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Dopamine D5 receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
7-Methyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecineKi12.7 [1]
11-Methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaen-6-olKi1.69 [1]
HaloperidolKi38.0 [1], 48.0 [2], 58.0 [3], 260.0 [4]
ClozapineKi198.0 [1], 235.0 [2], 780.0 [3], 1000.0 [4]
AripiprazoleKi1000.0 [1], 1051.0 [2], 1600.0 [3]

References
This online resource may be cited as follows
MLA
"Quest DatabaseDopamine D5 receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.15 Dec2025https://www.aatbio.com/data-sets/dopamine-d5-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 15). Quest DatabaseDopamine D5 receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/dopamine-d5-receptor-inhibitors-ic50-ki.
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