Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Abemaciclib | IC50 | 2.0 [1] | |
| Cyc065 | IC50 | 232.0 [1] | |
| N-[5-Fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]-6-(2-methoxyethyl)-7,8-dihydro-5H-1,6-naphthyridin-2-amine | IC50 | 3.2 [1] | |
| 6-Ethyl-N-[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]-7,8-dihydro-5H-1,6-naphthyridin-2-amine | IC50 | 1.5 [1] | |
| 6-(2-Fluoroethyl)-N-[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]-7,8-dihydro-5H-1,6-naphthyridin-2-amine | IC50 | 10.0 [1] | |
MLA | "Quest Database™ Cyclin-dependent kinase 4/G1/S-specific cyclin-E1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 15 Dec. 2025, https://www.aatbio.com/data-sets/cyclin-dependent-kinase-4-g1-s-specific-cyclin-e1-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 15). Quest Database™ Cyclin-dependent kinase 4/G1/S-specific cyclin-E1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cyclin-dependent-kinase-4-g1-s-specific-cyclin-e1-inhibitors-ic50-ki. | |
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