Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| [(3R)-1-[2-[1-(4-Chloropyrazol-1-yl)cyclopropyl]-1H-imidazo[4,5-b]pyridin-5-yl]piperidin-3-yl]-pyrrolidin-1-ylmethanone | IC50 | 1.3 [1], 5.5 [2], 14.0 [3], 35.9 [4] | |
| [(3R)-1-[2-[(1S)-1-(4-Chloropyrazol-1-yl)ethyl]-1H-imidazo[4,5-b]pyridin-5-yl]piperidin-3-yl]-pyrrolidin-1-ylmethanone | IC50 | 4.6 [1], 20.0 [2], 38.5 [3] | |
| [(3R)-1-[2-[(1R)-1-(4-Chloropyrazol-1-yl)ethyl]-1H-imidazo[4,5-b]pyridin-5-yl]piperidin-3-yl]-pyrrolidin-1-ylmethanone | IC50 | 5.5 [1], 33.7 [2], 34.0 [3] | |
| 2-[4-[4-[1-(Phenylcarbamoyl)indol-5-yl]phenyl]cyclohexyl]acetic acid | IC50 | 50000.0 [1] | |
| 2-[4-[4-[4-(Phenylcarbamoyl)-2,3-dihydro-1,4-benzoxazin-7-yl]phenyl]cyclohexyl]acetic acid | IC50 | 10000.0 [1] | |
MLA | "Quest Database™ Diacylglycerol O-acyltransferase 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 15 Dec. 2025, https://www.aatbio.com/data-sets/diacylglycerol-o-acyltransferase-2-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 15). Quest Database™ Diacylglycerol O-acyltransferase 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/diacylglycerol-o-acyltransferase-2-inhibitors-ic50-ki. | |
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