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Cytosolic phospholipase A2 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
1-[3-(4-Octylphenoxy)-2-oxopropyl]indole-5-carboxylic acidIC5035.0 [1]
4-[3-[4-(Decyloxy)phenoxy]acetonyloxy]benzoic acidIC5011.0 [1]
3-(Methoxycarbonyl)-1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indole-5-carboxylic acidIC501.1 [1], 4.9 [2], 5.0 [3], 1400.0 [4]
1-[3-(4-Octylphenoxy)-2-oxopropyl]indole-5-carboxamideIC50120.0 [1], 770.0 [2]
1-[3-(4-Octylphenoxy)-2-oxopropyl]indole-6-carboxylic acidIC501100.0 [1], 4700.0 [2]
3-Formyl-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-5-carboxylic acidIC509.7 [1], 16.0 [2], 380.0 [3]
3-Acetyl-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-5-carboxylic acidIC506.4 [1], 12.0 [2], 16.0 [3], 1000.0 [4]
3-Cyano-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-5-carboxylic acidIC5011.0 [1], 15.0 [2], 370.0 [3]
3-Chloro-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-5-carboxylic acidIC50110.0 [1], 120.0 [2], 1500.0 [3]
3-Tert-butyl-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-5-carboxylic acidIC50230.0 [1], 340.0 [2], 3300.0 [3]
1-[3-(4-Octylphenoxy)-2-oxopropyl]indole-3,5-dicarboxylic acidIC50560.0 [1], 890.0 [2], 6500.0 [3]
Aacocf3IC502300.0 [1]
CdibaIC502700.0 [1], 3000.0 [2]
1-[3-(4-Decyloxyphenoxy)-2-oxopropyl]indole-5-carboxylic acidIC507.8 [1], 20.0 [2], 210.0 [3]
1-[3-(4-Decoxyphenoxy)-2-oxopropyl]-3-methoxycarbonylindole-5-carboxylic acidIC500.9 [1], 4.3 [2], 570.0 [3]
1-[3-(4-Octylphenoxy)-2-oxopropyl]indole-5-carbaldehydeIC504300.0 [1], 4900.0 [2]
EfipladibIC500.54 [1], 40.0 [2]
EcopladibIC50150.0 [1]
Cpla2alpha InhibitorIC501.8 [1], 31.0 [2]
4-[2-(1-Benzhydryl-2-{2-[(benzylsulfonyl)amino]ethyl}-5-chloro-1H-indol-3-yl)ethoxy]benzoic acidIC50110.0 [1]
4-(2-(1-Benzhydryl-5-chloro-2-methyl-1H-indol-3-yl)ethylsulfonyl)benzoic acidIC50800.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-(2-phenylethylsulfonylamino)ethyl]indol-3-yl]ethoxy]benzoic acidIC50500.0 [1], 520.0 [2]
1-(3-(4-Octylphenoxy)-2-oxopropyl)-1H-indazole-5-carboxylic acidIC505.0 [1]
1-(3-(4-Octylphenoxy)-2-oxopropyl)-1H-benzo[d]imidazole-5-carboxylic acidIC50150.0 [1]
1-(3-(4-Octylphenoxy)-2-oxopropyl)-1H-benzo[d]imidazole-6-carboxylic acidIC5085.0 [1]
1-[3-(4-Octylphenoxy)-2-oxopropyl]benzotriazole-5-carboxylic acidIC5026.0 [1]
3-[3-(4-Octylphenoxy)-2-oxopropyl]benzotriazole-5-carboxylic acidIC5016.0 [1]
1-(3-(4-Octylphenoxy)-2-oxopropyl)-1H-indazole-6-carboxylic acidIC5026.0 [1]
3-Methoxy-4-(1-benzhydryl-6-chloro-1H-indole-3-ylmethyl)benzoic acidIC50800.0 [1], 160000.0 [2]
1-(Carboxymethyl)-5-[3-(4-octylphenoxy)-2-oxopropoxy]indole-2-carboxylic acidIC50300.0 [1], 1300.0 [2]
