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Cytochrome P450 19A1 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
AminoglutethimideIC509000.0 [1]
AminoglutethimideKi680.0 [1]
FadrozoleIC5030.0 [1]
FadrozoleKi0.05 [1], 0.6 [2], 1.5 [3]
LetrozoleIC505.3 [1]
LetrozoleKi0.02 [1], 2.2 [2]
FormestaneIC50370.0 [1]
FormestaneKi27.0 [1], 43.0 [2], 50.0 [3], 54.0 [4], 542.0 [5]
Androst-4-en-17-oneIC50110.0 [1]
Androst-4-en-17-oneKi6.8 [1]
KetoconazoleIC501300.0 [1]
KetoconazoleKi398.11 [1]
AnastrozoleIC508.0 [1]
AnastrozoleKi0.13 [1]
NaringeninIC501000.0 [1]
Biochanin AIC5034000.0 [1]
Biochanin AKi12000.0 [1]
Androsta-1,4-diene-3,17-dioneIC50530.0 [1]
Androsta-1,4-diene-3,17-dioneKi43.0 [1], 120.0 [2], 260.0 [3]
ExemestaneIC5042.5 [1], 50.0 [2], 230.0 [3], 900.0 [4]
ExemestaneKi10.2 [1], 26.0 [2]
RogletimideIC505000.0 [1], 10000.0 [2], 45000.0 [3]
RogletimideKi1100.0 [1], 14000.0 [2]
2H-1-Benzopyran-2-one, 4-(1H-imidazol-1-ylmethyl)-7-phenoxy-IC5051.0 [1]
4-Imidazol-1-ylmethyl-1-nitro-xanthen-9-oneIC5040.0 [1]
3-Ethyl-1-n-octyl-3-(4-pyridyl)piperidine-2,6-dioneIC50800.0 [1], 5000.0 [2], 9000.0 [3]
3-Ethyl-1-n-octyl-3-(4-pyridyl)piperidine-2,6-dioneKi120.0 [1], 480.0 [2]
ResveratrolIC5025000.0 [1], 25400.0 [2]
ResveratrolKi41670.0 [1]
ChrysinIC501.0 [1], 500.0 [2], 800.0 [3], 1500.0 [4]
ChrysinKi2600.0 [1]
E-NorendoxifenIC5076.8 [1], 90.0 [2], 102.0 [3]
E-NorendoxifenKi48.0 [1]
19-Hydroxy-4-androsten-17-oneIC5049.0 [1], 270.0 [2]
19-Hydroxy-4-androsten-17-oneKi5.8 [1], 12.5 [2], 13.0 [3]
3alpha,4alpha-Epoxy-5alpha-androstan-17-oneIC50145.0 [1], 180.0 [2]
3alpha,4alpha-Epoxy-5alpha-androstan-17-oneKi38.0 [1]
(7R,8R,9S,10R,13S,14S)-10,13-Dimethyl-7-prop-2-enyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-3,17-dioneIC50470.0 [1]
(7R,8R,9S,10R,13S,14S)-10,13-Dimethyl-7-prop-2-enyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-3,17-dioneKi45.0 [1]
(8R,9S,10S,13S,14S)-10-(Hydroxymethyl)-13-methyl-1,2,3,4,7,8,9,11,12,14,15,16-dodecahydrocyclopenta[a]phenanthren-17-oneIC506900.0 [1]
(8R,9S,10S,13S,14S)-10-(Hydroxymethyl)-13-methyl-1,2,3,4,7,8,9,11,12,14,15,16-dodecahydrocyclopenta[a]phenanthren-17-oneKi1000.0 [1]
AndrostenedioneIC50260.0 [1], 300.0 [2]
AndrostenedioneKi20.0 [1], 35.0 [2]
ApigeninIC50900.0 [1], 1000.0 [2], 1200.0 [3], 10000.0 [4]
FlavanoneIC508000.0 [1], 28000.0 [2], 28500.0 [3]
4-[(5r)-5,6,7,8-Tetrahydroimidazo[1,5-A]pyridin-5-Yl]benzonitrileIC50680.0 [1], 794.33 [2], 2290.87 [3], 6000.0 [4]
Fadrozole hydrochlorideIC500.03 [1], 6.4 [2], 30.0 [3]
Fadrozole hydrochlorideKi1.5 [1]
RivizorIC501.38 [1], 1.41 [2], 29.0 [3], 44.2 [4]
PlomestaneIC5056.2 [1]
PlomestaneKi4.0 [1], 6.2 [2], 15.2 [3]
YM511 (pharmaceutical)IC500.12 [1], 0.5 [2]
NorendoxifenIC5030.0 [1], 1029.0 [2]
NorendoxifenKi442.0 [1]
Androst-5-en-17-oneIC50660.0 [1]
Androst-5-en-17-oneKi120.0 [1]
4-(1H-Imidazol-1-ylmethyl)benzonitrileIC507.0 [1], 15.0 [2], 1096.48 [3], 1200.0 [4]
4-[4-Cyanophenyl(1H-1-imidazolyl)methyl]benzonitrileIC503.0 [1], 3.5 [2], 4.0 [3], 18.2 [4]
4-Bromo-1-imidazol-1-ylmethyl-xanthen-9-oneIC50933.25 [1], 940.0 [2]
3-((1H-Imidazol-1-yl)methyl)-9H-xanthen-9-oneIC50389.05 [1], 390.0 [2]
