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Dopamine D1 receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
(R)-2,3,4,5-Tetrahydro-8-chloro-3-methyl-5-phenyl-1H-3-benzazepin-7-olIC500.66 [1], 0.74 [2], 0.82 [3], 1.4 [4], 520.0 [5]
(R)-2,3,4,5-Tetrahydro-8-chloro-3-methyl-5-phenyl-1H-3-benzazepin-7-olKi0.15 [1]
HaloperidolKi107.0 [1]
7-Methyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecineKi60.4 [1]
Sch-23390 maleateIC500.22 [1], 0.27 [2], 1.7 [3], 30.0 [4]

References
This online resource may be cited as follows
MLA
"Quest DatabaseDopamine D1 receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.7 Dec2025https://www.aatbio.com/data-sets/dopamine-d1-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 7). Quest DatabaseDopamine D1 receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/dopamine-d1-receptor-inhibitors-ic50-ki.
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