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Cholesteryl ester transfer protein Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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1,1,1-Trifluoro-3-((3-phenoxyphenyl)(3-(1,1,2,2-tetrafluoroethoxy)benzyl)amino)propan-2-olIC50200.0 [1]
(2R)-1,1,1-Trifluoro-3-[3-phenoxy-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]propan-2-olIC5036.0 [1]
TorcetrapibIC5018.0 [1]
AnacetrapibIC5033.8 [1]
3-[3-(4-Chloro-3-ethylphenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]-1,1,1-trifluoropropan-2-olIC5030.0 [1]
1-[(1S)-1-(5-Chloropyridin-2-yl)-1-[3-fluoro-5-(1,1,2,2-tetrafluoroethoxy)phenyl]-2-phenylethyl]-3-cyclopentylureaIC507.0 [1]
1-[(1S)-1-(5-Chloropyridin-2-yl)-1-[3-fluoro-5-(trifluoromethyl)phenyl]-2-phenylethyl]-3-cyclopentylureaIC5020.0 [1]
1-[(1R)-1-(5-Chloropyridin-2-yl)-1-[3-fluoro-5-(trifluoromethyl)phenyl]-2-phenylethyl]-3-cyclopentylureaIC501200.0 [1]
1,1,1-Trifluoro-3-[(3-phenoxyphenyl)(3-ethoxybenzyl)amino]-2-propanolIC501600.0 [1], 6000.0 [2], 70000.0 [3]
1,1,1-Trifluoro-3-((3-phenoxyphenyl)(3-(trifluoromethoxy)benzyl)amino)propan-2-olIC501000.0 [1], 40000.0 [2]
1,1,1-Trifluoro-3-((3-fluorophenyl)(3-(trifluoromethyl)benzyl)amino)propan-2-olIC5040000.0 [1], 200000.0 [2]
(2R)-3-[3-(4-Chloro-3-ethylphenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]-1,1,1-trifluoropropan-2-olIC500.77 [1], 73.0 [2], 80.0 [3], 3000.0 [4], 59000.0 [5]
1,1,1-Trifluoro-3-(phenyl(3-(trifluoromethyl)benzyl)amino)propan-2-olIC5015000.0 [1], 200000.0 [2]
1,1,1-Trifluoro-3-((3-fluorophenyl)(3-(trifluoromethoxy)benzyl)amino)propan-2-olIC5012000.0 [1], 12022.64 [2], 200000.0 [3]
1,1,1-Trifluoro-3-[(3-phenoxyphenyl)[3-(2-furanyl)benzyl]amino]-2-propanolIC50480.0 [1], 52000.0 [2]
1,1,1-Trifluoro-3-[N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]-3-(5,6,7,8-tetrahydronaphthalen-2-yloxy)anilino]propan-2-olIC5090.0 [1], 5200.0 [2], 90011.91 [3]
3-[3-(3-Tert-butylphenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]-1,1,1-trifluoropropan-2-olIC5080.0 [1], 100.0 [2], 3800.0 [3], 80001.84 [4]
1,1,1-Trifluoro-3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(m-tolyloxy)phenyl)amino)propan-2-olIC5090.0 [1], 13300.0 [2], 90011.91 [3]
3-[(3-Phenoxyphenyl)[4-(trifluoromethoxy)benzyl]amino]-1,1,1-trifluoropropane-2-olIC503500.0 [1], 4000.0 [2], 120000.0 [3]
1,1,1-Trifluoro-3-[3-(3-methoxyphenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]propan-2-olIC501000.0 [1], 15600.0 [2], 1000000.0 [3]
