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DNA topoisomerase II alpha Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
EtoposideIC5056000.0 [1]
DoxorubicinIC50880.0 [1], 1000.0 [2], 3000.0 [3]
MerbaroneIC5032000.0 [1], 40000.0 [2], 120000.0 [3]
3-[(E)-4-Hydroxybenzylidene]-6-hydroxybenzofuran-2(3H)-oneIC50400000.0 [1]
3-[3-[3-(4-Aminobutylamino)propylamino]-2-hydroxypropoxy]-1-hydroxyxanthen-9-one;2,2,2-trifluoroacetic acidIC502500.0 [1], 10000.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseDNA topoisomerase II alpha Inhibitors (IC50, Ki)." AAT Bioquest, Inc.4 Dec2025https://www.aatbio.com/data-sets/dna-topoisomerase-ii-alpha-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 4). Quest DatabaseDNA topoisomerase II alpha Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/dna-topoisomerase-ii-alpha-inhibitors-ic50-ki.
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