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Coagulation factor III Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
Trichostatin AIC5020.0 [1]
SodiumIC501000000.0 [1], 2000000.0 [2]
Valproic acidIC501500000.0 [1], 2000000.0 [2]
EntinostatIC506000.0 [1], 10000.0 [2]
(1E,4Z,6E)-5-Hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-oneIC50199.63 [1]
ApicidinIC50150.0 [1], 200.0 [2]
({3-[3-(5-Carbamimidoyl-1H-1,3-benzodiazol-2-yl)-2-hydroxyphenyl]-4-hydroxyphenyl}methyl)ureaKi13.0 [1]
CurcuminIC5013.16 [1]
Oleanolic acidIC504.97 [1]
TetrahydropalmatineIC5022.78 [1]
RotundineIC5014.98 [1]
l-StepholidineIC50104.58 [1]
HederageninIC500.22 [1]
CanadineIC508.35 [1]
Echinocystic acidIC500.05 [1]
Oleanonic acidIC500.22 [1]
DibenzylideneacetoneIC500.05 [1]
4'-HydroxychalconeIC500.12 [1]
(1E,4E)-1,5-Bis(4-hydroxy-3-methoxyphenyl)penta-1,4-dien-3-oneIC50200.0 [1]
CyqualonIC50200.0 [1]
CorydalmineIC50152.43 [1]
1,5-Bis(4-hydroxyphenyl)penta-1,4-dien-3-oneIC502.58 [1]
2,6-DibenzylidenecyclohexanoneIC500.26 [1]
4,4'-DihydroxychalconeIC500.96 [1]
2,6-Bis(4-hydroxybenzylidene)cyclohexanoneIC500.94 [1]
Eclalbasaponin IIC509.58 [1]
4,4'-DimethoxychalconeIC5015.39 [1]
(1E,4E)-1,5-Bis(4-methoxyphenyl)penta-1,4-dien-3-oneIC5013.37 [1]
Benzyl oleanolateIC504.68 [1]
(2E)-3-(4-Hydroxyphenyl)-1-(4-methoxyphenyl)prop-2-en-1-oneIC50141.98 [1]
(RS)-NandinineIC5012.17 [1]
2,6-Bis(4-methoxybenzylidene)cyclohexanoneIC50200.0 [1]
Vitalboside AIC500.1 [1]
2-[3-(6-Carbamimidoyl-1H-benzimidazol-2-yl)-5-[5-[(carbamoylamino)methyl]-2-hydroxyphenyl]-4-hydroxyphenyl]butanedioic acidKi2.0 [1]
2-[3-(6-Carbamimidoyl-1H-benzimidazol-2-yl)-5-(5-fluoro-2-hydroxyphenyl)-4-hydroxyphenyl]butanedioic acidKi4.0 [1]
Oleanolic acid 28-O-beta-D-glucopyranosideIC500.04 [1]
Hederagenin 28-O-beta-D-glucopyranosyl esterIC500.28 [1]
NandinineIC5036.41 [1]
28-O-GlucopyranosylepiederageninIC506.46 [1]
[(2R,3R,4S,5S,6R)-3,4,5-Trihydroxy-6-(hydroxymethyl)oxan-2-yl] (4aS,6aR,6aS,6bR,8aR,10S,12aR,14bS)-2,2,6a,6b,9,9,12a-heptamethyl-10-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicene-4a-carboxylateIC5015.95 [1]
5-[[(2S)-1-Amino-4-methyl-1-oxopentan-2-yl]carbamoyl]-2-[2-[[4-(aminomethyl)phenyl]carbamoyl]-4-(methylamino)phenyl]benzoic acidIC50590.0 [1]
2-[2-[(4-Carbamimidoylphenyl)carbamoyl]phenyl]-5-(2-methylpropylcarbamoyl)benzoic acidIC5089.0 [1]
[(2S,3R,4S,5S,6R)-3,4,5-Trihydroxy-6-(hydroxymethyl)oxan-2-yl] (4aR,5R,6aR,6aS,6bR,8aR,10S,12aR,14bS)-5,10-dihydroxy-2,2,6a,6b,9,9,12a-heptamethyl-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicene-4a-carboxylateIC5010.61 [1]
