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Choline kinase alpha Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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12,20-Diaza-1,8-diazoniapentacyclo[19.2.2.23,6.28,11.114,18]triaconta-1(23),3(30),4,6(29),8(28),9,11(27),14,16,18(26),21,24-dodecaeneIC50300.0 [1]
Unii-PM765bvw4ZIC501920.0 [1], 2000.0 [2]
1-{4-[4-(4-Amino-1-quinoliniumylmethyl)phenethyl]benzyl}-4-quinoliniumamineIC5080000.0 [1]
1-{3-[3-(4-Amino-1-quinoliniumylmethyl)phenyl]benzyl}-4-quinoliniumamineIC501200.0 [1]
1-[[4-[4-[[4-(4-Chloro-N-methylanilino)pyridin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-N-(4-chlorophenyl)-N-methylpyridin-1-ium-4-amine;dibromideIC501800.0 [1]
1-[[3-[3-[[4-(4-Chloro-N-methylanilino)pyridin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-N-(4-chlorophenyl)-N-methylpyridin-1-ium-4-amine;dibromideIC501500.0 [1]
{4-[(4-Methyl-1,4-diazepan-1-yl)methyl]phenyl}methanamineIC5087000.0 [1]
6-(Trifluoromethyl)pyrimidin-4-amineIC50300000.0 [1]
Chembl4128522IC50920.0 [1]
6-[(4-Methyl-1,4-Diazepan-1-Yl)methyl]quinolineIC503900.0 [1]
7-Chloro-1-[[4-[2-[4-[[7-chloro-4-(4-chloro-N-methylanilino)quinolin-1-ium-1-yl]methyl]phenyl]ethyl]phenyl]methyl]-N-(4-chlorophenyl)-N-methylquinolin-1-ium-4-amine;dibromideIC505700.0 [1]
1-[[4-[4-[(4-Aminoquinolin-1-ium-1-yl)methyl]phenyl]phenyl]methyl]quinolin-1-ium-4-amine;dibromideIC5081100.0 [1]
7-Chloro-1-[[4-[4-[[7-chloro-4-(4-chloro-N-methylanilino)quinolin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-N-(4-chlorophenyl)-N-methylquinolin-1-ium-4-amine;dibromideIC5011400.0 [1]
2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi10000.0 [1]
2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi10000.0 [1]
1-Methyl-4-[[4-[4-[(4-methyl-1,4-diazepan-1-yl)methyl]phenyl]phenyl]methyl]-1,4-diazepaneIC50457.0 [1]
1-Methyl-4-[[4-[4-(trifluoromethyl)phenyl]phenyl]methyl]-1,4-diazepaneIC502600.0 [1]
(4-Methyl-1,4-diazepan-1-yl)-[4-[4-[(4-methyl-1,4-diazepan-1-yl)methyl]phenyl]phenyl]methanoneIC50251.0 [1]
1-[[2,6-Difluoro-4-[4-[(4-methyl-1,4-diazepan-1-yl)methyl]phenyl]phenyl]methyl]-4-methyl-1,4-diazepaneIC50255.0 [1]
1-[[2,3-Difluoro-4-[4-[(4-methyl-1,4-diazepan-1-yl)methyl]phenyl]phenyl]methyl]-4-methyl-1,4-diazepaneIC50233.0 [1]
2-[2-Fluoro-4-[(4-methyl-1,4-diazepan-1-yl)methyl]phenyl]-5-[(4-methyl-1,4-diazepan-1-yl)methyl]benzonitrileIC5085.0 [1]
1-[[2-Chloro-4-[4-[(4-methyl-1,4-diazepan-1-yl)methyl]phenyl]phenyl]methyl]-4-methyl-1,4-diazepaneIC50268.0 [1]
