]ethanone | IC50 | 516.0 [1], 30000.0 [2] |
 | 1-[4-[4-[(5-Propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]cyclohexyl]piperazin-1-yl]ethanone | IC50 | 2310.0 [1], 30000.0 [2] |
 | Staurosporine | IC50 | 120.0 [1] |
 | Alvocidib | IC50 | 514.0 [1] |
 | Dinaciclib | IC50 | 170.0 [1] |
 | Sns-032 | IC50 | 62.0 [1] |
 | 4-(2,6-Dichlorobenzamido)-N-(piperidin-4-yl)-1H-pyrazole-3-carboxamide | Ki | 2800.0 [1] |
 | (16E)-14-Methyl-20-oxa-5,7,14,27-tetrazatetracyclo[19.3.1.12,6.18,12]heptacosa-1(25),2(27),3,5,8,10,12(26),16,21,23-decaene | IC50 | 3.0 [1] |
 | BS-181 | IC50 | 134.0 [1] |
 | CID 23643976 | IC50 | 2870.0 [1] |
 | (3-((6-(2-Methoxyphenyl)pyrimidin-4-yl)amino)phenyl)methanesulfonamide | IC50 | 20000.0 [1] |
 | CID 78357764 | IC50 | 246.0 [1] |
 | CDK12 inhibitor 2 | IC50 | 10000.0 [1] |
 | 4-[[[4-[5-Chloro-2-[[4-(2-methoxyethylamino)cyclohexyl]amino]pyridin-4-yl]-1,3-thiazol-2-yl]amino]methyl]oxane-4-carbonitrile | IC50 | 1720.0 [1] |
 | 2-Anilino-7-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5,5-dimethylpyrrolo[2,3-d]pyrimidin-6-one | IC50 | 793.0 [1] |
 | 1-[4-[4-Amino-3-[4-(2-morpholin-4-ylethoxy)phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]phenyl]-3-(5-tert-butyl-1,2-oxazol-3-yl)urea | IC50 | 10000.0 [1] |
 | (2S,3R)-3-[2-[4-(Cyclopropylsulfonimidoyl)anilino]-5-(trifluoromethyl)pyrimidin-4-yl]oxybutan-2-ol | IC50 | 25.0 [1] |
 | 2-[5-[[[2-[(4-Aminocyclohexyl)amino]-9-cyclopentylpurin-6-yl]amino]methyl]pyridin-2-yl]phenol | IC50 | 306.0 [1] |
 | 2-[3-[3-(1H-Pyrrolo[2,3-b]pyridin-3-yl)propyl]triazol-4-yl]-1H-pyrrolo[2,3-b]pyridine | IC50 | 50000.0 [1] |
 | N-[3-[6-[(3-Bromophenyl)methylamino]purin-9-yl]cyclobutyl]-6-methylpyridine-2-carboxamide | IC50 | 359.0 [1] |
 | N-[3-[6-[(3-Chlorophenyl)methylamino]purin-9-yl]cyclobutyl]-6-methylpyridine-2-carboxamide | IC50 | 319.0 [1] |
 | 3-Benzyl-1-[4-[(5-cyanopyridin-2-yl)amino]cyclohexyl]-1-[4-(1-methylpyrazol-4-yl)phenyl]urea | IC50 | 10000.0 [1] |
 | 6-[[1-[4-(1-Methylpyrazol-4-yl)phenyl]sulfonylpiperidin-4-yl]amino]pyridine-3-carbonitrile | IC50 | 10000.0 [1] |
 | [(2S,3S,4S,5R)-5-(6-Bromo-5-carbamoyl-4-imino-7H-pyrrolo[2,3-d]pyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl 2-methylpropanoate | IC50 | 1200.0 [1] |
 | N-[1-[4-(4-Fluoroanilino)pyrimidin-2-yl]piperidin-4-yl]-4-methoxybenzamide | IC50 | 89.8 [1] |
 | 5-N-(2-Aminocyclohexyl)-7-N-benzyl-3-propan-2-yl-2H-pyrazolo[4,3-d]pyrimidine-5,7-diamine | IC50 | 100000.0 [1] |
 | 5-N-(4-Aminocyclohexyl)-7-N-benzyl-3-propan-2-yl-2H-pyrazolo[4,3-d]pyrimidine-5,7-diamine | IC50 | 100000.0 [1] |
 | 6-(Benzimidazol-1-yl)-N-[5-[2-(dimethylamino)ethoxy]pyridin-2-yl]pyrimidin-4-amine | IC50 | 1100.0 [1] |
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