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Dopamine D3 receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
HaloperidolIC500.06 [1], 10.0 [2]
HaloperidolKi4.4 [1], 4.6 [2], 10.4 [3], 18.0 [4]
ClozapineIC50450.0 [1]
ClozapineKi240.0 [1], 242.0 [2], 319.0 [3], 513.0 [4]
QuinpiroleKi23.99 [1], 24.0 [2], 420.0 [3]

References
This online resource may be cited as follows
MLA
"Quest DatabaseDopamine D3 receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.30 Dec2025https://www.aatbio.com/data-sets/dopamine-d3-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 30). Quest DatabaseDopamine D3 receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/dopamine-d3-receptor-inhibitors-ic50-ki.
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