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Dihydroorotate dehydrogenase Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
BrequinarIC508.0 [1]
BrequinarKi12.0 [1]
TeriflunomideIC50356.0 [1]
TeriflunomideKi30.0 [1], 2700.0 [2]
Brequinar sodiumIC508.0 [1], 15.0 [2]
Brequinar sodiumKi12.0 [1]
2-({2,6-Difluoro-4-[3-(trifluoromethoxy)phenyl]phenyl}carbamoyl)cyclopent-1-ene-1-carboxylic acidIC5033.0 [1]
2-[2,3,5,6-Tetrafluoro-3'-(trifluoromethoxy)-4-biphenylylcarbamoyl]-1-cyclopentene-1-carboxylic acidIC507.0 [1]
2-(1,1-Difluoroethyl)-5-Methyl-N-[4-(Trifluoromethyl)phenyl][1,2,4]triazolo[1,5-A]pyrimidin-7-AmineIC50100000.0 [1]
2-(4-Biphenylylcarbamoyl)-1-cyclopentene-1-carboxylic acidIC50410.0 [1]
LeflunomideIC5010000.0 [1], 13000.0 [2]
VidofludimusIC50134.0 [1]
5-Methyl-n-(naphthalen-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amineIC50200000.0 [1]
5-Methyl-N-[4-(trifluoromethyl)phenyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amineIC50100000.0 [1]
CID 51347103IC50100000.0 [1]
CID 51347104IC5030000.0 [1], 100000.0 [2]
2-(2,3,5,6-Tetrafluoro-2'-methoxy-4-biphenylylcarbamoyl)-1-cyclopentene-1-carboxylic acidIC508.0 [1]
3-{[(3-Fluoro-3'-Methoxybiphenyl-4-Yl)amino]carbonyl}thiophene-2-Carboxylic AcidIC5044.0 [1]
Diethyl 2-[(dibenzothiophen-2-ylamino)methylidene]propanedioateIC5030000.0 [1]
Diethyl 2-[(dibenzothiophen-2-ylamino)methylidene]propanedioateKi3630.0 [1]
Ethyl (Z)-2-cyano-3-[(9-ethylcarbazol-3-yl)amino]prop-2-enoateIC50491000.0 [1]
Ethyl (Z)-2-cyano-3-[(9-ethylcarbazol-3-yl)amino]prop-2-enoateKi60400.0 [1]
N-[3,5-Difluoro-4-(trifluoromethyl)phenyl]-5-methyl-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amineIC501600.0 [1], 2100.0 [2]
2-(1,1-Difluoroethyl)-N-[3,5-difluoro-4-(trifluoromethyl)phenyl]-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amineIC502100.0 [1], 2700.0 [2]
(E)-2-Cyano-3-hydroxy-N-[4-(trifluoromethyl)phenyl]but-2-enamideIC50200.0 [1], 435.0 [2]
1-{2-[(3-Chloro-4-methylphenyl)amino]-4-methyl-1,3-thiazol-5-yl}ethanoneIC50930.0 [1], 3937.0 [2]
2-({[3-Fluoro-3'-(trifluoromethoxy)biphenyl-4-YL]amino}carbonyl)cyclopent-1-ene-1-carboxylic acidIC50280.0 [1]
3-N-Benzyl-1-(4-methoxyphenyl)-5-N-[4-(pyrrolidine-1-carbonyl)phenyl]pyrazole-3,5-dicarboxamideKi26.0 [1], 50000.0 [2]
1-(4-Chlorophenyl)-5-N-phenyl-3-N-(pyridin-3-ylmethyl)pyrazole-3,5-dicarboxamideKi4.0 [1], 50000.0 [2]
3-Carbamoyl-5-{3-[4-(trifluoromethyl)phenyl]phenyl}benzoic acidKi6000.0 [1], 90000.0 [2]
3-Carbamoyl-5-[3-(3-methylphenyl)phenyl]benzoic AcidKi3700.0 [1], 50000.0 [2]
3-[3-(4-Tert-butylphenyl)phenyl]-5-carbamoylbenzoic acidKi4000.0 [1], 90000.0 [2]
1-(4-Chlorophenyl)-3-N-[(4-methylphenyl)methyl]-5-N-phenylpyrazole-3,5-dicarboxamideKi32.0 [1], 50000.0 [2]
1-(4-Methoxyphenyl)-3-N-(oxolan-2-ylmethyl)-5-N-[4-(pyrrolidine-1-carbonyl)phenyl]pyrazole-3,5-dicarboxamideKi331.0 [1], 50000.0 [2]