1-[[3-Fluoro-4-[4-[(4-methyl-1,4-diazepan-1-yl)methyl]phenyl]phenyl]methyl]-4-methyl-1,4-diazepaneIC50165.0 [1]
1-[[3-[[4-(4-Chloro-N-methylanilino)pyridin-1-ium-1-yl]methyl]phenyl]methyl]-N-(4-chlorophenyl)-N-methylpyridin-1-ium-4-amine;dibromideIC507200.0 [1]
(1S)-1-(1-Azabicyclo[2.2.2]octan-3-yl)-3-[2-(oxan-4-yloxy)phenyl]-1-phenylpropan-1-olIC5020.0 [1]
Chembl4126529IC506850.0 [1]
Chembl4126001IC502790.0 [1]
Chembl4129777IC502020.0 [1]
Chembl4127381IC503270.0 [1]
Chembl4127055IC5016220.0 [1]
[4-(4-Methyl-1,4-diazepan-1-yl)phenyl]methanolIC502000000.0 [1]
1-Methyl-4-[(4-phenylphenyl)methyl]-1,4-diazepaneIC501480.0 [1]
Azepan-1-yl-piperazin-1-yl-methanoneIC50300000.0 [1]
2-[4-[2-[4-[1,1,1,3,3,3-Hexafluoro-2-[4-[4-[1-(2-hydroxyethyl)pyridin-1-ium-4-yl]-5-(1,1,2,2,2-pentafluoroethyl)-1,3-oxazol-2-yl]phenyl]propan-2-yl]phenyl]-5-(1,1,2,2,2-pentafluoroethyl)-1,3-oxazol-4-yl]pyridin-1-ium-1-yl]ethanol;diiodideIC504200.0 [1]
2-[4-[2-[4-[4-[4-[1-[2-(Dimethylamino)-2-oxoethyl]pyridin-1-ium-4-yl]-5-(1,1,2,2,2-pentafluoroethyl)-1,3-oxazol-2-yl]phenyl]phenyl]-5-(1,1,2,2,2-pentafluoroethyl)-1,3-oxazol-4-yl]pyridin-1-ium-1-yl]-N,N-dimethylacetamide;diiodideIC503100.0 [1]
2-[4-[2-[4-[4-[4-[1-(2-Hydroxyethyl)pyridin-1-ium-4-yl]-5-(trifluoromethyl)-1,3-oxazol-2-yl]phenyl]phenyl]-5-(trifluoromethyl)-1,3-oxazol-4-yl]pyridin-1-ium-1-yl]ethanol;diiodideIC5023800.0 [1]
2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamideIC5010000.0 [1]
8-[(2R)-1-(3,5-Difluorophenyl)pyrrolidin-2-yl]-6-(morpholine-4-carbonyl)-2-morpholino-chromen-4-oneIC5050000.0 [1]
1-Methyl-4-(naphthalen-2-ylmethyl)-1,4-diazepaneIC502600.0 [1]
5-[(4-Methyl-1,4-diazepan-1-yl)methyl]-2-[4-[(4-methyl-1,4-diazepan-1-yl)methyl]phenyl]benzonitrileIC5066.0 [1]
1-Methyl-4-[[4-[4-(4-methylpiperazin-1-yl)phenyl]phenyl]methyl]-1,4-diazepaneIC501300.0 [1]
Methyl 4-[4-[(4-methyl-1,4-diazepan-1-yl)methyl]phenyl]benzoateIC504950.0 [1]
1-[[4-(4-Methoxyphenyl)phenyl]methyl]-4-methyl-1,4-diazepaneIC501430.0 [1]
6-[(1-Methyl-1,4-diazepan-6-yl)methyl]quinolineIC5017200.0 [1]
1-[[3,5-Bis[[4-(4-chloro-N-methylanilino)pyridin-1-ium-1-yl]methyl]phenyl]methyl]-N-(4-chlorophenyl)-N-methylpyridin-1-ium-4-amineIC501400.0 [1]
1,2-Di{4-[4-(1-azepanyl)-1-pyridiniumylmethyl]phenyl}ethane dibromideIC5015000.0 [1]
N-Methyl-1-[[3-[[4-(N-methylanilino)pyridin-1-ium-1-yl]methyl]phenyl]methyl]-N-phenylpyridin-1-ium-4-amineIC5037500.0 [1]
1,2-Di[4-(4-hexahydro-1-pyridinyl-1-pyridiniumylmethyl)phenyl]ethane dibromideIC509600.0 [1]
