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Dopamine D2 receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
HaloperidolIC500.16 [1], 0.7 [2]
HaloperidolKi0.66 [1], 0.89 [2], 2.0 [3], 2.5 [4], 2.84 [5]
ClozapineIC509.0 [1], 113.0 [2], 204.17 [3], 230.0 [4], 260.0 [5]
ClozapineKi130.0 [1], 144.0 [2], 220.0 [3]
AripiprazoleIC507.6 [1], 11.0 [2], 17.2 [3], 32.0 [4]

References
This online resource may be cited as follows
MLA
"Quest DatabaseDopamine D2 receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.5 Dec2025https://www.aatbio.com/data-sets/dopamine-d2-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 5). Quest DatabaseDopamine D2 receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/dopamine-d2-receptor-inhibitors-ic50-ki.
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