Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Seliciclib | IC50 | 450.0 [1] | |
| (5Z)-5-(Quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5H)-one | IC50 | 19.0 [1] | |
| (5Z)-5-(Quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5H)-one | Ki | 35.0 [1] | |
| (Z)-2-((1R,2S)-2-Phenylcyclopropylamino)-5-(quinolin-6-ylmethylene)thiazol-4(5H)-one | IC50 | 2340.0 [1], 2410.0 [2], 2490.0 [3], 3340.0 [4], 6580.0 [5] | |
| (Z)-2-((1R,2S)-2-Phenylcyclopropylamino)-5-(quinolin-6-ylmethylene)thiazol-4(5H)-one | Ki | 20.0 [1] | |
MLA | "Quest Database™ Cyclin-dependent kinase 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 1 Nov. 2025, https://www.aatbio.com/data-sets/cyclin-dependent-kinase-1-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, November 1). Quest Database™ Cyclin-dependent kinase 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cyclin-dependent-kinase-1-inhibitors-ic50-ki. | |
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