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Cyclin-dependent kinases regulatory subunit 1/S-phase kinase-associated protein 2 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
AdaphostinIC5036000.0 [1]
Benzenesulfonamide, 4-methyl-N-8-quinolinyl-IC502180.0 [1]
Ubiquitination-IN-1IC50170.0 [1]
N-(5-Pyridin-3-ylquinolin-8-yl)pyridine-3-sulfonamideIC501670.0 [1]
4-Methyl-N-(5-pyridin-3-ylquinolin-8-yl)benzenesulfonamideIC501730.0 [1]
N-[5-(Furan-2-yl)quinolin-8-yl]-4-methylbenzenesulfonamideIC50550.0 [1]
4-Methoxy-N-(5-pyridin-4-ylquinolin-8-yl)benzenesulfonamideIC502450.0 [1]
4-Methyl-N-(5-phenylquinolin-8-yl)benzenesulfonamideIC50540.0 [1]
4-Methoxy-N-(5-pyridin-3-ylquinolin-8-yl)benzenesulfonamideIC50580.0 [1]
N-(5-Pyridin-3-ylquinolin-8-yl)cyclopropanesulfonamideIC507160.0 [1]
N-(5-Phenylquinolin-8-yl)methanesulfonamideIC502200.0 [1]
4-Methoxy-N-(5-phenylquinolin-8-yl)benzenesulfonamideIC508020.0 [1]
N-[4-[(5-Pyridin-3-ylquinolin-8-yl)sulfamoyl]phenyl]acetamideIC5014490.0 [1]
N-(5-Pyridin-4-ylquinolin-8-yl)pyridine-3-sulfonamideIC501210.0 [1]
N-[6-(4-Methoxyphenoxy)quinolin-8-yl]-4-methylbenzenesulfonamideIC501150.0 [1]
N-(5-Pyridin-3-ylquinolin-8-yl)methanesulfonamideIC5015130.0 [1]
N-[6-(3,5-Difluorophenoxy)quinolin-8-yl]-4-methylbenzenesulfonamideIC503570.0 [1]
4-Methyl-N-(5-thiophen-3-ylquinolin-8-yl)benzenesulfonamideIC505540.0 [1]
N-[4-[(5-Pyridin-4-ylquinolin-8-yl)sulfamoyl]phenyl]acetamideIC506550.0 [1]
N-[6-(3-Cyanophenoxy)quinolin-8-yl]-4-methylbenzenesulfonamideIC501740.0 [1]
N-[5-(1-Benzothiophen-2-yl)quinolin-8-yl]-4-methylbenzenesulfonamideIC507840.0 [1]
N-(5-Phenylquinolin-8-yl)cyclopropanesulfonamideIC5012100.0 [1]
N-(5-Pyridin-4-ylquinolin-8-yl)cyclopropanesulfonamideIC5010940.0 [1]
N-[4-[(5-Phenylquinolin-8-yl)sulfamoyl]phenyl]acetamideIC507600.0 [1]
N-(5-Phenylquinolin-8-yl)pyridine-3-sulfonamideIC502200.0 [1]
N-(5-Phenylquinolin-8-yl)-3-(trifluoromethyl)benzenesulfonamideIC506700.0 [1]
N-(5-Bromoquinolin-8-yl)-4-methylbenzenesulfonamideIC50840.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Cyclin-dependent kinases regulatory subunit 1/S-phase kinase-associated protein 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.10 May2024https://www.aatbio.com/data-sets/cyclin-dependent-kinases-regulatory-subunit-1-s-phase-kinase-associated-protein-2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 10). Quest Database™ Cyclin-dependent kinases regulatory subunit 1/S-phase kinase-associated protein 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cyclin-dependent-kinases-regulatory-subunit-1-s-phase-kinase-associated-protein-2-inhibitors-ic50-ki.
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