logo
AAT Bioquest

Dual specificity mitogen-activated protein kinase kinase 4 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
StaurosporineIC501.0 [1]
(Z)-3-Amino-3-(4-aminophenylthio)-2-(2-(trifluoromethyl)phenyl)acrylonitrileIC5010000.0 [1]
5Z-7-OxozeaenolIC503000.0 [1]
JNK Inhibitor VIC5010000.0 [1]
CID 59604787IC5010000.0 [1]
CID 72547959IC505000.0 [1]
N-[3-[2-Amino-3-cyano-6-(2-hydroxyphenyl)pyridin-4-yl]phenyl]-5-oxooxolane-2-carboxamideIC5020000.0 [1]
N-{3-[2-Amino-3-cyano-6-(2-hydroxy-phenyl)-pyridin-4-yl]-phenyl}-3-piperidin-1-yl-propionamideIC5020000.0 [1]
2-[[1-Cyclopentyl-5-[1-(Oxetan-3-Yl)piperidin-4-Yl]pyrazol-3-Yl]amino]pyridine-4-CarbonitrileIC505000.0 [1]
(13R,15S)-13-Methyl-16-oxa-8,9,12,22,24-pentazahexacyclo[15.6.2.16,9.112,15.02,7.021,25]heptacosa-1(24),2,4,6,17,19,21(25)-heptaene-23,27-dioneIC501000.0 [1]
2-Methoxy-12-(2-hydroxyethyl)-13,14-dihydronaphthol[2,1-a]pyrrolo[3,4-c]carbazole-5-oneIC503000.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
2-Isopropoxy-12-(2-hydroxyethyl)-13,14-dihydronaphthol[2,1-a]pyrrolo[3,4-c]carbazole-5-oneIC503000.0 [1]
3-[5-Chloro-4-[(2,4-difluorophenyl)methoxy]-6-oxopyrimidin-1-yl]-N-(2-hydroxyethyl)-4-methylbenzamideIC5010000.0 [1]
VinylcyanamideIC501000.0 [1]
4-(4-(2-(Cyclopentylamino)pyrimidin-4-yl)-1H-pyrazol-3-yl)cyclohexanolIC50920.0 [1]
2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamideIC5010000.0 [1]
4-(1-Hydroxypropan-2-ylamino)-2-methyl-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
2-Methyl-4-piperidin-1-yl-9H-pyrimido[4,5-b]indole-6-carboxylic acidIC501000.0 [1]
2-Amino-4-(azepan-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
2-Methyl-4-piperidin-1-yl-9H-pyrimido[4,5-b]indole-6-carboxamideIC501000.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Dual specificity mitogen-activated protein kinase kinase 4 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/dual-specificity-mitogen-activated-protein-kinase-kinase-4-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Dual specificity mitogen-activated protein kinase kinase 4 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/dual-specificity-mitogen-activated-protein-kinase-kinase-4-inhibitors-ic50-ki.
BibTeXEndNoteRefMan