1-{4-[4-(4-Cyano-1-pyridiniumylmethyl)phenethyl]benzyl}-4-pyridiniumcarbonitrile dibromideIC501000000.0 [1]
1,2-Di[4-(4-tetrahydro-1H-1-pyrrolyl-1-pyridiniumylmethyl)phenyl]ethane dibromideIC5020000.0 [1]
1-[[4-[2-[4-[[4-(Dimethylamino)pyridin-1-ium-1-yl]methyl]phenyl]ethyl]phenyl]methyl]-N,N-dimethylpyridin-1-ium-4-amineIC5017000.0 [1]
1-[[4-[2-[4-[[4-[Bis(prop-2-enyl)amino]pyridin-1-ium-1-yl]methyl]phenyl]ethyl]phenyl]methyl]-N,N-bis(prop-2-enyl)pyridin-1-ium-4-amineIC5017000.0 [1]
1-{4-[4-(4-Hydroxymethyl-1-pyridiniumylmethyl)phenethyl]benzyl}-4-pyridiniumylmethanol dibromideIC50100000.0 [1]
1,2-Di[4-(4-methyl-1-pyridiniumylmethyl)phenyl]ethane dibromideIC50100000.0 [1]
1-{4-[4-(4-Amino-1-pyridiniumylmethyl)phenethyl]benzyl}-4-pyridiniumamine dibromideIC5023000.0 [1]
1-[[4-[2-[4-[(4-Carboxypyridin-1-ium-1-yl)methyl]phenyl]ethyl]phenyl]methyl]pyridin-1-ium-4-carboxylic acidIC50136700.0 [1]
12,19-Diaza-1,8-diazoniapentacyclo[18.2.2.23,6.28,11.214,17]triaconta-1(22),3(30),4,6(29),8(28),9,11(27),14,16,20,23,25-dodecaeneIC502100.0 [1]
13,21-Diaza-1,9-diazoniapentacyclo[20.2.2.29,12.13,7.115,19]triaconta-1(24),3(30),4,6,9(29),10,12(28),15,17,19(27),22,25-dodecaeneIC5013200.0 [1]
Pyridinium, 1,1'-[1,3-phenylenebis(methylene)]bis[4-(1-piperidinyl)-IC5052800.0 [1]
Pyridinium, 1,1'-[1,3-phenylenebis(methylene)]bis[4-(1-pyrrolidinyl)-IC5084200.0 [1]
4-Piperidin-1-yl-1-[[4-[4-[(4-piperidin-1-ylpyridin-1-ium-1-yl)methyl]phenyl]phenyl]methyl]pyridin-1-iumIC508800.0 [1]
1-[[3-[3-[(4-Amino-7-chloroquinolin-1-ium-1-yl)methyl]phenyl]phenyl]methyl]-7-chloroquinolin-1-ium-4-amineIC5020600.0 [1]
N-Methyl-1-[[4-[4-[[4-(N-methylanilino)quinolin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-N-phenylquinolin-1-ium-4-amineIC503000.0 [1]
N-Methyl-1-[[4-[2-[4-[[4-(N-methylanilino)quinolin-1-ium-1-yl]methyl]phenyl]ethyl]phenyl]methyl]-N-phenylquinolin-1-ium-4-amineIC501400.0 [1]
4-Pyrrolidin-1-yl-1-[[4-[4-[(4-pyrrolidin-1-ylpyridin-1-ium-1-yl)methyl]phenyl]phenyl]methyl]pyridin-1-iumIC5011100.0 [1]
4-Piperidin-1-yl-1-[[3-[3-[(4-piperidin-1-ylpyridin-1-ium-1-yl)methyl]phenyl]phenyl]methyl]pyridin-1-iumIC501900.0 [1]
1-[[4-[2-[4-[[4-(4-Chloro-N-methylanilino)quinolin-1-ium-1-yl]methyl]phenyl]ethyl]phenyl]methyl]-N-(4-chlorophenyl)-N-methylquinolin-1-ium-4-amineIC504800.0 [1]
1-[[3-[[4-(3,5-Dichloro-N-methylanilino)pyridin-1-ium-1-yl]methyl]phenyl]methyl]-N-(3,5-dichlorophenyl)-N-methylpyridin-1-ium-4-amineIC508400.0 [1]