1-(4-Methoxyphenyl)-5-N-phenyl-3-N-(pyridin-3-ylmethyl)pyrazole-3,5-dicarboxamideKi12.0 [1], 5000.0 [2]
1-(4-Chlorophenyl)-5-N-(4-piperidin-1-ylphenyl)-3-N-(pyridin-3-ylmethyl)pyrazole-3,5-dicarboxamideKi8.0 [1], 50000.0 [2]
5-N-Benzyl-1-(4-methoxyphenyl)-3-N-[4-(pyrrolidine-1-carbonyl)phenyl]pyrazole-3,5-dicarboxamideKi1500.0 [1], 50000.0 [2]
3-N-Benzyl-5-N-(4-carbamoylphenyl)-1-(4-chlorophenyl)pyrazole-3,5-dicarboxamideKi6.0 [1], 50000.0 [2]
3-N-Benzhydryl-5-N-benzyl-1-(4-methoxyphenyl)pyrazole-3,5-dicarboxamideKi2400.0 [1], 50000.0 [2]
1-(4-Methoxyphenyl)-3-N-(2-methylpropyl)-5-N-[4-(pyrrolidine-1-carbonyl)phenyl]pyrazole-3,5-dicarboxamideKi138.0 [1], 50000.0 [2]
3-N-Benzyl-1-(4-chlorophenyl)-5-N-(2-methylpropyl)pyrazole-3,5-dicarboxamideKi91.0 [1], 50000.0 [2]
4-Quinolinecarboxylic acid, 2-[1,1'-biphenyl]-4-yl-6-fluoro-3-hydroxy-IC505.0 [1]
4-Quinolinecarboxylic acid, 2-[1,1'-biphenyl]-4-yl-6-fluoro-3-hydroxy-Ki40.0 [1]
Aslan003IC5015.0 [1]
2-([1,1'-Biphenyl]-4-yl)-3-methylquinoline-4-carboxylic acidIC5075.4 [1]
2-([1,1'-Biphenyl]-4-yl)-3-methylquinoline-4-carboxylic acidKi1.7 [1]
5-(Benzimidazol-1-yl)-N-propylthiophene-2-carboxamideIC5030000.0 [1]
2-Biphenyl-4-yl-1H-benzoimidazole-4-carboxylic acidIC50750.0 [1], 795.0 [2]
2-(1,1-Difluoroethyl)-N-[3-fluoro-4-(trifluoromethyl)phenyl]-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amineIC5017000.0 [1], 45000.0 [2]
3-N-Benzyl-1-(4-chlorophenyl)-5-N-phenylpyrazole-3,5-dicarboxamideKi4.0 [1], 50000.0 [2]
2-[2,3,5,6-Tetrafluoro-4-(3-methoxyphenyl)anilino]pyridine-3-carboxylic acidIC503.0 [1]
2-[2,5-Difluoro-4-(3-methoxyphenyl)anilino]pyridine-3-carboxylic acidIC5087.9 [1], 88.0 [2]
2-[4-(3-Ethoxyphenyl)-2,6-difluoroanilino]pyridine-3-carboxylic acidIC5019.0 [1], 19.01 [2]
2-[4-(3-Cyclobutyloxyphenyl)-2,6-difluoroanilino]pyridine-3-carboxylic acidIC5089.95 [1], 90.0 [2]
2-[2-Chloro-4-(3-methoxyphenyl)anilino]pyridine-3-carboxylic acidIC50149.97 [1], 150.0 [2]
3-[4-(3-Ethoxyphenyl)-2-fluoroanilino]pyridine-4-carboxylic acidIC5019.0 [1], 19.01 [2]
3-[4-(3-Methoxyphenyl)-2-(trifluoromethoxy)anilino]pyridine-4-carboxylic acidIC5014.0 [1]
3-[2-Fluoro-4-[3-(trifluoromethoxy)phenyl]anilino]pyridine-4-carboxylic acidIC50199.99 [1], 200.0 [2]
2-[2,6-Difluoro-4-(3-methoxyphenyl)anilino]-5-ethylpyridine-3-carboxylic acidIC5011.99 [1], 12.0 [2]
2-[2-Fluoro-4-(3-methoxyphenyl)-5-methylanilino]pyridine-3-carboxylic acidIC5099.0 [1], 99.08 [2]
2-[2-Fluoro-4-[3-(trifluoromethoxy)phenyl]anilino]-5-methylpyridine-3-carboxylic acidIC50109.9 [1], 110.0 [2]
2-[2,6-Difluoro-4-(3-methoxyphenyl)anilino]-5-methylpyridine-3-carboxylic acidIC5011.99 [1], 12.0 [2]
5-Cyclopropyl-2-[2-fluoro-4-(3-methoxyphenyl)anilino]pyridine-3-carboxylic acidIC5032.96 [1], 33.0 [2]
5-Cyclopropyl-2-[4-(3-cyclopropyloxyphenyl)-2,6-difluoroanilino]pyridine-3-carboxylic acidIC506.0 [1]
2-(2,6-Difluoro-3-methyl-4-phenylanilino)pyridine-3-carboxylic acidIC505.0 [1]