1-Methyl-5-[3-(4-octylphenoxy)-2-oxopropoxy]indole-2-carboxylic acidIC50600.0 [1], 1200.0 [2]
1-(5-Carboxypentyl)-5-[3-(4-octylphenoxy)-2-oxopropoxy]indole-2-carboxylic acidIC50500.0 [1], 600.0 [2]
1-(3-Carboxypropyl)-5-[3-(4-octylphenoxy)-2-oxopropoxy]indole-2-carboxylic acidIC50300.0 [1], 400.0 [2]
ZafirlukastIC5085000.0 [1]
AmentoflavoneIC50100000.0 [1]
PyrrophenoneIC50110.0 [1]
OchnaflavoneIC50100000.0 [1]
Methoxy arachidonyl fluorophosphonateIC50640.0 [1]
4-[3-[1-Benzhydryl-5-chloro-2-[2-[(2,6-dimethylphenyl)methylsulfonylamino]ethyl]indol-3-yl]propyl]benzoic acidIC5010.0 [1]
4-(2-Oxohexadecanamido)butanoic acidIC504400.0 [1]
CID 45102612IC5012.0 [1]
4-(2-Oxo-3-(4-(5-phenylpentylthio)phenoxy)propoxy)benzoic acidIC5040.0 [1]
3-(5-Carboxypentanoyl)-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-5-carboxylic acidIC5022.0 [1]
3-[(1E,3Z,5E,7E)-1-Carboxy-2,6-dimethyl-8-(2,6,6-trimethylcyclohexen-1-yl)octa-1,3,5,7-tetraen-3-yl]benzoic acidIC5040000.0 [1]
2-Amino-2-(hydroxymethyl)propane-1,3-diol;3-[1-(4-phenoxyphenyl)-3-(2-phenylethyl)indol-5-yl]propanoic acidIC5020.0 [1]
Carbamic acid,N-[6-(2-methyl-4,5-diphenyl-1H-imidazol-1-yl)hexyl]-,2-fluorophenyl esterKi15000.0 [1]
6-(4-Oxo-2-phenyl-chromen-6-yl)-2-phenyl-chromen-4-oneIC5048100.0 [1]
4-[3-[1-Benzhydryl-5-chloro-2-[2-[(2-methylphenyl)methylsulfonylamino]ethyl]indol-3-yl]propyl]benzoic acidIC5026.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-(cyclohexylmethylsulfonylamino)ethyl]indol-3-yl]ethoxy]benzoic acidIC50200.0 [1]
4-[2-[2-[2-(Benzenesulfonamido)ethyl]-1-benzhydryl-5-chloroindol-3-yl]ethoxy]benzoic acidIC503000.0 [1]
4-[(Z)-(2,4-Dioxo-1,3-thiazolidin-5-ylidene)methyl]-N-[[(2S,4R)-1-[2-(4-fluorobenzoyl)benzoyl]-4-[(2-phenylphenyl)methoxy]pyrrolidin-2-yl]methyl]benzamideIC5078.0 [1]
N-[[(2S,4R)-1-(2-Benzoylbenzoyl)-4-[(2-phenylphenyl)methoxy]pyrrolidin-2-yl]methyl]-4-[(Z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]benzamideIC50165.0 [1]
1-[3-(4-Octylphenoxy)-2-oxopropyl]indole-2-carboxylic acidIC508000.0 [1]
Methyl 1-[3-(4-octylphenoxy)-2-oxopropyl]indole-5-carboxylateIC5010000.0 [1]
1-[3-(4-Octylphenoxy)-2-oxopropyl]indole-3-carboxylic acidIC5010000.0 [1]
1-[3-(4-Octylphenoxy)-2-oxopropyl]indole-4-carboxylic acidIC5010000.0 [1]
1-[3-(4-Octylphenoxy)-2-oxopropyl]indole-5-carbonitrileIC5010000.0 [1]
2-{4-[4-(4-Oxo-4H-chromen-2-yl)phenyl]phenyl}-4H-chromen-4-oneIC506000.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-[(2-chlorophenyl)methylsulfonylamino]ethyl]indol-3-yl]ethoxy]benzoic acidIC5052.0 [1]
6-[3-(4-Oxo-4H-chromen-2-yl)-phenyl]-2-phenyl-chromen-4-oneIC5016800.0 [1]
3-(3-Carboxypropanoyl)-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-5-carboxylic acidIC50210.0 [1]
2-{4-[3-(4-Oxo-4H-chromen-2-yl)phenyl]phenyl}-4H-chromen-4-oneIC5038700.0 [1]
