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Cytochrome P450 26A1 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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LiarozoleIC50890.0 [1]
Methyl 3-imidazol-1-yl-2,2-dimethyl-3-[4-(naphthalen-2-ylamino)phenyl]propanoateIC503.0 [1], 30.0 [2]
N-[4-[(1R,2R)-2-(Dimethylamino)-1-imidazol-1-ylpropyl]phenyl]-1,3-benzothiazol-2-amineIC5010.0 [1]
4-((+/-)-(1H-Imidazol-1-yl)-(E)-retinoic acidIC502.4 [1], 6.3 [2], 10.9 [3]
Methyl (2E,4E,6E,8E)-9-(3-imidazol-1-yl-2,6,6-trimethylcyclohexen-1-yl)-3,7-dimethylnona-2,4,6,8-tetraenoateIC5040.0 [1], 200.0 [2], 215.0 [3]
1-Imidazol-1-yl-N,N-dimethyl-1-(6-phenylmethoxynaphthalen-2-yl)propan-2-amineIC5050.0 [1]
(2E,4E,6E,8E)-1-Imidazol-1-yl-9-(3-imidazol-1-yl-2,6,6-trimethylcyclohexen-1-yl)-3,7-dimethylnona-2,4,6,8-tetraen-1-oneIC505.2 [1], 10.0 [2], 24.7 [3]
(2E,4E,6E,8E)-N-(4-Hydroxyphenyl)-9-(3-imidazol-1-yl-2,6,6-trimethylcyclohexen-1-yl)-3,7-dimethylnona-2,4,6,8-tetraenamideIC5024.0 [1], 56.0 [2]
(R)-TalarozoleIC504.0 [1], 5.0 [2]
3-[6-(2-Dimethylamino-1-imidazol-1-yl-propyl)-naphthalen-2-yloxy]-2,2-dimethyl-propionic acidIC5046.0 [1], 3300.0 [2]
[4-(Imidazol-1-yl-phenyl-methyl)-phenyl]-naphthalen-2-yl-amineIC50500.0 [1]
Methyl 2,2-dimethyl-3-[4-(naphthalen-2-ylamino)phenyl]-3-(1,2,4-triazol-1-yl)propanoateIC500.3 [1], 0.35 [2]
Methyl 3-(4-anilinophenyl)-3-imidazol-1-yl-2,2-dimethylpropanoateIC5010.0 [1]
Methyl 3-[4-(1,3-benzodioxol-5-ylamino)phenyl]-3-imidazol-1-yl-2,2-dimethylpropanoateIC508.0 [1]
Methyl (2E,4E,6E,8E)-9-[(3R)-3-imidazol-1-yl-2,6,6-trimethylcyclohexen-1-yl]-3,7-dimethylnona-2,4,6,8-tetraenoateIC50680.0 [1], 6000.0 [2]
BexaroteneIC5013500.0 [1]
TalarozoleIC505.1 [1]
CID 127019IC507800.0 [1]
CID 10389639IC5060.0 [1]
4-(2-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)-(1,3)dithiolan-2-yl)benzoic acidIC501300.0 [1]
6-(5,5,8,8-Tetramethyl-6,7-dihydronaphthalene-2-carbonyl)naphthalene-2-carboxylic acidIC501630.0 [1]
4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-naphthalene-2-carbonyl)-benzoic acidIC5025000.0 [1]
CID 44547183IC500.35 [1]
Methyl 3-(4-anilinophenyl)-2,2-dimethyl-3-(1,2,4-triazol-1-yl)propanoateIC5013.0 [1]
(E)-3-[4-(5,5,8,8-Tetramethyl-6,7-dihydronaphthalene-2-carbonyl)phenyl]prop-2-enoic acidIC504700.0 [1]
2-[4-[[6-[2-(Dimethylamino)-1-imidazol-1-ylpropyl]naphthalen-2-yl]oxymethyl]phenyl]acetic acidIC5025.0 [1]
3-[6-(2-Dimethylamino-1-imidazol-1-yl-propyl)-naphthalen-2-yloxymethyl]-benzoic acidIC506.3 [1]
