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DNA-dependent protein kinase Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-oneIC501400.0 [1]
2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-oneKi6000.0 [1]
8-(4-Dibenzothienyl)-2-(4-morpholinyl)-4H-1-benzopyran-4-oneIC5028.0 [1]
8-(4-Dibenzothienyl)-2-(4-morpholinyl)-4H-1-benzopyran-4-oneKi0.65 [1]
2-(Morpholin-4-yl)-benzo[h]chromen-4-oneIC50230.0 [1]
CID 11964036IC505.0 [1]
2-(4-Morpholinyl)-4H-1-benzopyran-4-oneIC501260.0 [1], 1300.0 [2], 4300.0 [3], 10000.0 [4]
2-(4-Methoxyphenyl)-6-morpholino-4H-pyran-4-oneIC50220.0 [1]
3-Morpholino-1H-benzo[f]chromen-1-oneIC501250.0 [1], 4000.0 [2]
2-Morpholino-6-(4-methoxyphenyl)-4H-thiopyran-4-oneIC50280.0 [1]
PI-103IC502.0 [1], 14.0 [2], 48.5 [3]
6-[(E)-Hydrazinylidenemethyl]-2-oxo-5-pyridin-4-yl-1H-pyridine-3-carbonitrileIC508000.0 [1], 100000.0 [2]
2-Morpholino-4H-benzo[g]chromen-4-oneIC50390.0 [1], 400.0 [2]
2-(4-Chlorophenyl)-6-morpholin-4-yl-thiopyran-4-oneIC50530.0 [1]
2-(4-Chlorophenyl)-6-morpholino-4H-pyran-4-oneIC50180.0 [1]
2-Morpholino-6-phenyl-4H-pyran-4-oneIC501100.0 [1], 1300.0 [2]
6-Methoxy-4-morpholin-4-yl-chromen-2-oneIC501200.0 [1], 1700.0 [2], 1750.0 [3]
8-Dibenzofuran-4-yl-2-morpholin-4-ylchromen-4-oneIC5040.0 [1], 41.0 [2]
8-(Biphenyl-3-yl)-2-morpholino-4H-chromen-4-oneIC50180.0 [1]
2-Morpholino-6-phenyl-4H-thiopyran-4-oneIC50650.0 [1], 720.0 [2]
WortmanninKi120.0 [1]
IdelalisibIC506700.0 [1]
2-Morpholino-6-(thianthren-1-yl)-4H-pyran-4-oneIC501800.0 [1], 2500.0 [2]
3-Amino-6-(4-(methylsulfonyl)phenyl)-N-phenylpyrazine-2-carboxamideIC5026.0 [1], 4400.0 [2]
N-(5-(4-Chloro-3-(N-(2-hydroxyethyl)sulfamoyl)phenyl)-4-methylthiazol-2-yl)acetamideIC5064.0 [1]
N-(7,8-Dimethoxy-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl)-3-pyridinecarboxamideIC5013.0 [1]
2-Morpholino-4H-pyrimido[2,1-a]isoquinolin-4-oneIC50280.0 [1]
4-Morpholin-4-yl-chromen-2-oneIC504800.0 [1], 4820.0 [2]
CID 46244454IC5030000.0 [1]
2-(2-Methyl-morpholin-4-yl)-benzo[h]chromen-4-oneIC50190.0 [1]
8-Methoxy-2-morpholin-4-yl-chromen-4-oneIC501200.0 [1], 1800.0 [2]
3-Amino-n,6-diphenylpyrazine-2-carboxamideIC50620.0 [1], 8000.0 [2]
2-(4-Fluorophenyl)-6-morpholino-4H-pyran-4-oneIC50350.0 [1]
2-Thiomorpholino-4H-benzo[h]chromen-4-oneIC501380.0 [1]
7-Methoxy-4-morpholin-4-yl-chromen-2-oneIC505400.0 [1], 11310.0 [2]
CID 11508681IC50800.0 [1]
8-Benzo[b]thiophen-2-yl-2-morpholin-4-yl-chromen-4-oneIC50800.0 [1]
2-Morpholin-4-yl-8-thiophen-2-ylchromen-4-oneIC50700.0 [1]
2-Morpholin-4-yl-8-thiophen-3-ylchromen-4-oneIC50300.0 [1]
8-(4-Hydroxymethylphenyl)-2-morpholin-4-ylchromen-4-oneIC50600.0 [1]
2-(4-(Benzo[b]thiophen-3-yl)phenyl)-6-morpholino-4H-thiopyran-4-oneIC50160.0 [1], 330.0 [2]
2-Morpholino-6-[4-(4-methyl-1-naphthyl)phenyl]-4H-thiopyran-4-oneIC50260.0 [1]
2-Morpholino-6-(3'-hydroxy-3-biphenylyl)-4H-thiopyran-4-oneIC50920.0 [1]
2-Morpholino-6-(3-bromophenyl)-4H-thiopyran-4-oneIC50700.0 [1], 800.0 [2]
2-Morpholino-6-(4-tert-butylphenyl)-4H-thiopyran-4-oneIC50920.0 [1], 1100.0 [2]
2-Morpholino-6-(4-bromophenyl)-4H-thiopyran-4-oneIC50680.0 [1]
6-(4-Methoxyphenyl)-2-morpholin-4-ylpyridin-4-olIC50100000.0 [1]
Methyl (E)-3-[2-[3-(6-morpholin-4-yl-4-oxothiopyran-2-yl)phenyl]phenyl]prop-2-enoateIC50840.0 [1]
2-(2-Methoxyphenyl)-6-morpholino-4H-pyran-4-oneIC50310.0 [1], 380.0 [2]
2-(3-Methoxyphenyl)-6-morpholino-4H-pyran-4-oneIC50540.0 [1]
