 | Seliciclib | IC50 | 800.0 [1] |
| Seliciclib | Ki | 790.0 [1] |
 | Alvocidib | IC50 | 4.59 [1] |
| Alvocidib | Ki | 3.0 [1] |
 | Dinaciclib | IC50 | 4.0 [1], 178.0 [2] |
 | 4-[(E)-(3,5-Diamino-1h-Pyrazol-4-Yl)diazenyl]phenol | IC50 | 150.0 [1], 350.0 [2] |
| 4-[(E)-(3,5-Diamino-1h-Pyrazol-4-Yl)diazenyl]phenol | Ki | 350.0 [1] |
 | Staurosporine | IC50 | 3.3 [1], 14.0 [2] |
| Staurosporine | Ki | 7.0 [1] |
 | Abemaciclib | IC50 | 57.0 [1], 101.0 [2] |
| Abemaciclib | Ki | 57.0 [1] |
 | Sns-032 | IC50 | 4.0 [1], 40.0 [2] |
 | 4-(2,6-Dichlorobenzamido)-N-(piperidin-4-yl)-1H-pyrazole-3-carboxamide | IC50 | 10.0 [1] |
| 4-(2,6-Dichlorobenzamido)-N-(piperidin-4-yl)-1H-pyrazole-3-carboxamide | Ki | 100.0 [1] |
 | (3-((6-(2-Methoxyphenyl)pyrimidin-4-yl)amino)phenyl)methanesulfonamide | IC50 | 44.0 [1], 230.0 [2] |
 | 4-(4-Methoxy-1h-Pyrrolo[2,3-B]pyridin-3-Yl)pyrimidin-2-Amine | IC50 | 6.0 [1] |
 | 4-(1H-Pyrrolo[2,3-B]pyridin-3-YL)pyrimidin-2-amine | IC50 | 26.0 [1], 30.0 [2] |
 | Ribociclib | IC50 | 197.0 [1] |
 | Rohitukine | IC50 | 300.0 [1] |
 | CID 23643976 | IC50 | 20.0 [1] |
 | Leucettine L41 | IC50 | 10000.0 [1], 18000.0 [2] |
 | (2R)-2-{[4-(Benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-ol | IC50 | 43.0 [1] |
 | 3-[[5-Cyano-4-[4-Methyl-2-(Methylamino)-1,3-Thiazol-5-Yl]pyrimidin-2-Yl]amino]benzenesulfonamide | Ki | 6.0 [1] |
 | [4-(2-Amino-4-methyl-thiazol-5-YL)-pyrimidin-2-YL]-(3-nitro-phenyl)-amine | Ki | 4.0 [1] |
 | [3-[[6-(2-Benzyloxyphenyl)pyrimidin-4-yl]amino]phenyl]methyl-propyl-phosphinic acid | IC50 | 142.0 [1] |
 | 4-(4-Propoxy-1h-Pyrrolo[2,3-B]pyridin-3-Yl)pyrimidin-2-Amine | IC50 | 5.6 [1], 6.0 [2] |
 | Meriolin 9 | IC50 | 10000.0 [1] |
 | Meriolin 2 | IC50 | 18.0 [1] |
 | 4-[4-Methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-[3-(morpholine-4-carbonyl)anilino]pyrimidine-5-carbonitrile | Ki | 43.0 [1] |
 | 4-(4-Methyl-2-(methylamino)thiazol-5-yl)-2-(3-nitrophenylamino)pyrimidine-5-carbonitrile | Ki | 6.0 [1] |
 | 2-[3-(1,4-Diazepan-1-yl)anilino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Ki | 7.0 [1] |
 | N-Methyl-5-[2-(3-nitroanilino)pyrimidin-4-yl]-4-phenyl-1,3-thiazol-2-amine | Ki | 5000.0 [1], 9835.0 [2] |
 | 1-[4-[4-[[5-(Oxan-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]cyclohexyl]piperazin-1-yl]ethanone | IC50 | 1890.0 [1], 30000.0 [2] |
 | 3-Benzyl-1-[4-[(5-cyanopyridin-2-yl)amino]cyclohexyl]-1-[4-(1-methylpyrazol-4-yl)phenyl]urea | IC50 | 30000.0 [1] |
 | 1-[4-[4-[(5-Propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]cyclohexyl]piperazin-1-yl]ethanone | IC50 | 890.0 [1], 30000.0 [2] |