3-[6-[(1R,2R)-2-(Dimethylamino)-1-imidazol-1-ylbutyl]naphthalen-2-yl]oxy-2,2-dimethylpropanoic acidIC501.3 [1]
3-[6-(2-Dimethylamino-1-imidazol-1-yl-propyl)-naphthalen-2-yloxy]-2,2-dimethyl-propionamideIC5047.0 [1]
3-[6-(2-Dimethylamino-1-imidazol-1-yl-propyl)-naphthalen-2-yloxy]-2,2,N,N-tetramethyl-propionamideIC5035.0 [1]
3-[6-(2-Dimethylamino-1-imidazol-1-yl-propyl)-naphthalen-2-yloxy]-2,2,N-trimethyl-propionamideIC5054.0 [1]
4-[6-(2-Dimethylamino-1-imidazol-1-yl-propyl)-naphthalen-2-yloxymethyl]-benzoic acid methyl esterIC5085.0 [1]
1-[6-(2,2-Dimethylpropoxy)naphthalen-2-yl]-1-imidazol-1-yl-N,N-dimethylpropan-2-amineIC5073.0 [1]
3-[6-(2-Dimethylamino-1-imidazol-1-yl-propyl)-naphthalen-2-yloxymethyl]-benzoic acid methyl esterIC5018.0 [1]
1-Imidazol-1-yl-N,N-dimethyl-1-[6-[(4-nitrophenyl)methoxy]naphthalen-2-yl]propan-2-amineIC5077.0 [1]
1-Imidazol-1-yl-N,N-dimethyl-1-[6-[[4-[(2-methylpropan-2-yl)oxy]phenyl]methoxy]naphthalen-2-yl]propan-2-amineIC5086.0 [1]
Methyl 2-[4-[[6-[2-(dimethylamino)-1-imidazol-1-ylpropyl]naphthalen-2-yl]oxymethyl]phenyl]acetateIC50100.0 [1]
4-[[6-[2-(Dimethylamino)-1-imidazol-1-ylpropyl]naphthalen-2-yl]oxymethyl]benzonitrileIC5071.0 [1]
1-[[6-[(1R,2R)-2-[Ethyl(methyl)amino]-1-imidazol-1-ylpropyl]naphthalen-2-yl]oxymethyl]cyclopentane-1-carboxylic acidIC504.2 [1]
4-[6-(2-Dimethylamino-1-imidazol-1-yl-propyl)-naphthalen-2-yloxymethyl]-benzoic acidIC5012.0 [1]
3-[4-(5,5,8,8-Tetramethyl-6,7-dihydronaphthalene-2-carbonyl)phenyl]propanoic acidIC505000.0 [1]
2-[4-[(5,5,8,8-Tetramethyl-6,7-dihydronaphthalen-2-yl)sulfonyl]phenyl]acetic acidIC505000.0 [1]
3-[(5-Tert-butyl-2-methylfuran-3-carbonyl)amino]-3-(3-nitrophenyl)propanoic acidIC503040.0 [1]
3-[(5-Tert-butyl-2-methylfuran-3-carbonyl)amino]-3-(4-methylphenyl)propanoic acidIC503260.0 [1]
3-[(5-Tert-butyl-2-methylfuran-3-carbonyl)amino]-3-(3,4-dichlorophenyl)propanoic acidIC502620.0 [1]
3-[(5-Tert-butyl-2-methylfuran-3-carbonyl)amino]-3-(3-fluorophenyl)propanoic acidIC502810.0 [1]
3-[(5-Tert-butyl-2-methylfuran-3-carbonyl)amino]-3-(4-chlorophenyl)propanoic acidIC503020.0 [1]
3-[(5-Tert-butyl-2-methylfuran-3-carbonyl)amino]-3-(4-propan-2-ylphenyl)propanoic acidIC505070.0 [1]
3-(3,4-Dichlorophenyl)-3-[(2,5-dimethylfuran-3-carbonyl)amino]propanoic acidIC502830.0 [1]
3-[(2,5-Dimethylfuran-3-carbonyl)amino]-3-(4-methylphenyl)propanoic acidIC503090.0 [1]
3-(4-Chlorophenyl)-3-[(2,5-dimethylfuran-3-carbonyl)amino]propanoic acidIC502730.0 [1]
3-[(2,5-Dimethylfuran-3-carbonyl)amino]-3-(4-propan-2-ylphenyl)propanoic acidIC504020.0 [1]
3-[(2,5-Dimethylfuran-3-carbonyl)amino]-3-(3-methylphenyl)propanoic acidIC503140.0 [1]