2-Morpholino-6-(4-tert-butylphenyl)-4H-pyran-4-oneIC50480.0 [1]
4H-Naphtho(1,2-b)pyran-4-one, 2-(1-piperidinyl)-IC503810.0 [1]
8-(4-Methoxyphenyl)-2-(morpholin-4-yl)-4H-1-benzopyran-4-oneIC50900.0 [1]
4-Morpholino-7-(thiophen-2-yl)-2H-chromen-2-oneIC50600.0 [1]
3-Amino-6-[4-[1-(dimethylamino)propan-2-ylsulfonyl]phenyl]-N-phenylpyrazine-2-carboxamideIC508000.0 [1]
3-Amino-6-[4-[1-(dimethylamino)propan-2-ylsulfonyl]phenyl]-N-phenylpyrazine-2-carboxamideKi6.0 [1]
2-Hydroxy-4-morpholin-4-yl-benzaldehydeIC50400.0 [1]
2-Morpholino-6-(3-fluorophenyl)-4H-pyran-4-oneIC50530.0 [1], 690.0 [2]
2-Morpholino-6-[4-(1-naphthyl)phenyl]-4H-thiopyran-4-oneIC50160.0 [1], 190.0 [2]
[(4E,6Z,8S,9S,10E,12S,13R,14S,16R)-13-Hydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-19-[5-(2-morpholin-4-yl-4-oxochromen-7-yl)oxypentylamino]-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl] carbamateIC505000.0 [1], 10000.0 [2]
CaffeineIC5010000000.0 [1]
GefitinibIC5050000.0 [1]
SorafenibIC5050000.0 [1]
SuraminIC501700.0 [1]
TrifluoperazineIC50100000.0 [1]
SunitinibIC5050000.0 [1]
DasatinibIC5050000.0 [1]
VanillinIC501500000.0 [1]
FlavoneIC5010000.0 [1]
alpha-NaphthoflavoneIC504980.0 [1]
TanespimycinIC5040000.0 [1]
Schisandrin BIC501000000000.0 [1]
PictilisibIC501230.0 [1]
BuparlisibIC506917.0 [1]
Torin 1IC506.34 [1]
AlpelisibIC509100.0 [1]
2-(4-Amino-1-isopropyl-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-1H-indol-5-olIC50410.0 [1]
Ku-0063794IC5010000.0 [1]
Torin 2IC500.5 [1]
N-[4-({3-[(3,5-Dimethoxyphenyl)amino]quinoxalin-2-yl}sulfamoyl)phenyl]-3-methoxy-4-methylbenzamideIC50150.0 [1]
IsogranulatimideIC5010000.0 [1]
TaselisibIC504800.0 [1]
Imino-methyl-[1-[6-[(3R)-3-methylmorpholin-4-yl]-2-(1H-pyrrolo[2,3-b]pyridin-4-yl)pyrimidin-4-yl]cyclopropyl]-oxo-lambda6-sulfaneIC5030000.0 [1]
PilaralisibIC504800.0 [1]
DNA-PK Inhibitor IIIIC50120.0 [1]
CB-5083IC50500.0 [1]
1-Cyclopentyl-3-(1H-pyrrolo[2,3-b]pyridin-5-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineIC5060.0 [1]
LeniolisibIC50880.0 [1]
N-[6-[6-Chloro-5-[[(4-fluorophenyl)sulfonyl]amino]-3-pyridinyl]-1,3-benzothiazol-2-yl]acetamideIC503.0 [1]
2-[[4-Amino-3-(3-hydroxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]methyl]-5-methyl-3-(2-methylphenyl)quinazolin-4-oneIC5048000.0 [1]
1-Tert-Butyl-3-Naphthalen-2-Yl-1h-Pyrazolo[3,4-D]pyrimidin-4-AmineIC50420.0 [1]
CID 59604787IC508831.0 [1]
2-Methyl-2-[4-(2-oxo-9-quinolin-3-yl-4H-[1,3]oxazino[5,4-c]quinolin-1-yl)phenyl]propanenitrileIC5036.0 [1]
6-NitroveratraldehydeIC5015000.0 [1]
(S)-2-(2-(2-Methylindolin-1-yl)-2-oxoethyl)-6-morpholinopyrimidin-4(3H)-oneIC502000.0 [1]
DNA-PK Inhibitor VIC50270.0 [1]
3-Morpholino-5-phenylcyclohex-2-enoneIC5010000.0 [1]
2-Pyridin-4-yl-benzo[h]chromen-4-oneIC5010000.0 [1]
4-[2-[(6-Methoxypyridin-3-yl)amino]-5-[(4-methylsulfonylpiperazin-1-yl)methyl]pyridin-3-yl]-6-methyl-1,3,5-triazin-2-amineIC5010000.0 [1]
CID 118502708IC50140.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ DNA-dependent protein kinase Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/dna-dependent-protein-kinase-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 8). Quest Database™ DNA-dependent protein kinase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/dna-dependent-protein-kinase-inhibitors-ic50-ki.
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