2-[4-(3-Cyclopropyloxyphenyl)-2,6-difluoroanilino]pyridine-3-carboxylic acidIC5017.0 [1], 17.02 [2]
2-[2,6-Difluoro-4-(2-fluoro-3-methoxyphenyl)anilino]pyridine-3-carboxylic acidIC5052.97 [1], 53.0 [2]
5-Cyclopropyl-2-[4-(3-ethoxyphenyl)-2,5-difluoroanilino]pyridine-3-carboxylic acidIC5023.0 [1], 23.01 [2]
5-Cyclopropyl-2-[2,6-difluoro-4-[3-(trifluoromethoxy)phenyl]anilino]pyridine-3-carboxylic acidIC504.0 [1]
5-Chloro-2-(2,6-difluoro-4-phenylanilino)pyridine-3-carboxylic acidIC508.0 [1]
2-[2,6-Difluoro-4-(2-methylphenyl)anilino]pyridine-3-carboxylic acidIC5010.99 [1], 11.0 [2]
2-[4-(2-Chlorophenyl)-2,6-difluoro-3-methylanilino]pyridine-3-carboxylic acidIC504.0 [1]
2-[2,6-Difluoro-3-methyl-4-[3-(trifluoromethoxy)phenyl]anilino]pyridine-3-carboxylic acidIC506.0 [1]
2-[4-(2-Chlorophenyl)-2,6-difluoroanilino]-5-cyclopropylpyridine-3-carboxylic acidIC505.0 [1]
2-[4-(3-Ethoxyphenyl)-2-fluoroanilino]pyridine-3-carboxylic acidIC50199.99 [1], 200.0 [2]
Cyclosporin AIC5050000.0 [1]
Niflumic acidIC5017000.0 [1]
AtovaquoneIC5014500.0 [1]
ClonixinIC5013000.0 [1]
CinchophenIC50144000.0 [1]
FlunixinIC508000.0 [1]
3',4'-DihydroxyflavoneIC5012380.0 [1]
CID 51347395IC50100000.0 [1]
2-[(4-Chlorobenzyl)sulfanyl]-5-methyl[1,2,4]triazolo[1,5-a]pyrimidin-7(4H)-oneIC5039000.0 [1]
N,N-Dimethyl-N'-(5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)-benzene-1,4-diamineIC50100000.0 [1]
OxycinchophenIC5012000.0 [1]
2-((4-Methoxyphenyl)amino)benzoic acidIC5010000.0 [1]
N-(3-Chlorophenyl)-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amineIC50100000.0 [1]
2-Phenylamino-4-Methyl-5-Acetyl ThiazoleIC5010000.0 [1]
Ethyl 2-[(4-chlorophenyl)amino]-4-oxo-4,5-dihydrothiophene-3-carboxylateIC5050000.0 [1]
2-Benzylsulfanyl-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-olIC5089000.0 [1]
N-(4-Isopropylphenyl)-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amineIC50100000.0 [1]
N-(3-Fluoro-4-methylphenyl)-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amineIC50100000.0 [1]
N-(4-Chlorophenyl)-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amineIC50100000.0 [1]
2-[(2-Chlorobenzyl)thio]-5-methyl[1,2,4]triazolo[1,5-a]pyrimidin-7(4H)-oneIC5012000.0 [1]
Ethyl 2-anilino-4-oxo-4,5-dihydro-3-thiophenecarboxylateIC5050000.0 [1]
2-(4-Chloro-phenylamino)-nicotinic acidIC50400.0 [1]
Diethyl 2-(2-toluidinomethylene)malonateIC50292200.0 [1]
5-Methyl-N-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amineIC50200000.0 [1]
N-(1,3-Benzothiazol-2-yl)-3-methoxybenzamideIC506830.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Dihydroorotate dehydrogenase Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/dihydroorotate-dehydrogenase-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Dihydroorotate dehydrogenase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/dihydroorotate-dehydrogenase-inhibitors-ic50-ki.
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