3-(2-Bromophenyl)-3-[(2,5-dimethylfuran-3-carbonyl)amino]propanoic acidIC502340.0 [1]
3-(2-Bromophenyl)-3-[(5-tert-butyl-2-methyl-1-propylpyrrole-3-carbonyl)amino]propanoic acidIC503130.0 [1]
3-[(5-Tert-butyl-2-methyl-1-propylpyrrole-3-carbonyl)amino]-3-(4-tert-butylphenyl)propanoic acidIC505190.0 [1]
3-[(5-Tert-butyl-2-methyl-1-propylpyrrole-3-carbonyl)amino]-3-(2-nitrophenyl)propanoic acidIC503350.0 [1]
3-[(5-Tert-butyl-2-methyl-1-propylpyrrole-3-carbonyl)amino]-3-(4-methoxyphenyl)propanoic acidIC503480.0 [1]
3-[(5-Chloro-3-methyl-1-phenylpyrazole-4-carbonyl)amino]-3-(3,4-dichlorophenyl)propanoic acidIC502070.0 [1]
3-(2-Bromophenyl)-3-[(5-chloro-3-methyl-1-phenylpyrazole-4-carbonyl)amino]propanoic acidIC501360.0 [1]
3-(4-Tert-butylphenyl)-3-[(5-chloro-3-methyl-1-phenylpyrazole-4-carbonyl)amino]propanoic acidIC503220.0 [1]
3-(3-Bromophenyl)-3-[(5-chloro-3-methyl-1-phenylpyrazole-4-carbonyl)amino]propanoic acidIC501870.0 [1]
3-[(5-Tert-butyl-2-methylfuran-3-carbonyl)amino]-3-phenylpropanoic acidIC503210.0 [1]
3-[4-[2-(5,5,8,8-Tetramethyl-6,7-dihydronaphthalen-2-yl)-1,3-dithiolan-2-yl]phenyl]propanoic acidIC50270.0 [1]
2-[4-[(5,5,8,8-Tetramethyl-6,7-dihydronaphthalen-2-yl)sulfanyl]phenyl]acetic acidIC5010600.0 [1]
3-[4-[(5,5,8,8-Tetramethyl-6,7-dihydronaphthalen-2-yl)sulfonyl]phenyl]propanoic acidIC505000.0 [1]
(E)-3-[4-[2-(5,5,8,8-Tetramethyl-6,7-dihydronaphthalen-2-yl)-1,3-dioxolan-2-yl]phenyl]prop-2-enoic acidIC50240.0 [1]
3-[4-[2-(5,5,8,8-Tetramethyl-6,7-dihydronaphthalen-2-yl)-1,3-dioxolan-2-yl]phenyl]propanoic acidIC50340.0 [1]
3-[4-[(5,5,8,8-Tetramethyl-6,7-dihydronaphthalen-2-yl)methyl]phenyl]propanoic acidIC501660.0 [1]
2-[3-[(5,5,8,8-Tetramethyl-6,7-dihydronaphthalen-2-yl)sulfonyl]phenyl]acetic acidIC505000.0 [1]
2-[3-[(5,5,8,8-Tetramethyl-6,7-dihydronaphthalen-2-yl)sulfanyl]phenyl]acetic acidIC505000.0 [1]
6-[2-(5,5,8,8-Tetramethyl-6,7-dihydronaphthalen-2-yl)-1,3-dioxolan-2-yl]naphthalene-2-carboxylic acidIC50110.0 [1]
Methyl 3-imidazol-1-yl-2-[(4-phenylbenzoyl)amino]propanoateIC50370.0 [1]
Ethyl 3-imidazol-1-yl-2-[(4-phenylbenzoyl)amino]propanoateIC50650.0 [1]
Propyl 3-imidazol-1-yl-2-[(4-phenylbenzoyl)amino]propanoateIC50790.0 [1]
Propan-2-yl 3-imidazol-1-yl-2-[(4-phenylbenzoyl)amino]propanoateIC50540.0 [1]
2-Methylpropyl 3-imidazol-1-yl-2-[(4-phenylbenzoyl)amino]propanoateIC50970.0 [1]
Methyl 2-[(5-chloro-3-methyl-1-phenylpyrazole-4-carbonyl)amino]-3-imidazol-1-ylpropanoateIC50220.0 [1]
Ethyl 2-[(5-chloro-3-methyl-1-phenylpyrazole-4-carbonyl)amino]-3-imidazol-1-ylpropanoateIC50600.0 [1]