6-[4-(4-Oxo-4H-chromen-2-yl)-phenyl]-2-phenyl-chromen-4-oneIC5011900.0 [1]
3-(4-(4-Oxo-4H-chromen-2-yl)phenyl)-2-phenyl-4H-chromen-4-oneIC508420.0 [1]
4-[3-[1-Benzhydryl-5-chloro-2-[2-[(2-methoxyphenyl)sulfonylamino]ethyl]indol-3-yl]propyl]benzoic acidIC50100.0 [1]
1-Imidazol-1-yl-3-(4-octylphenoxy)propan-2-oneIC50500.0 [1]
1-Benzimidazol-1-yl-3-(4-octylphenoxy)propan-2-oneIC5010000.0 [1]
1-Benzotriazol-1-yl-3-(4-octylphenoxy)propan-2-oneIC502200.0 [1]
3-Butanoyl-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-5-carboxylic acidIC5010.0 [1]
3-Hexanoyl-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-5-carboxylic acidIC5071.0 [1]
1-(4-Octylphenoxy)-3-(pyrazol-1-yl)propan-2-oneIC5010000.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-(methanesulfonamido)ethyl]indol-3-yl]ethoxy]benzoic acidIC50650.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-[2-(2-sulfanylideneimidazolidin-1-yl)ethylsulfonylamino]ethyl]indol-3-yl]ethoxy]benzoic acidIC50750.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-[(2,6-dimethylphenyl)sulfanylmethylsulfonylamino]ethyl]indol-3-yl]ethoxy]benzoic acidIC50330.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-[2-(4-methylpyrazol-1-yl)ethylsulfonylamino]ethyl]indol-3-yl]ethoxy]benzoic acidIC50760.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-[2-(4-pyridin-2-ylpiperazin-1-yl)ethylsulfonylamino]ethyl]indol-3-yl]ethoxy]benzoic acidIC50290.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-[2-(3-methylpyrazol-1-yl)ethylsulfonylamino]ethyl]indol-3-yl]ethoxy]benzoic acidIC50510.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-(2-morpholin-4-ylethylsulfonylamino)ethyl]indol-3-yl]ethoxy]benzoic acidIC50390.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-[2-(1,3-thiazolidin-3-yl)ethylsulfonylamino]ethyl]indol-3-yl]ethoxy]benzoic acidIC50330.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-[(4-chlorophenyl)methylsulfonylamino]ethyl]indol-3-yl]ethoxy]benzoic acidIC50120.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-[(3,5-dichlorophenyl)methylsulfonylamino]ethyl]indol-3-yl]ethoxy]benzoic acidIC50190.0 [1]
4-[3-[1-Benzhydryl-5-chloro-2-[2-[2-(3,5-dimethylpyrazol-1-yl)ethylsulfonylamino]ethyl]indol-3-yl]propyl]benzoic acidIC50300.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-(methylsulfonylmethylsulfonylamino)ethyl]indol-3-yl]ethoxy]benzoic acidIC50150.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-(phenylsulfanylmethylsulfonylamino)ethyl]indol-3-yl]ethoxy]benzoic acidIC50190.0 [1]
