Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Staurosporine | IC50 | 6.0 [1], 15.0 [2] | |
| Senexin B | IC50 | 24.0 [1] | |
| [5-Amino-8-[4-(1-methylpyrazol-4-yl)phenyl]-1,6-naphthyridin-2-yl]-(3-methoxyazetidin-1-yl)methanone | IC50 | 1.1 [1], 5.1 [2] | |
| 3-Chloranyl-4-Pyridin-4-Yl-1h-Pyrrole-2-Carboxamide | IC50 | 5.0 [1], 7.0 [2] | |
| [1-Amino-4-[4-(1-methylpyrazol-4-yl)phenyl]isoquinolin-6-yl]-(3-methoxyazetidin-1-yl)methanone | IC50 | 12.0 [1], 32.7 [2] | |
MLA | "Quest Database™ CDK8/Cyclin C Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 14 Dec. 2025, https://www.aatbio.com/data-sets/cdk8-cyclin-c-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 14). Quest Database™ CDK8/Cyclin C Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cdk8-cyclin-c-inhibitors-ic50-ki. | |
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