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Dopamine D4 receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
ClozapineIC5058.0 [1], 120.0 [2], 138.0 [3], 156.0 [4], 168.0 [5]
ClozapineKi28.4 [1]
HaloperidolIC501.3 [1], 5.0 [2], 6.0 [3], 6.5 [4]
HaloperidolKi2.3 [1]
3-((4-(4-Chlorophenyl)piperazin-1-yl)methyl)-1H-pyrrolo[2,3-b]pyridineKi0.43 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseDopamine D4 receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.13 Dec2025https://www.aatbio.com/data-sets/dopamine-d4-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 13). Quest DatabaseDopamine D4 receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/dopamine-d4-receptor-inhibitors-ic50-ki.
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