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Cell division control protein 42 homolog Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
FasudilIC505000.0 [1], 8000.0 [2]
Y-27632 DihydrochlorideIC508000.0 [1]
Chelerythrine chlorideIC50100000.0 [1]
Sanguinarium ChlorideIC5032000.0 [1]
DemethyleneberberineIC50100000.0 [1]
Secramine AIC509000.0 [1]
Secramine BIC507000.0 [1]
N-(7-Chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-(dimethylamino)-2-phenylacetamideIC508000.0 [1]
N-(7-Chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-(cyclopropylamino)-2-phenylacetamideIC508000.0 [1]
N-(7-Chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-(methylamino)-2-phenylacetamideIC501300.0 [1]
(3S,4R)-N-(7-Chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-4-(4-chlorophenyl)pyrrolidine-3-carboxamideIC5054.0 [1]
2-Amino-N-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-phenylacetamideIC501700.0 [1]
[(2S,3R,4S,5S)-5-(2-Amino-6-oxo-1H-purin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl phosphono hydrogen phosphateIC501400.0 [1]
N-(7-Chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-phenylacetamideIC505400.0 [1]
N-[3-(4-Dimethylaminomethyl-phenylcarbamoyl)-benzyl]-3,4-dimethoxy-benzamideIC505000.0 [1]
3-Chloro-N-[3-(4-dimethylaminomethyl-phenylcarbamoyl)-benzyl]-4-methoxy-benzamideIC505000.0 [1]
3,4-Dimethoxy-N-[3-(3-piperidin-3-yl-propionylamino)-benzyl]-benzamideIC505000.0 [1]
3-[3-(4-Cyano-phenyl)-ureidomethyl]-N-(1,2,3,4-tetrahydro-isoquinolin-7-yl)-benzamideIC505000.0 [1]
3-[3-(4-Cyano-phenyl)-ureidomethyl]-N-(2-piperidin-3-yl-ethyl)-benzamideIC505000.0 [1]
3-[3-(3-Cyano-phenyl)-ureidomethyl]-N-(2-piperidin-3-yl-ethyl)-benzamideIC505000.0 [1]
3-[3-(4-Cyano-phenyl)-ureidomethyl]-N-(4-dimethylaminomethylphenyl)-benzamideIC505000.0 [1]
3,4-Dimethoxy-N-[3-(2-piperidin-3-yl-ethylcarbamoyl)-benzyl]-benzamideIC505000.0 [1]
3,4-Dimethoxy-N-[3-(1,2,3,4-tetrahydro-isoquinolin-7-ylcarbamoyl)-benzyl]-benzamideIC505000.0 [1]
3,4-Dimethoxy-N-[3-(2-piperidin-4-yl-ethylcarbamoyl)-benzyl]-benzamideIC505000.0 [1]
3,4-Dimethoxy-N-[3-(2-methyl-1,2,3,4-tetrahydro-isoquinolin-7-ylcarbamoyl)-benzyl]-benzamideIC505000.0 [1]
3-[[(4-Carbamoylphenyl)carbamoylamino]methyl]-N-(1,2,3,4-tetrahydroisoquinolin-7-yl)benzamideIC505000.0 [1]
6,8,13,13a-Tetrahydro-5H-isoquinolino[2,1-b]isoquinoline-2,3,9,10-tetrol;hydrochlorideIC50100000.0 [1]
6,7-Dimethoxy-1-methyl-3-naphthalen-2-ylisoquinoline;hydrochlorideIC50100000.0 [1]
2-(Benzylamino)-N-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)acetamideIC508000.0 [1]
3-(Tert-butylamino)-4-[[2-(4-pyridin-4-ylanilino)pyrimidin-4-yl]amino]cyclobut-3-ene-1,2-dioneKi4400.0 [1]
5,6-Dihydroisoquinolino[2,1-b]isoquinolin-7-ium-2,3,9,10-tetrol;chlorideIC506000.0 [1]
3-(3,4-Dihydroxy-phenyl)-6,7-dimethoxy-1-methyl-isoquinolinium chlorideIC50100000.0 [1]
5-Methylbenzo[c]phenanthridin-5-ium-2,3,7,8-tetrolIC5022000.0 [1]
7,8-Dimethoxy-5-methylbenzo[c]phenanthridin-5-ium-2,3-diolIC5073000.0 [1]
8-Methylisoquinolino[2,1-b]isoquinolin-7-ium-3,4,10,11-tetrolIC5026000.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Cell division control protein 42 homolog Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/cell-division-control-protein-42-homolog-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Cell division control protein 42 homolog Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cell-division-control-protein-42-homolog-inhibitors-ic50-ki.
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