3-[3-(3,4-Dimethylphenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]-1,1,1-trifluoropropan-2-olIC5080.0 [1], 6500.0 [2], 80001.84 [3]
1,1,1-Trifluoro-3-[N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]-3-[4-(trifluoromethyl)phenoxy]anilino]propan-2-olIC50100.0 [1], 6900.0 [2], 100000.0 [3]
1,1,1-Trifluoro-3-[3-(3-fluoro-2-nitrophenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]propan-2-olIC50100.0 [1], 5600.0 [2], 100000.0 [3]
1,1,1-Trifluoro-3-[N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]-3-[4-(trifluoromethoxy)phenoxy]anilino]propan-2-olIC50400.0 [1], 30100.0 [2], 400036.85 [3]
1,1,1-Trifluoro-3-[3-(4-propoxyphenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]propan-2-olIC5080.0 [1], 400.0 [2], 34200.0 [3], 400036.85 [4]
3-[3-(3-Ethyl-5-methylphenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]-1,1,1-trifluoropropan-2-olIC5080.0 [1], 3400.0 [2], 80001.84 [3]
3-((3-(1,1,2,2-Tetrafluoroethoxy)benzyl)(3-(4-aminophenoxy)phenyl)amino)-1,1,1-trifluoropropan-2-olIC50700.0 [1], 707.95 [2], 9000.0 [3], 700003.16 [4]
1,1,1-Trifluoro-3-((3-(4-nitrophenoxy)phenyl)(3-(1,1,2,2-tetrafluoroethoxy)benzyl)amino)propan-2-olIC50500.0 [1], 29300.0 [2], 500034.53 [3]
1,1,1-Trifluoro-3-[3-(4-fluoro-3-methylphenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]propan-2-olIC5080.0 [1], 3100.0 [2], 80001.84 [3]
1,1,1-Trifluoro-3-((3-(3-fluorophenoxy)phenyl)(3-(1,1,2,2-tetrafluoroethoxy)benzyl)amino)propan-2-olIC50300.0 [1], 9700.0 [2], 299985.32 [3]
3-((3-(1,1,2,2-Tetrafluoroethoxy)benzyl)(3-(4-chlorophenoxy)phenyl)amino)-1,1,1-trifluoropropan-2-olIC50300.0 [1], 10000.0 [2], 299985.32 [3]
3-[3-(3,5-Difluorophenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]-1,1,1-trifluoropropan-2-olIC50200.0 [1], 11500.0 [2], 200032.24 [3]
1,1,1-Trifluoro-3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(p-tolyloxy)phenyl)amino)propan-2-olIC50100.0 [1], 11400.0 [2], 90011.91 [3]
1,1,1-Trifluoro-3-[3-(3-propan-2-ylphenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]propan-2-olIC5020.0 [1], 2300.0 [2], 20003.22 [3]
(S)-1,1,1-Trifluoro-3-((3-phenoxyphenyl)(3-(1,1,2,2-tetrafluoroethoxy)benzyl)amino)propan-2-olIC50800.0 [1], 20000.0 [2]
3-((3-(1,1,2,2-Tetrafluoroethoxy)benzyl)(3-(3-ethylphenoxy)phenyl)amino)-1,1,1-trifluoropropan-2-olIC5060.0 [1], 60.26 [2], 1000.0 [3], 60006.74 [4]
1,1,1-Trifluoro-3-[3-(3-methyl-4-propan-2-ylphenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]propan-2-olIC50200.0 [1], 27200.0 [2], 200032.24 [3]
1-[1-(5-Chloropyridin-2-yl)-1-[3-fluoro-5-(trifluoromethyl)phenyl]-2-phenylethyl]-3-cyclopentylureaIC5030.0 [1], 31.0 [2], 5500.0 [3]
