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Cholecystokinin B receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
N-[(3R)-2,3-Dihydro-1-methyl-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-yl]-N'-(3-methylphenyl)ureaIC504.0 [1]
N-[(3R)-2,3-Dihydro-1-methyl-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-yl]-N'-(3-methylphenyl)ureaKi1.58 [1], 1.8 [2], 2.95 [3]
SincalideKi0.28 [1], 0.3 [2], 0.64 [3], 0.65 [4]
DevazepideIC50245.0 [1]
DevazepideKi3.69 [1], 29.51 [2], 51.29 [3], 62.0 [4], 87.1 [5]

References
This online resource may be cited as follows
MLA
"Quest DatabaseCholecystokinin B receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.13 Dec2025https://www.aatbio.com/data-sets/cholecystokinin-b-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 13). Quest DatabaseCholecystokinin B receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cholecystokinin-b-receptor-inhibitors-ic50-ki.
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