2,3,10-Trimethoxy-6,8,13,13a-tetrahydro-5H-isoquinolino[2,1-b]isoquinolin-9-olIC50187.26 [1]
Nandinine, (-)-IC506.75 [1]
9,10-Dimethoxy-6,8,13,13a-tetrahydro-5H-isoquinolino[2,1-b]isoquinoline-2,3-diolIC50968.9 [1]
4-EpihederageninIC501.29 [1]
2-[3-(6-Carbamimidoyl-1H-benzimidazol-2-yl)-5-[5-(carbamoylamino)-2-hydroxyphenyl]-4-hydroxyphenyl]butanedioic acidKi44.0 [1]
2-[3-[5-(Aminomethyl)-2-hydroxyphenyl]-5-(6-carbamimidoyl-1H-benzimidazol-2-yl)-4-hydroxyphenyl]butanedioic acidKi35.0 [1]
2-[3-(6-Carbamimidoyl-1H-benzimidazol-2-yl)-5-(5-carboxy-2-hydroxyphenyl)-4-hydroxyphenyl]butanedioic acidKi43.0 [1]
2-[3-(6-Carbamimidoyl-1H-benzimidazol-2-yl)-5-(5-carbamoyl-2-hydroxyphenyl)-4-hydroxyphenyl]butanedioic acidKi14.0 [1]
2-[3-(6-Carbamimidoyl-1H-benzimidazol-2-yl)-5-[5-(2-carboxyethyl)-2-hydroxyphenyl]-4-hydroxyphenyl]butanedioic acidKi13.0 [1]
2-[3-[5-(2-Amino-2-oxoethyl)-2-hydroxyphenyl]-5-(6-carbamimidoyl-1H-benzimidazol-2-yl)-4-hydroxyphenyl]butanedioic acidKi12.0 [1]
2-[3-(6-Carbamimidoyl-1H-benzimidazol-2-yl)-5-[5-(carboxymethyl)-2-hydroxyphenyl]-4-hydroxyphenyl]butanedioic acidKi12.0 [1]
[(2S,3R,4S,5S,6R)-3,4,5-Trihydroxy-6-(hydroxymethyl)oxan-2-yl] (1R,3aS,5aR,5bR,7aR,8R,9S,11aR,11bR,13bS)-9-hydroxy-8-(hydroxymethyl)-5a,5b,8,11a-tetramethyl-1-prop-1-en-2-yl-1,2,3,4,5,6,7,7a,9,10,11,11b,12,13,13a,13b-hexadecahydrocyclopenta[a]chrysene-3a-carboxylateIC500.03 [1]
[(2S,3R,4S,5S,6R)-3,4,5-Trihydroxy-6-(hydroxymethyl)oxan-2-yl] (4aR,5R,6aR,6aS,6bR,8aR,9S,10S,12aR,14bS)-5,10-dihydroxy-9-(hydroxymethyl)-2,2,6a,6b,9,12a-hexamethyl-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicene-4a-carboxylateIC500.8 [1]
[(2R,3R,4S,5S,6R)-3,4,5-Trihydroxy-6-(hydroxymethyl)oxan-2-yl] (1R,3aS,5aR,5bR,7aR,9S,11aR,11bR,13bS)-5a,5b,8,8,11a-pentamethyl-1-prop-1-en-2-yl-9-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1,2,3,4,5,6,7,7a,9,10,11,11b,12,13,13a,13b-hexadecahydrocyclopenta[a]chrysene-3a-carboxylateIC500.64 [1]
[(2S,3R,4S,5S,6R)-3,4,5-Trihydroxy-6-(hydroxymethyl)oxan-2-yl] (1R,3aS,5aR,5bR,7aR,9S,11aR,11bR,13bS)-9-hydroxy-5a,5b,8,8,11a-pentamethyl-1-prop-1-en-2-yl-1,2,3,4,5,6,7,7a,9,10,11,11b,12,13,13a,13b-hexadecahydrocyclopenta[a]chrysene-3a-carboxylateIC500.08 [1]
(1R,3As,5aR,5bR,7aR,8R,9S,11aR,11bR,13bS)-9-hydroxy-8-(hydroxymethyl)-5a,5b,8,11a-tetramethyl-1-prop-1-en-2-yl-1,2,3,4,5,6,7,7a,9,10,11,11b,12,13,13a,13b-hexadecahydrocyclopenta[a]chrysene-3a-carboxylic acidIC500.22 [1]