2-Phenyl-7-methoxy-3-(1H-imidazole-1-ylmethyl)chromoneIC50549.54 [1], 550.0 [2]
1-Imidazol-1-ylmethyl-9-oxo-9H-xanthene-4-carbonitrileIC502290.87 [1], 2300.0 [2]
1-Imidazol-1-ylmethyl-4-nitro-xanthen-9-oneIC50970.0 [1], 977.24 [2]
(7Z)-6-(4-Chlorophenyl)-7-(pyridin-4-ylmethylidene)-5,6-dihydroindolizin-8-oneIC50150.0 [1], 200.0 [2]
(7Z)-6-(4-Chlorophenyl)-7-(pyridin-4-ylmethylidene)-5,6-dihydroindolizin-8-oneKi10.3 [1]
4-Imidazol-1-ylmethyl-9-oxo-9H-xanthene-1-carbonitrileIC5042.66 [1], 43.0 [2]
1-Ethyl-5-((4-fluorophenyl)(1H-imidazol-1-yl)methyl)-1H-indoleIC5040.0 [1], 41.0 [2]
7-Benzyloxy-4-(1H-imidazol-1-ylmethyl)-2H-chromen-2-oneIC50150.0 [1], 151.36 [2]
2H-1-Benzopyran-2-one, 4-(1H-imidazol-1-ylmethyl)-7-methoxy-IC50280.0 [1], 281.84 [2]
3-(Naphthalen-2-yl)pyridineIC502000.0 [1], 5700.0 [2], 5727.0 [3]
7-(Benzyloxy)-3-phenyl-2-[(pyridin-4-ylmethyl)sulfanyl]-4H-chromen-4-oneIC50210.0 [1], 210000.0 [2]
7-(Benzyloxy)-3-phenyl-2-[(pyridin-4-ylmethyl)sulfanyl]-4H-chromen-4-oneKi220.0 [1]
(3As,3bR,9aR,9bS,11aS)-9a,11a-dimethyl-3,3a,3b,4,5,9b,10,11-octahydronaphtho[2,1-e][2]benzofuran-1,7-dioneKi260.0 [1], 390.0 [2], 410.0 [3]
3-CapabhIC5012.0 [1], 150.0 [2], 230.0 [3], 780.0 [4]
3-n-Octyl-3-(4-pyridyl)piperidine-2,6-dioneIC50330.0 [1], 600.0 [2]
3-n-Octyl-3-(4-pyridyl)piperidine-2,6-dioneKi90.0 [1], 200.0 [2]
1-(4-Aminophenyl)-3-azabicyclo[3.1.0]hexane-2,4-dioneIC501800.0 [1], 7000.0 [2], 11000.0 [3]
1-(4-Aminophenyl)-3-azabicyclo[3.1.0]hexane-2,4-dioneKi1200.0 [1]
1-(4-Amino-phenyl)-3-pentyl-3-aza-bicyclo[3.1.0]hexane-2,4-dioneIC5023.0 [1], 85.0 [2], 140.0 [3]
1-(4-Amino-phenyl)-3-pentyl-3-aza-bicyclo[3.1.0]hexane-2,4-dioneKi20.0 [1]
2-(1H-Imidazol-1-yl)-7-methoxy-3-phenyl-4H-chromen-4-oneIC50770.0 [1], 776247116628.69 [2]
2-(1H-Imidazol-1-yl)-7-methoxy-3-phenyl-4H-chromen-4-oneKi680.0 [1]
2-(1H-Imidazol-1-yl)-7-methoxy-3-(4-methoxyphenyl)-4H-chromen-4-oneIC502000.0 [1], 1949844599758.04 [2]
2-(1H-Imidazol-1-yl)-7-methoxy-3-(4-methoxyphenyl)-4H-chromen-4-oneKi1820.0 [1]
7-(Benzyloxy)-2-(1H-imidazol-1-yl)-3-phenyl-4H-chromen-4-oneIC50520.0 [1], 512861383991.37 [2]
7-(Benzyloxy)-2-(1H-imidazol-1-yl)-3-phenyl-4H-chromen-4-oneKi250.0 [1]
7-(Benzyloxy)-2-(1H-imidazol-1-yl)-3-(4-methoxyphenyl)-4H-chromen-4-oneIC504700.0 [1], 4677351412871.98 [2]
7-(Benzyloxy)-2-(1H-imidazol-1-yl)-3-(4-methoxyphenyl)-4H-chromen-4-oneKi4400.0 [1]
(E/Z)-N,N-Didesmethyl-4-hydroxy TamoxifenIC5090.0 [1], 102.2 [2]
(E/Z)-N,N-Didesmethyl-4-hydroxy TamoxifenKi77.0 [1]
XolegelIC50951.48 [1], 1600.0 [2], 2600.0 [3]
NizoralIC5016000.0 [1], 110000.0 [2]
NizoralKi65000.0 [1]
FlavoneIC508.0 [1], 8000.0 [2], 10000.0 [3]
alpha-NaphthoflavoneIC5070.0 [1], 2000.0 [2]
alpha-NaphthoflavoneKi20.0 [1]
AbirateroneIC505000.0 [1], 20000.0 [2], 50000.0 [3]
OsilodrostatIC50856.0 [1], 1584.89 [2], 6000.0 [3]
7-MethoxyflavanoneIC508000.0 [1]
7alpha-AptaKi18.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Cytochrome P450 19A1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/cytochrome-p450-19a1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Cytochrome P450 19A1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cytochrome-p450-19a1-inhibitors-ic50-ki.
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