Chondroitin sulfate N-acetylgalactosaminyltransferase 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	(2S)-2-[[4-[4-[(6-Fluoro-1,3-benzothiazol-2-yl)amino]phenyl]benzoyl]amino]-3-methylbutanoic acid	IC50	35000.0 [1]
	(2S)-2-[[3-[4-[(6-Fluoro-1,3-benzothiazol-2-yl)amino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	120000.0 [1]
	(S)-2-[(3-{4-[3-(4-Fluoro-phenyl)-ureido]-phenyl}-isoxazole-5-carbonyl)-amino]-3-methyl-butyric acid	IC50	60000.0 [1]
	(2S)-2-[[3-[4-[(2-Chlorophenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	44000.0 [1]
	(2S)-2-[[5-[4-[(2-Chlorophenyl)carbamoylamino]phenyl]-1,3-oxazole-2-carbonyl]amino]-3-methylbutanoic acid	IC50	282000.0 [1]
	(2S)-2-[[3-[4-[(3-Chlorophenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	45000.0 [1]
	(2S)-2-[[3-[4-[(4-Chlorophenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	124000.0 [1]
	(2S)-3-Methyl-2-[[3-[4-[[3-(trifluoromethyl)phenyl]carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]butanoic acid	IC50	66000.0 [1]
	(2S)-3-Methyl-2-[[5-[4-[[3-(trifluoromethyl)phenyl]carbamoylamino]phenyl]-1,3-oxazole-2-carbonyl]amino]butanoic acid	IC50	458000.0 [1]
	(2S)-2-[[3-[4-[(3,4-Dimethylphenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	44000.0 [1]
	(2S)-2-[[3-[4-[(4-Chloro-2-phenoxyphenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	86000.0 [1]
	(2S)-2-[[5-[4-[(4-Chloro-2-phenoxyphenyl)carbamoylamino]phenyl]-1,3-oxazole-2-carbonyl]amino]-3-methylbutanoic acid	IC50	230000.0 [1]
	(2S)-2-[[3-[4-[(4-Chloro-2-fluorophenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	24000.0 [1]
	(2S)-2-[[3-[4-[(2,4-Difluorophenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	62000.0 [1]
	(2S)-2-[[3-[4-[(2,4-Difluorophenyl)carbamoylamino]phenyl]-1,2,4-oxadiazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	259000.0 [1]
	(2S)-3-Methyl-2-[[3-[4-[(4-methylphenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]butanoic acid	IC50	61000.0 [1]
	(2S)-2-[[3-[4-[(4-Methoxyphenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	64000.0 [1]
	(2S)-2-[[3-[4-[(2-Fluorophenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	141000.0 [1]
	(2S)-2-[[3-[4-[(3-Fluorophenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	94000.0 [1]
	(2S)-3-Methyl-2-[[3-[4-[(2-methylphenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]butanoic acid	IC50	84000.0 [1]
	(2S)-3-Methyl-2-[[3-[4-[(3-methylphenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]butanoic acid	IC50	54000.0 [1]
	(2S)-3-Methyl-2-[[3-[4-[[2-(trifluoromethyl)phenyl]carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]butanoic acid	IC50	54000.0 [1]
	(2S)-3-Methyl-2-[[3-[4-[[4-(trifluoromethyl)phenyl]carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]butanoic acid	IC50	80000.0 [1]
	(2S)-2-[[3-[4-[(3,4-Difluorophenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	75000.0 [1]
	(2S)-2-[[3-[4-[(3,5-Difluorophenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	75000.0 [1]
	(2S)-2-[[3-[4-[(2,5-Difluorophenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	141000.0 [1]
	(2S)-2-[[3-[4-[(2,6-Difluorophenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	185000.0 [1]
	(2S)-2-[[3-[4-[(2,4-Dimethylphenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	85000.0 [1]
	(2S)-2-[[3-[4-[(3,5-Dimethylphenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	114000.0 [1]
	(2S)-2-[[3-[4-[(2-Fluoro-5-methylphenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	54000.0 [1]
	(2S)-2-[[3-[4-[(3-Fluoro-4-methylphenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	178000.0 [1]
	(2S)-2-[[3-[4-[(4-Fluoro-2-methylphenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	90000.0 [1]
	(2S)-2-[[3-[4-[(5-Fluoro-2-methylphenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid	IC50	69000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 33 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Chondroitin sulfate N-acetylgalactosaminyltransferase 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/chondroitin-sulfate-n-acetylgalactosaminyltransferase-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Chondroitin sulfate N-acetylgalactosaminyltransferase 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/chondroitin-sulfate-n-acetylgalactosaminyltransferase-1-inhibitors-ic50-ki.
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