7-Chloro-1-[[3-[3-[(7-chloro-4-pyrrolidin-1-ylquinolin-1-ium-1-yl)methyl]phenyl]phenyl]methyl]-4-pyrrolidin-1-ylquinolin-1-iumIC501200.0 [1]
1-[[4-[4-[[7-Amino-8-methyl-4-(N-methylanilino)quinolin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-4-N,8-dimethyl-4-N-phenylquinolin-1-ium-4,7-diamineIC5096100.0 [1]
4-(Azepan-1-yl)-1-[[3-[3-[[4-(azepan-1-yl)quinolin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]quinolin-1-iumIC50500.0 [1]
1-[[4-[2-[4-[[7-Amino-8-methyl-4-(N-methylanilino)quinolin-1-ium-1-yl]methyl]phenyl]ethyl]phenyl]methyl]-4-N,8-dimethyl-4-N-phenylquinolin-1-ium-4,7-diamineIC50133000.0 [1]
1-[[4-[[4-(4-Chloro-N-methylanilino)pyridin-1-ium-1-yl]methyl]phenyl]methyl]-N-(4-chlorophenyl)-N-methylpyridin-1-ium-4-amineIC502900.0 [1]
N-Methyl-1-[[3-[3-[[4-(N-methylanilino)pyridin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-N-phenylpyridin-1-ium-4-amineIC50400.0 [1]
1-[[3-[3-[(4-Anilinoquinolin-1-ium-1-yl)methyl]phenyl]phenyl]methyl]-N-phenylquinolin-1-ium-4-amineIC501300.0 [1]
7-Chloro-1-[[4-[2-[4-[[7-chloro-4-(dimethylamino)quinolin-1-ium-1-yl]methyl]phenyl]ethyl]phenyl]methyl]-N,N-dimethylquinolin-1-ium-4-amineIC509000.0 [1]
1-[[3-[3-[[4-(4-Chloro-N-methylanilino)quinolin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-N-(4-chlorophenyl)-N-methylquinolin-1-ium-4-amineIC502100.0 [1]
Pyridinium, 1,1'-[1,4-phenylenebis(methylene)]bis[4-(1-piperidinyl)-IC5037700.0 [1]
N-Methyl-1-[[3-[3-[[4-(N-methylanilino)quinolin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-N-phenylquinolin-1-ium-4-amineIC50400.0 [1]
1-[[4-[4-[(4-Anilinoquinolin-1-ium-1-yl)methyl]phenyl]phenyl]methyl]-N-phenylquinolin-1-ium-4-amineIC5017800.0 [1]
4-(Azepan-1-yl)-1-[[4-[2-[4-[[4-(azepan-1-yl)quinolin-1-ium-1-yl]methyl]phenyl]ethyl]phenyl]methyl]quinolin-1-iumIC50600.0 [1]
7-Chloro-1-[[3-[3-[[7-chloro-4-(dimethylamino)quinolin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-N,N-dimethylquinolin-1-ium-4-amineIC509600.0 [1]
4-(Azepan-1-yl)-1-[[4-[4-[[4-(azepan-1-yl)quinolin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]quinolin-1-iumIC502200.0 [1]
1-[[4-[2-[4-[[4-(Dimethylamino)quinolin-1-ium-1-yl]methyl]phenyl]ethyl]phenyl]methyl]-N,N-dimethylquinolin-1-ium-4-amineIC5010200.0 [1]
1-[[3-[3-[[7-Amino-8-methyl-4-(N-methylanilino)quinolin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-4-N,8-dimethyl-4-N-phenylquinolin-1-ium-4,7-diamineIC5056800.0 [1]
4-Pyrrolidin-1-yl-1-[[3-[3-[(4-pyrrolidin-1-ylpyridin-1-ium-1-yl)methyl]phenyl]phenyl]methyl]pyridin-1-iumIC505800.0 [1]