Propyl 2-[(5-chloro-3-methyl-1-phenylpyrazole-4-carbonyl)amino]-3-imidazol-1-ylpropanoateIC50620.0 [1]
Propan-2-yl 2-[(5-chloro-3-methyl-1-phenylpyrazole-4-carbonyl)amino]-3-imidazol-1-ylpropanoateIC50460.0 [1]
2-Methylpropyl 2-[(5-chloro-3-methyl-1-phenylpyrazole-4-carbonyl)amino]-3-imidazol-1-ylpropanoateIC501020.0 [1]
Methyl 2-(1,3-benzothiazole-2-carbonylamino)-3-imidazol-1-ylpropanoateIC50410.0 [1]
Ethyl 2-(1,3-benzothiazole-2-carbonylamino)-3-imidazol-1-ylpropanoateIC50740.0 [1]
Propyl 2-(1,3-benzothiazole-2-carbonylamino)-3-imidazol-1-ylpropanoateIC50840.0 [1]
Propan-2-yl 2-(1,3-benzothiazole-2-carbonylamino)-3-imidazol-1-ylpropanoateIC50630.0 [1]
2-Methylpropyl 2-(1,3-benzothiazole-2-carbonylamino)-3-imidazol-1-ylpropanoateIC501110.0 [1]
4-[(2Z)-2-Hydroxyimino-2-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)ethoxy]benzoic acidIC503500.0 [1]
1-(5,6,7,8-Tetrahydro-5,5,8,8-tetramethyl-2-naphthyl)-2-(4-carboxyphenoxy)ethanolIC502800.0 [1]
1-(Benzofuran-2-yl(4-ethylphenyl)methyl)-1H-1,2,4-triazoleIC504500.0 [1]
N-[4-[Imidazol-1-yl(phenyl)methyl]phenyl]-1,3-benzoxazol-2-amineIC50900.0 [1]
1-(5,6,7,8-Tetrahydro-5,5,8,8-tetramethyl-2-naphthyl)-2-(4-carboxyphenoxy)ethanoneIC504000.0 [1]
3-[[6-[2-(Dimethylamino)-1-imidazol-1-ylpropyl]naphthalen-2-yl]oxymethyl]-N-methylbenzamideIC5037.0 [1]
3-[[6-[2-(Dimethylamino)-1-imidazol-1-ylpropyl]naphthalen-2-yl]oxymethyl]-N,N-dimethylbenzamideIC5014.4 [1]
Methyl 2-[4-[[6-[2-(dimethylamino)-1-imidazol-1-ylpropyl]naphthalen-2-yl]oxymethyl]phenoxy]acetateIC50153.0 [1]
3-[[6-[2-(Dimethylamino)-1-imidazol-1-ylpropyl]naphthalen-2-yl]oxymethyl]benzamideIC5048.0 [1]
2-[4-[[6-[2-(Dimethylamino)-1-imidazol-1-ylpropyl]naphthalen-2-yl]oxymethyl]phenoxy]acetic acidIC508.0 [1]
[6-(2-Dimethylamino-1-imidazol-1-yl-propyl)-naphthalen-2-yloxy]-acetic acidIC50335.0 [1]
3-[6-[(1R,2R)-2-[Cyclohexyl(methyl)amino]-1-imidazol-1-ylpropyl]naphthalen-2-yl]oxy-2,2-dimethylpropanoic acidIC50125.0 [1]
3-[6-[(1R,2R)-2-(Dimethylamino)-1-imidazol-1-ylpropyl]naphthalen-2-yl]oxy-2,2-dimethylpropanoic acidIC5020.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Cytochrome P450 26A1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 7 May. 2024, https://www.aatbio.com/data-sets/cytochrome-p450-26a1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 7). Quest Database™ Cytochrome P450 26A1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cytochrome-p450-26a1-inhibitors-ic50-ki.
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