(17-Methoxy-5,7-dioxa-13-azapentacyclo[11.8.0.02,10.04,8.015,20]henicosa-2,4(8),9,15(20),16,18-hexaen-16-yl) acetateIC5063.06 [1]
1-(2,6-Difluorophenyl)-3-{[3-(2-hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}ureaKi33.0 [1]
[2'-Hydroxy-3'-(1H-pyrrolo[3,2-c]pyridin-2-yl)-biphenyl-3-ylmethyl]-ureaKi800.0 [1]
2-[3-(4-Amino-1H-pyrrolo[3,2-c]pyridin-2-yl)-5-[3-[[(2,6-difluorophenyl)carbamoylamino]methyl]phenyl]-4-hydroxyphenyl]-2-methylpropanoic acidKi2.6 [1]
1-{[3-(2-Hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}-3-pentylureaKi335.0 [1]
3-{[3-(2-Hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}-1-(2-phenylethyl)ureaKi270.0 [1]
1-[[3-[2-Hydroxy-3-(1H-pyrrolo[3,2-c]pyridin-2-yl)phenyl]phenyl]methyl]-3-(2-thiophen-2-ylethyl)ureaKi350.0 [1]
3-{[3-(2-Hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}-1-phenylureaKi61.5 [1]
1-(2-Fluorophenyl)-3-{[3-(2-hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}ureaKi57.0 [1]
1-(3-Fluorophenyl)-3-{[3-(2-hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}ureaKi130.0 [1]
1-(4-Fluorophenyl)-3-{[3-(2-hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}ureaKi110.0 [1]
1-(2,4-Difluorophenyl)-3-{[3-(2-hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}ureaKi100.0 [1]
1-(3,4-Difluorophenyl)-3-{[3-(2-hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}ureaKi330.0 [1]
1-(3,5-Difluorophenyl)-3-{[3-(2-hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}ureaKi830.0 [1]
1-(2-Chlorophenyl)-3-{[3-(2-hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}ureaKi57.0 [1]
3-{[3-(2-Hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}-1-(2-methoxyphenyl)ureaKi47.0 [1]
3-{[3-(2-Hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}-1-(3-methoxyphenyl)ureaKi100.0 [1]
3-{[3-(2-Hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}-1-(4-methoxyphenyl)ureaKi88.0 [1]
1-(2,4-Dimethoxyphenyl)-3-{[3-(2-hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}ureaKi28.0 [1]
1-(3-Acetylphenyl)-3-{[3-(2-hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}ureaKi60.0 [1]
1-(4-Acetylphenyl)-3-{[3-(2-hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}ureaKi190.0 [1]
4-[[3-[2-Hydroxy-3-(1H-pyrrolo[3,2-c]pyridin-2-yl)phenyl]phenyl]methylcarbamoylamino]benzoic acidKi58.0 [1]
1-{[3-(2-Hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}-3-thiophen-2-ylureaKi160.0 [1]
1-{[3-(2-Hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}-3-thiophen-3-ylureaKi130.0 [1]
