Cyclin-dependent kinase 2-associated protein 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	2-(Carbamoylamino)-5-Phenyl-N-[(3s)-Piperidin-3-Yl]thiophene-3-Carboxamide	IC50	5100.0 [1]
	(S)-1-(3-(Piperidin-3-ylcarbamoyl)-5-(4-(piperidine-1-carbonyl)phenyl)thiophen-2-yl)urea	IC50	10800.0 [1]
	1-(3-((S)-Piperidin-3-ylcarbamoyl)-5-(3-chlorophenyl)thiophen-2-yl)urea	IC50	8800.0 [1]
	(S)-1-(5-(4-Fluorophenyl)-3-(piperidin-3-ylcarbamoyl)thiophen-2-yl)urea	IC50	3300.0 [1]
	2-(Carbamoylamino)-5-(4-Chlorophenyl)-N-[(3s)-Piperidin-3-Yl]thiophene-3-Carboxamide	IC50	3700.0 [1]
	1-(5-(4-(2-(Diethylamino)ethoxy)phenyl)-3-(pyrrolidin-3-ylcarbamoyl)thiophen-2-yl)urea	IC50	100000.0 [1]
	1-(5-(4-(2-(Diethylamino)ethoxy)phenyl)-3-(piperidin-3-ylcarbamoyl)thiophen-2-yl)urea	IC50	4800.0 [1]
	1-(5-(4-(2-(Diethylamino)ethoxy)phenyl)-3-((3-(hydroxymethyl)phenyl)carbamoyl)thiophen-2-yl)urea	IC50	100000.0 [1]
	1-(5-(4-(2-(Diethylamino)ethoxy)phenyl)-3-(pyridin-3-ylcarbamoyl)thiophen-2-yl)urea	IC50	44000.0 [1]
	1-(5-(4-(2-(Diethylamino)ethoxy)phenyl)-3-(piperidin-4-ylcarbamoyl)thiophen-2-yl)urea	IC50	69000.0 [1]
	2-(Carbamoylamino)-5-[3-[2-(diethylamino)ethoxy]phenyl]-N-piperidin-3-ylthiophene-3-carboxamide	IC50	27000.0 [1]
	2-(Carbamoylamino)-5-[3-[2-(diethylamino)ethoxy]phenyl]-N-[(3S)-piperidin-3-yl]thiophene-3-carboxamide	IC50	3600.0 [1]
	(S)-1-(5-(4-Hydroxyphenyl)-3-(piperidin-3-ylcarbamoyl)thiophen-2-yl)urea	IC50	10200.0 [1]
	1-(3-((S)-Piperidin-3-ylcarbamoyl)-5-(3-fluorophenyl)thiophen-2-yl)urea	IC50	5600.0 [1]
	(S)-1-(3-(Piperidin-3-ylcarbamoyl)-5-p-tolylthiophen-2-yl)urea	IC50	5500.0 [1]
	(S)-1-(5-(4-Cyanophenyl)-3-(piperidin-3-ylcarbamoyl)thiophen-2-yl)urea	IC50	3600.0 [1]
	(S)-1-(3-(Piperidin-3-ylcarbamoyl)-5-(4-(trifluoromethyl)phenyl)thiophen-2-yl)urea	IC50	5400.0 [1]
	(S)-1-(5-(4-(Dimethylamino)phenyl)-3-(piperidin-3-ylcarbamoyl)thiophen-2-yl)urea	IC50	8400.0 [1]
	(S)-1-(5-(4-(Methylsulfonyl)phenyl)-3-(piperidin-3-ylcarbamoyl)thiophen-2-yl)urea	IC50	2200.0 [1]
	1-(3-((S)-Piperidin-3-ylcarbamoyl)-5-(thiophen-2-yl)thiophen-2-yl)urea	IC50	5600.0 [1]
	1-(3-((S)-Piperidin-3-ylcarbamoyl)-5-(thiophen-3-yl)thiophen-2-yl)urea	IC50	5300.0 [1]
	1-(3-((S)-Piperidin-3-ylcarbamoyl)-5-(pyridin-3-yl)thiophen-2-yl)urea	IC50	3300.0 [1]
	(S)-1-(3-(Piperidin-3-ylcarbamoyl)-5-(pyridin-4-yl)thiophen-2-yl)urea	IC50	1800.0 [1]
	(S)-1-(5-(4-(Dimethylcarbamoyl)phenyl)-3-(piperidin-3-ylcarbamoyl)thiophen-2-yl)urea	IC50	3700.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 24 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Cyclin-dependent kinase 2-associated protein 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/cyclin-dependent-kinase-2-associated-protein-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Cyclin-dependent kinase 2-associated protein 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cyclin-dependent-kinase-2-associated-protein-1-inhibitors-ic50-ki.
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