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CDK8/Cyclin C Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
StaurosporineIC506.0 [1], 15.0 [2]
Senexin BIC5024.0 [1]
[5-Amino-8-[4-(1-methylpyrazol-4-yl)phenyl]-1,6-naphthyridin-2-yl]-(3-methoxyazetidin-1-yl)methanoneIC501.1 [1], 5.1 [2]
3-Chloranyl-4-Pyridin-4-Yl-1h-Pyrrole-2-CarboxamideIC505.0 [1], 7.0 [2]
[1-Amino-4-[4-(1-methylpyrazol-4-yl)phenyl]isoquinolin-6-yl]-(3-methoxyazetidin-1-yl)methanoneIC5012.0 [1], 32.7 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseCDK8/Cyclin C Inhibitors (IC50, Ki)." AAT Bioquest, Inc.14 Dec2025https://www.aatbio.com/data-sets/cdk8-cyclin-c-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 14). Quest DatabaseCDK8/Cyclin C Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cdk8-cyclin-c-inhibitors-ic50-ki.
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