DalcetrapibIC504100.0 [1], 6000.0 [2]
1,1,1-Trifluoro-3-((4-phenoxyphenyl)(3-(trifluoromethoxy)benzyl)amino)propan-2-olIC5025000.0 [1]
1,1,1-Trifluoro-3-((4-fluoro-3-(furan-2-yl)benzyl)(3-phenoxyphenyl)amino)propan-2-olIC50720.0 [1], 49000.0 [2]
1,1,1-Trifluoro-3-[(3-phenoxyphenyl)[3-(2-thienyl)benzyl]amino]-2-propanolIC501120.0 [1], 83000.0 [2]
3-[3-[3-(Dimethylamino)phenoxy]-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]-1,1,1-trifluoropropan-2-olIC50199.53 [1], 200.0 [2], 200032.24 [3]
1,1,1-Trifluoro-3-[N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]-3-[[3-(trifluoromethoxy)phenyl]methoxy]anilino]propan-2-olIC5060.0 [1], 300.0 [2], 5700.0 [3]
1,1,1-Trifluoro-3-[(3-phenoxyphenyl)(3-biphenylylmethyl)amino]-2-propanolIC504420.0 [1], 47000.0 [2]
3-((3-(1,1,2,2-Tetrafluoroethoxy)benzyl)(3-(benzyloxy)phenyl)amino)-1,1,1-trifluoropropan-2-olIC50200.0 [1], 12100.0 [2]
1,1,1-Trifluoro-3-((3-(trifluoromethoxy)benzyl)(3-(trifluoromethoxy)phenyl)amino)propan-2-olIC501500.0 [1], 46000.0 [2]
1,1,1-Trifluoro-3-[N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]-3-[3-(trifluoromethyl)phenoxy]anilino]propan-2-olIC50200.0 [1], 10300.0 [2]
3-[3-(4-Chloro-3-methylphenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]-1,1,1-trifluoropropan-2-olIC50200.0 [1], 200032.24 [2]
1,1,1-Trifluoro-3-[3-(4-phenylphenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]propan-2-olIC502500.0 [1], 2511.89 [2], 2500345.36 [3]
3-((3-(1,1,2,2-Tetrafluoroethoxy)benzyl)(3-(2-chlorophenoxy)phenyl)amino)-1,1,1-trifluoropropan-2-olIC50300.0 [1], 299985.32 [2]
1,1,1-Trifluoro-3-[3-(4-propan-2-ylphenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]propan-2-olIC50400.0 [1], 31300.0 [2]
1,1,1,3,3,3-Hexafluoro-2-[3-[(3-phenoxy-N-(3,3,3-trifluoro-2-hydroxypropyl)anilino)methyl]phenyl]propan-2-olIC50420.0 [1], 4900.0 [2]
3-((3-(1,1,2,2-Tetrafluoroethoxy)benzyl)(3-(4-benzylphenoxy)phenyl)amino)-1,1,1-trifluoropropan-2-olIC502400.0 [1], 2399937.88 [2]
Methyl N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-N-[[2-(2-methoxy-5-propan-2-ylphenyl)-5-(trifluoromethyl)phenyl]methyl]carbamateIC50108.0 [1], 126.0 [2]
Unii-I0J230bjooIC507.0 [1], 25.0 [2], 50.0 [3]
3-((3-Tert-butoxybenzyl)(3-phenoxyphenyl)amino)-1,1,1-trifluoropropan-2-olIC50660.0 [1], 29000.0 [2]
1,1,1-Trifluoro-3-((3-phenoxybenzyl)(3-phenoxyphenyl)amino)propan-2-olIC505200.0 [1], 70000.0 [2]
1,1,1-Trifluoro-3-((3-phenoxyphenyl)(3-(2,2,2-trifluoroethoxy)benzyl)amino)propan-2-olIC501000.0 [1], 65000.0 [2]