3-{[3-(2-Hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}-1-pyridin-2-ylureaKi2700.0 [1]
3-{[3-(2-Hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}-1-pyridin-3-ylureaKi155.0 [1]
N-[[3-[2-Hydroxy-3-(1H-pyrrolo[3,2-c]pyridin-2-yl)phenyl]phenyl]methyl]pyrrolidine-1-carboxamideKi17000.0 [1]
N-[[3-[2-Hydroxy-3-(1H-pyrrolo[3,2-c]pyridin-2-yl)phenyl]phenyl]methyl]-4-methylpiperazine-1-carboxamideKi130000.0 [1]
N-[[3-[2-Hydroxy-3-(1H-pyrrolo[3,2-c]pyridin-2-yl)phenyl]phenyl]methyl]-2-phenylacetamideKi2000.0 [1]
2-(2,6-Difluorophenyl)-N-[[3-[2-hydroxy-3-(1H-pyrrolo[3,2-c]pyridin-2-yl)phenyl]phenyl]methyl]acetamideKi9500.0 [1]
3-Hydroxy-N-[[3-[2-hydroxy-3-(1H-pyrrolo[3,2-c]pyridin-2-yl)phenyl]phenyl]methyl]-2-phenylpropanamideKi220.0 [1]
3-Hydroxy-N-[[3-[2-hydroxy-3-(1H-pyrrolo[3,2-c]pyridin-2-yl)phenyl]phenyl]methyl]-2-pyridin-3-ylpropanamideKi610.0 [1]
2-Hydroxy-N-[[3-[2-hydroxy-3-(1H-pyrrolo[3,2-c]pyridin-2-yl)phenyl]phenyl]methyl]-2-phenylacetamideKi850.0 [1]
1-Benzyl-1-hydroxy-3-{[3-(2-hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}ureaKi72.0 [1]
2-[6-(3-Carbamimidoylphenoxy)-4-[di(propan-2-yl)amino]-3,5-difluoropyridin-2-yl]oxy-5-(2-methylpropylcarbamoyl)benzoic acid;2,2,2-trifluoroacetic acidIC5020.0 [1]
(2S)-2-Hydroxy-N-[[3-[2-hydroxy-3-(1H-pyrrolo[3,2-c]pyridin-2-yl)phenyl]phenyl]methyl]-3-phenylpropanamideKi220.0 [1]
(2S)-N-[[3-[3-(4-Amino-1H-pyrrolo[3,2-c]pyridin-2-yl)-2-hydroxyphenyl]phenyl]methyl]-2-hydroxy-3-phenylpropanamideKi81.0 [1]
2-[3-(4-Amino-1H-pyrrolo[3,2-c]pyridin-2-yl)-4-hydroxy-5-[3-[[[(2S)-2-hydroxy-3-phenylpropanoyl]amino]methyl]phenyl]phenyl]-2-methylpropanoic acidKi15.0 [1]
4-[[3-[3-(4-Amino-1H-pyrrolo[3,2-c]pyridin-2-yl)-5-(2-carboxypropan-2-yl)-2-hydroxyphenyl]phenyl]methylcarbamoylamino]benzoic acidKi20.0 [1]
3-(4-Amino-1H-pyrrolo[3,2-c]pyridin-2-yl)-4-hydroxy-5-[3-[[[(2S)-2-hydroxy-3-phenylpropanoyl]amino]methyl]phenyl]benzoic acidKi1.3 [1]
2-[2-[[4-(Aminomethyl)phenyl]carbamoyl]-4-(methylamino)phenyl]-5-[[(2S)-1-hydroxy-4-methylpentan-2-yl]carbamoyl]benzoic acidIC501300.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Coagulation factor III Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/coagulation-factor-iii-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 8). Quest Database™ Coagulation factor III Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/coagulation-factor-iii-inhibitors-ic50-ki.
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