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Cysteinyl leukotriene receptor 1 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
MontelukastIC500.5 [1], 0.78 [2], 2.3 [3]
MontelukastKi1.14 [1]
ZafirlukastIC501.8 [1], 1.9 [2], 14.0 [3]
ZafirlukastKi0.86 [1]
Leukotriene D4IC500.7 [1], 7.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseCysteinyl leukotriene receptor 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.5 Dec2025https://www.aatbio.com/data-sets/cysteinyl-leukotriene-receptor-1-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 5). Quest DatabaseCysteinyl leukotriene receptor 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cysteinyl-leukotriene-receptor-1-inhibitors-ic50-ki.
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