N-(4-(5-Chlorobenzo[d]oxazol-2-yl)phenyl)-2-(o-tolyloxy)acetamideIC50470.0 [1], 1107.0 [2], 21000.0 [3]
(2S)-1,1,1-Trifluoro-3-[(2R)-2-[3-(1,1,2,2-tetrafluoroethoxy)phenyl]-5-[3-(trifluoromethoxy)phenyl]-3,4-dihydro-2H-quinolin-1-yl]propan-2-olIC5039.0 [1], 200.0 [2], 1200.0 [3]
N-(4-(5-Cyanobenzo[d]oxazol-2-yl)phenyl)-2-(o-tolyloxy)acetamideIC5057.0 [1], 130.0 [2], 3300.0 [3]
1,1,1-Trifluoro-3-((3-(4-fluorophenoxy)phenyl)(3-(1,1,2,2-tetrafluoroethoxy)benzyl)amino)propan-2-olIC5030.0 [1], 4100.0 [2], 29998.53 [3]
1,1,1-Trifluoro-3-[N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]-3-[3-(trifluoromethoxy)phenoxy]anilino]propan-2-olIC5030.0 [1], 3800.0 [2], 29998.53 [3]
1,1,1-Trifluoro-3-[3-phenoxy-N-[[3-(3,3,3-trifluoro-2-hydroxypropoxy)phenyl]methyl]anilino]propan-2-olIC501288.25 [1], 1300.0 [2], 62000.0 [3]
1,1,1-Trifluoro-3-[3-(4-propylphenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]propan-2-olIC50200.0 [1], 21300.0 [2], 200032.24 [3]
N-[4-(5-Cyano-7-methyl-1,3-benzoxazol-2-yl)phenyl]-2-[4-[4-(trifluoromethyl)phenyl]piperazin-1-yl]acetamideIC5016.0 [1], 18.0 [2]
3-[3-(2,3-Dichlorophenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]-1,1,1-trifluoropropan-2-olIC5030.0 [1], 600.0 [2], 29998.53 [3]
(5S)-4-Cyclohexyl-3-[(S)-fluoro-[4-(trifluoromethyl)phenyl]methyl]-7,7-dimethyl-2-propan-2-yl-6,8-dihydro-5H-quinolin-5-olIC5023.0 [1], 30.0 [2], 75.0 [3]
(5S)-4-Cyclohexyl-3-[(S)-fluoro-[4-(trifluoromethyl)phenyl]methyl]-2-propan-2-ylspiro[6,8-dihydro-5H-quinoline-7,1'-cyclobutane]-5-olIC5017.0 [1], 33.0 [2], 70.0 [3]
(5S)-4-Cyclohexyl-2-cyclopentyl-3-[(S)-fluoro-[4-(trifluoromethyl)phenyl]methyl]spiro[6,8-dihydro-5H-quinoline-7,1'-cyclobutane]-5-olIC5022.0 [1], 60.0 [2], 62.0 [3]
(3S,6S,9S)-9-Benzyl-13-hexan-2-yl-6-methyl-3-(2-methylpropyl)-1-oxa-4,7,10-triazacyclotridecane-2,5,8,11-tetroneIC50300.0 [1], 40000.0 [2], 50000.0 [3]
3-[[(8As)-2,5,5,8a-tetramethyl-3,4,4a,6,7,8-hexahydronaphthalen-1-yl]methyl]-4-methoxybenzene-1,2-diolIC501000.0 [1], 5000.0 [2], 5200.0 [3]
EvacetrapibIC5026.0 [1], 110.0 [2]
3-[3-(Cyclohexylmethoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]-1,1,1-trifluoropropan-2-olIC50200.0 [1]
1,1,1-Trifluoro-3-((3-fluorophenyl)(2-(trifluoromethyl)benzyl)amino)propan-2-olIC50100000.0 [1]
(R)-1,1,1-Trifluoro-3-((3-(trifluoromethylthio)benzyl)(3,4,5-trimethoxyphenyl)amino)propan-2-olIC505000.0 [1]
1,1,1-Trifluoro-3-((3-fluorophenyl)(4-(trifluoromethoxy)benzyl)amino)propan-2-olIC5015000.0 [1]
3-(Benzyl(3-fluorophenyl)amino)-1,1,1-trifluoropropan-2-olIC50100000.0 [1]