 | Harmine | IC50 | 720.0 [1] |
 | 5,6-Dichloro-1-beta-D-ribofuranosylbenzimidazole | Ki | 340.0 [1] |
 | Palbociclib | Ki | 364.0 [1] |
 | Doramapimod | IC50 | 30000.0 [1] |
 | Indirubin-3'-monoxime | IC50 | 2400.0 [1] |
 | Kenpaullone | IC50 | 64.0 [1] |
 | Fascaplysin | IC50 | 250000.0 [1] |
 | N3-(4-Fluorophenyl)-1h-pyrazolo[3,4-d]pyrimidine-3,4-diamine | Ki | 10000.0 [1] |
 | Pik-75 | IC50 | 1.37 [1] |
 | O6-Cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | IC50 | 1070.0 [1] |
 | Paullone | IC50 | 810.0 [1] |
 | Cercosporamide | IC50 | 220.0 [1] |
 | Olomoucine II | IC50 | 815.0 [1] |
 | 4-Methyl-5-(2-((4-morpholinophenyl)amino)-pyrimidin-4-yl)thiazol-2-amine | Ki | 480.0 [1] |
 | Pha-793887 | IC50 | 138.0 [1] |
 | BS-181 | IC50 | 1790.0 [1] |
 | 3-(2-Aminopyrimidin-4-yl)-1H-indol-4-ol | IC50 | 2400.0 [1] |
 | RGB-286638 free base | IC50 | 1.0 [1] |
 | Voruciclib | IC50 | 22.0 [1] |
 | (2S,3S)-3-((7-(Benzylamino)-3-isopropylpyrazolo[1,5-a]pyrimidin-5-yl)amino)butane-1,2,4-triol | IC50 | 90.0 [1] |
 | Leucettamine B | IC50 | 10000.0 [1] |
 | CID 71561915 | Ki | 4.0 [1] |
 | CID 78357764 | IC50 | 11.0 [1] |
 | 3,5-Diamino-4-phenylazopyrazole | IC50 | 15000.0 [1] |
 | N-[2-(1H-Indol-3-yl)ethyl]-N-methyl-4-phenylbenzamide | IC50 | 1000000.0 [1] |
 | 5-(2-Aminopyrimidin-4-yl)-2-phenyl-1H-pyrrole-3-carboxamide | IC50 | 394.0 [1] |
 | Cyc065 | IC50 | 26.0 [1] |
 | Cyclapolin 9 | IC50 | 100000.0 [1] |
 | 4-[4-Methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-(4-methyl-3-morpholin-4-ylsulfonylanilino)pyrimidine-5-carbonitrile | Ki | 22.0 [1] |
 | Ethyl 4-[(4-fluorophenyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxylate | Ki | 10000.0 [1] |
 | (2~{R},3~{S})-3-[[9-Propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-ol | IC50 | 110.0 [1] |
 | (2-Methyl-4,5-dihydro-thiazolo[4,5-h]quinazolin-8-yl)-(3-nitro-phenyl)-amine | Ki | 2.0 [1] |
 | 2(3H)-Thiazolone, 3,4-diMethyl-5-[2-[[4-(1-piperazinyl)phenyl]aMino]-4-pyriMidinyl]- | Ki | 0.4 [1] |
 | N-(2-(1H-Indol-3-yl)ethyl)-4-chloro-N-methylbenzamide | IC50 | 1000000.0 [1] |
 | N-(2-(1H-Indol-3-yl)ethyl)-4-tert-butyl-N-methylbenzamide | IC50 | 1000000.0 [1] |
 | N-[5-[[6-(3-Aminophenyl)pyrimidin-4-yl]amino]-2-methyl-phenyl]methanesulfonamide | IC50 | 129.0 [1] |
 | CDK12 inhibitor 2 | IC50 | 16000.0 [1] |
 | 2-N-(4-Aminocyclohexyl)-8-propan-2-yl-4-N-[(4-pyridin-2-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazine-2,4-diamine | IC50 | 49.0 [1] |