4-[2-[1-Benzhydryl-2-[2-(benzylsulfonylamino)ethyl]-5-morpholin-4-ylindol-3-yl]ethoxy]benzoic acidIC50600.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-(2-pyrazol-1-ylethylsulfonylamino)ethyl]indol-3-yl]ethoxy]benzoic acidIC50320.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-[2-(1,2,4-triazol-1-yl)ethylsulfonylamino]ethyl]indol-3-yl]ethoxy]benzoic acidIC50410.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-[2-(triazol-1-yl)ethylsulfonylamino]ethyl]indol-3-yl]ethoxy]benzoic acidIC50500.0 [1]
4-[3-[1-Benzhydryl-5-chloro-2-[2-(2-morpholin-4-ylethylsulfonylamino)ethyl]indol-3-yl]propyl]benzoic acidIC50200.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-[2-(3,5-dimethylpyrazol-1-yl)ethylsulfonylamino]ethyl]indol-3-yl]ethoxy]benzoic acidIC50450.0 [1]
4-[3-[1-Benzhydryl-5-chloro-2-[2-[2-(2,6-dimethylpiperidin-1-yl)ethylsulfonylamino]ethyl]indol-3-yl]propyl]benzoic acidIC50100.0 [1]
4-[2-[1-Benzhydryl-5-chloro-2-[2-[(3,5-dichlorophenyl)sulfanylmethylsulfonylamino]ethyl]indol-3-yl]ethoxy]benzoic acidIC50200.0 [1]
(E)-3-[4-[(Z)-(2,4-Dioxo-1,3-thiazolidin-5-ylidene)methyl]phenyl]-N-[[(2S,4R)-1-[2-(4-fluorobenzoyl)benzoyl]-4-[2-methylpropyl-[(2-phenylphenyl)methyl]amino]pyrrolidin-2-yl]methyl]prop-2-enamideIC503.1 [1]
N-[[(2S,4R)-1-[2-(4-Fluorobenzoyl)benzoyl]-4-[(2-phenylphenyl)methylsulfanyl]pyrrolidin-2-yl]methyl]-4-[(Z)-(4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]benzamideIC5072.0 [1]
N-[[(2S,4R)-1-[2-(2,4-Difluorobenzoyl)benzoyl]-4-[2-methylpropyl-[(2-phenylphenyl)methyl]amino]pyrrolidin-2-yl]methyl]-4-[(Z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]benzamideIC506.2 [1]
N-[[(2S,4R)-4-[2-Bromo-6-(2-methylpropyl)phenoxy]-1-[2-(4-fluorobenzoyl)benzoyl]pyrrolidin-2-yl]methyl]-4-[(Z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]benzamideIC5038.0 [1]
4-[(Z)-(2,4-Dioxo-1,3-thiazolidin-5-ylidene)methyl]-N-[[(2S,4R)-1-[2-(4-fluorobenzoyl)benzoyl]-4-[2-methylpropyl-[(2-phenylphenyl)methyl]amino]pyrrolidin-2-yl]methyl]benzamideIC5021.0 [1]
N-[[(2S,4R)-1-[2-(4-Fluorobenzoyl)benzoyl]-4-[(2-phenylphenyl)methoxy]pyrrolidin-2-yl]methyl]-4-[(Z)-(4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]benzamideIC5090.0 [1]
N-[[(2S,4R)-4-[2-Bromo-6-(2-methylpropyl)phenoxy]-1-[2-(2,4-difluorobenzoyl)benzoyl]pyrrolidin-2-yl]methyl]-4-[(Z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]benzamideIC5022.0 [1]
N-[[(2S,4R)-1-[2-(2,4-Difluorobenzoyl)benzoyl]-4-[2-(2-methylpropyl)-6-(2-propan-2-ylphenyl)phenoxy]pyrrolidin-2-yl]methyl]-4-[(Z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]benzamideIC502.1 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Cytosolic phospholipase A2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/cytosolic-phospholipase-a2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Cytosolic phospholipase A2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cytosolic-phospholipase-a2-inhibitors-ic50-ki.
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