1,1,1-Trifluoro-3-((3-fluorophenyl)(3-methylbenzyl)amino)propan-2-olIC50100000.0 [1]
4-(3-((3-(1,1,2,2-Tetrafluoroethoxy)benzyl)(3,3,3-trifluoro-2-hydroxypropyl)amino)phenoxy)phenolIC503500.0 [1]
3-((3-Cyclopropylbenzyl)(3-phenoxyphenyl)amino)-1,1,1-trifluoropropan-2-olIC501000.0 [1]
1,1,1-Trifluoro-3-((3-(pyridin-3-yloxy)phenyl)(3-(1,1,2,2-tetrafluoroethoxy)benzyl)amino)propan-2-olIC501300.0 [1]
Methyl 3-(((3-phenoxyphenyl)(3,3,3-trifluoro-2-hydroxypropyl)amino)methyl)benzoateIC5016000.0 [1]
1,1,1-Trifluoro-3-((3-isopropoxyphenyl)(3-(1,1,2,2-tetrafluoroethoxy)benzyl)amino)propan-2-olIC50300.0 [1], 302.0 [2]
3-((3-Cyclopentylbenzyl)(3-phenoxyphenyl)amino)-1,1,1-trifluoropropan-2-olIC50300.0 [1]
1,1,1-Trifluoro-3-((3-fluorophenyl)(4-methylbenzyl)amino)propan-2-olIC5065000.0 [1]
3-((3-(1,1,2,2-Tetrafluoroethoxy)benzyl)(3-(cyclohexyloxy)phenyl)amino)-1,1,1-trifluoropropan-2-olIC502600.0 [1]
3-[3-(2,3-Difluorophenoxy)-N-[[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methyl]anilino]-1,1,1-trifluoropropan-2-olIC50100.0 [1]
3-((3-(1,1,2,2-Tetrafluoroethoxy)benzyl)(3-(cyclopentyloxy)phenyl)amino)-1,1,1-trifluoropropan-2-olIC50400.0 [1]
3-((3-(Trifluoromethyl)benzyl)(3-chlorophenyl)amino)-1,1,1-trifluoropropan-2-olIC5012000.0 [1]
1,1,1-Trifluoro-3-((3-fluorophenyl)(3-phenoxybenzyl)amino)propan-2-olIC5015000.0 [1]
3-((Biphenyl-4-ylmethyl)(3-fluorophenyl)amino)-1,1,1-trifluoropropan-2-olIC5020000.0 [1]
1,1,1-Trifluoro-3-(m-tolyl(3-(trifluoromethyl)benzyl)amino)propan-2-olIC5010000.0 [1]
1,1,1-Trifluoro-3-((3-(2-nitrophenoxy)phenyl)(3-(1,1,2,2-tetrafluoroethoxy)benzyl)amino)propan-2-olIC50398.11 [1], 400.0 [2]
1,1,1-Trifluoro-3-((3-(trifluoromethyl)benzyl)(3-(trifluoromethyl)phenyl)amino)propan-2-olIC5010000.0 [1]
1,1,1-Trifluoro-3-[(3-phenoxyphenyl)[3-(1-methyl-2-pyrrolyl)benzyl]amino]-2-propanolIC506790.0 [1]
1,1,1-Trifluoro-3-[(3-phenoxyphenyl)[3-(3-furanyl)benzyl]amino]-2-propanolIC50910.0 [1]
1,1,1-Trifluoro-3-[(3-phenoxyphenyl)[3-(2-pyridinyl)benzyl]amino]-2-propanolIC5022900.0 [1]
1,1,1-Trifluoro-3-((3-(furan-2-yl)-4-methylbenzyl)(3-phenoxyphenyl)amino)propan-2-olIC503960.0 [1], 3981.07 [2]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Cholesteryl ester transfer protein Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/cholesteryl-ester-transfer-protein-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 8). Quest Database™ Cholesteryl ester transfer protein Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cholesteryl-ester-transfer-protein-inhibitors-ic50-ki.
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