 | 4-[[[4-[5-Chloro-2-[[4-(2-methoxyethylamino)cyclohexyl]amino]pyridin-4-yl]-1,3-thiazol-2-yl]amino]methyl]oxane-4-carbonitrile | IC50 | 1.0 [1] |
 | (4Z)-2-[4-[2-[2-[2-(2-Aminoethoxy)ethoxy]ethoxy]ethoxy]anilino]-4-(1,3-benzodioxol-5-ylmethylidene)-1H-imidazol-5-one | IC50 | 3700.0 [1] |
 | 2-(2-Fluorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydroxy-1-methylpiperidin-4-yl]chromen-4-one | IC50 | 2.8 [1] |
 | 5,7-Dihydroxy-8-[(3S,4R)-3-hydroxy-1-methylpiperidin-4-yl]-2-phenylchromen-4-one | IC50 | 9.0 [1] |
 | 2-(4-Fluorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydroxy-1-methylpiperidin-4-yl]chromen-4-one | IC50 | 2.1 [1] |
 | 2-(4-Bromophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydroxy-1-methylpiperidin-4-yl]chromen-4-one | IC50 | 5.5 [1] |
 | 5,7-Dihydroxy-8-[(3S,4R)-3-hydroxy-1-methylpiperidin-4-yl]-2-[4-(trifluoromethyl)phenyl]chromen-4-one | IC50 | 19.0 [1] |
 | 5,7-Dihydroxy-8-[(3S,4R)-3-hydroxy-1-methylpiperidin-4-yl]-2-(4-hydroxyphenyl)chromen-4-one | IC50 | 9.6 [1] |
 | 5,7-Dihydroxy-8-[(3S,4R)-3-hydroxy-1-methylpiperidin-4-yl]-2-pyridin-4-ylchromen-4-one | IC50 | 6.5 [1] |
 | 2-(4-Ethenylphenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydroxy-1-methylpiperidin-4-yl]chromen-4-one | IC50 | 9.5 [1] |
 | (2r)-2-{[7-(Benzylamino)-3-(Propan-2-Yl)-1h-Pyrazolo[4,3-D]pyrimidin-5-Yl]amino}butan-1-Ol | IC50 | 1000.0 [1] |
 | (Arylindolyl)maleimide deriv. 27 | IC50 | 80.0 [1] |
 | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
 | 3-[[6-(2-Methoxyphenyl)pyrimidin-4-yl]amino]benzenesulfonamide | IC50 | 52.0 [1] |
 | 2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 30 | Ki | 2.0 [1] |
 | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
 | N-[5-[[6-(2-Methoxyphenyl)pyrimidin-4-yl]amino]-2-methylphenyl]methanesulfonamide | IC50 | 30.0 [1] |
 | 2-Anilino-7-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5,5-dimethylpyrrolo[2,3-d]pyrimidin-6-one | IC50 | 1582.0 [1] |
 | 2-[3-(4-Acetyl-1,4-diazepan-1-yl)anilino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Ki | 7.0 [1] |
 | CID 76072859 | IC50 | 749.0 [1] |
 | CID 86579886 | IC50 | 360.0 [1] |
 | 6-(2-Methoxyphenyl)-N-[4-[propan-2-yloxy(propyl)phosphoryl]oxyphenyl]pyrimidin-4-amine | IC50 | 407.0 [1] |
 | CID 86579888 | IC50 | 2840.0 [1] |
 | CID 86579889 | IC50 | 10000.0 [1] |
 | 6-(3-Nitrophenyl)-N-[4-[propan-2-yloxy(propyl)phosphoryl]oxyphenyl]pyrimidin-4-amine | IC50 | 10000.0 [1] |
 | CID 86579891 | IC50 | 3840.0 [1] |
 | 6-(3-Aminophenyl)-N-[4-[propan-2-yloxy(propyl)phosphoryl]oxyphenyl]pyrimidin-4-amine | IC50 | 6060.0 [1] |
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