Structure | Compound Name | Standard Type | Standard Values (in nM) |
---|---|---|---|
3-(6-(Dimethylamino)-4-methylpyridin-3-yl)-2,5-dimethyl-N,N-dipropylpyrazolo[1,5-a]pyrimidin-7-amine | IC50 | 4.0 [1], 50.0 [2] | |
3-(6-(Dimethylamino)-4-methylpyridin-3-yl)-2,5-dimethyl-N,N-dipropylpyrazolo[1,5-a]pyrimidin-7-amine | Ki | 3.5 [1], 7.8 [2], 8.3 [3], 12.0 [4] | |
Butyl-(2,5-dimethyl-7-(2,4,6-trimethylphenyl)-7H-pyrrolo(2,3-d)pyrimidin-4-yl)ethylamine | IC50 | 11.0 [1], 15.85 [2] | |
CID 9909468 | IC50 | 39.81 [1], 82.0 [2] | |
CID 9909468 | Ki | 1.7 [1], 1.8 [2], 2.0 [3] | |
MLA | "Quest Database™ Corticotropin releasing factor receptor 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 30 Sep. 2025, https://www.aatbio.com/data-sets/corticotropin-releasing-factor-receptor-1-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, September 30). Quest Database™ Corticotropin releasing factor receptor 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/corticotropin-releasing-factor-receptor-1-inhibitors-ic50-ki. | |
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