7-Chloro-1-[[4-[4-[[7-chloro-4-(dimethylamino)quinolin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-N,N-dimethylquinolin-1-ium-4-amineIC5020600.0 [1]
1-[[3-[3-[[7-Amino-4-(4-chloro-N-methylanilino)-8-methylquinolin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-4-N-(4-chlorophenyl)-4-N,8-dimethylquinolin-1-ium-4,7-diamineIC50147000.0 [1]
N-Methyl-1-[[4-[4-[[4-(N-methylanilino)pyridin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-N-phenylpyridin-1-ium-4-amineIC504300.0 [1]
7-Chloro-1-[[4-[4-[(7-chloro-4-pyrrolidin-1-ylquinolin-1-ium-1-yl)methyl]phenyl]phenyl]methyl]-4-pyrrolidin-1-ylquinolin-1-iumIC5019800.0 [1]
7-Chloro-1-[[4-[4-[[7-chloro-4-(N-methylanilino)quinolin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-N-methyl-N-phenylquinolin-1-ium-4-amineIC5011400.0 [1]
1-[[3-[3-[(4-Amino-3-methylquinolin-1-ium-1-yl)methyl]phenyl]phenyl]methyl]-3-methylquinolin-1-ium-4-amineIC5011900.0 [1]
1-[[3-[3-[[4-(Dimethylamino)quinolin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-N,N-dimethylquinolin-1-ium-4-amineIC504400.0 [1]
1-[[4-[2-[4-[(4-Amino-7-chloroquinolin-1-ium-1-yl)methyl]phenyl]ethyl]phenyl]methyl]-7-chloroquinolin-1-ium-4-amineIC50200000.0 [1]
7-Chloro-1-[[3-[3-[[7-chloro-4-(N-methylanilino)quinolin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-N-methyl-N-phenylquinolin-1-ium-4-amineIC503100.0 [1]
1-[[4-[[4-(3,5-Dichloro-N-methylanilino)pyridin-1-ium-1-yl]methyl]phenyl]methyl]-N-(3,5-dichlorophenyl)-N-methylpyridin-1-ium-4-amineIC509700.0 [1]
Pyridinium, 1,1'-[1,4-phenylenebis(methylene)]bis[4-(1-pyrrolidinyl)-IC5024000.0 [1]
1-[[4-[4-[[4-(Dimethylamino)quinolin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-N,N-dimethylquinolin-1-ium-4-amineIC5039700.0 [1]
1-[[4-[2-[4-[(4-Anilinoquinolin-1-ium-1-yl)methyl]phenyl]ethyl]phenyl]methyl]-N-phenylquinolin-1-ium-4-amineIC502300.0 [1]
1-[[4-[4-[[7-Amino-4-(4-chloro-N-methylanilino)-8-methylquinolin-1-ium-1-yl]methyl]phenyl]phenyl]methyl]-4-N-(4-chlorophenyl)-4-N,8-dimethylquinolin-1-ium-4,7-diamineIC5046100.0 [1]
Items per page: 1 - 10 of 100
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References

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MLA

"Quest Database™ Choline kinase alpha Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/choline-kinase-alpha-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Choline kinase alpha Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/choline-kinase-alpha-inhibitors-ic50-ki.
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