Elastase 1 Inhibitors (IC50, Ki)

Name: Elastase 1 Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Telaprevir	IC50	30.0 ^[1]
	Boceprevir	IC50	10000.0 ^[1]
	Z-Pro-prolinal	IC50	51.6 ^[1]
	Polyozellin	IC50	2720.0 ^[1]
	(1R,21S,24S)-21-Tert-butyl-N-[(1R,2S)-1-(cyclopropylsulfonylcarbamoyl)-2-ethenylcyclopropyl]-16,16-dimethyl-3,19,22-trioxo-2,18-dioxa-4,20,23-triazatetracyclo[21.2.1.14,7.06,11]heptacosa-6(11),7,9-triene-24-carboxamide	IC50	10000.0 ^[1]
	Kynapcin-12	IC50	1250.0 ^[1]
	Kynapcin-24	Ki	290.0 ^[1]
	Methyl (3S)-3-[[(2S)-1-[(2S)-2-[[(2S)-2-[(4-methoxy-4-oxobutanoyl)amino]propanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-4-methyl-2-oxopentanoate	Ki	200.0 ^[1]
	Methyl (3S)-3-[[(2S)-1-[(2S)-2-[[(2S)-1-acetylpyrrolidine-2-carbonyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-2-oxobutanoate	Ki	850.0 ^[1]
	(2S)-1-[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-[[(2S)-2-[[(3S,9S,12S,15S,18S,21S,24S,27S)-12-(3-Carbamimidamidopropyl)-18-(carboxymethyl)-3,15-bis[(4-hydroxyphenyl)methyl]-21,24-bis(1H-indol-3-ylmethyl)-2,5,8,11,14,17,20,23,26-nonaoxo-1,4,7,10,13,16,19,22,25-nonazabicyclo[25.3.0]triacontane-9-carbonyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]acetyl]amino]acetyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-hydroxybutanoyl]amino]-3-phenylpropanoyl]amino]-3-methylpentanoyl]amino]-3-hydroxypropanoyl]pyrrolidine-2-carboxylic acid	IC50	1100.0 ^[1]
	Methyl 4-oxo-4-[[(2R)-1-oxo-3-phenyl-1-[(2S)-2-[[(3S)-1,1,1-trifluoro-4-methyl-2-oxopentan-3-yl]carbamoyl]pyrrolidin-1-yl]propan-2-yl]amino]butanoate	Ki	660.0 ^[1]
	Tert-butyl N-[(2S)-1-oxo-3-phenyl-1-[(2S)-2-[[(3S)-1,1,1-trifluoro-4-methyl-2-oxopentan-3-yl]carbamoyl]pyrrolidin-1-yl]propan-2-yl]carbamate	Ki	160.0 ^[1]
	Benzyl N-[(2S)-1-oxo-1-[[(2S)-1-oxo-1-[(2S)-2-[[(3S)-1,1,1-trifluoro-4-methyl-2-oxopentan-3-yl]carbamoyl]pyrrolidin-1-yl]propan-2-yl]amino]propan-2-yl]carbamate	Ki	1.0 ^[1]
	Methyl 4-oxo-4-[[(2S)-1-oxo-1-[[(2S)-1-oxo-1-[(2S)-2-[[(3S)-1,1,1-trifluoro-4-methyl-2-oxopentan-3-yl]carbamoyl]pyrrolidin-1-yl]propan-2-yl]amino]propan-2-yl]amino]butanoate	Ki	14.0 ^[1]
	Methyl (3S)-3-[[(2S)-1-[(2S)-2-[[(2S)-2-[(4-methoxy-4-oxobutanoyl)amino]propanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-2-oxo-4-phenylbutanoate	Ki	1000000.0 ^[1]
	Methyl 4-oxo-4-[[(2S)-1-oxo-1-[[(2S)-1-oxo-1-[(2S)-2-[[(2S)-4,4,4-trifluoro-3-oxo-1-phenylbutan-2-yl]carbamoyl]pyrrolidin-1-yl]propan-2-yl]amino]propan-2-yl]amino]butanoate	Ki	1500000.0 ^[1]
	Acetyl-Pro-Ala-Pro-Ala-trifluoro methane	Ki	800000.0 ^[1]
	Acetyl-Ala-Ala-Pro-Ala-trifluromethane	Ki	250.0 ^[1]
	Ethyl (3S)-2-oxo-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-(phenylmethoxycarbonylamino)propanoyl]amino]propanoyl]amino]propanoyl]amino]butanoate	Ki	300.0 ^[1]
	Methyl 4-[[(5S)-5-(1-adamantylsulfonylamino)-6-oxo-6-[(2S)-2-[[(3S)-1,1,1-trifluoro-4-methyl-2-oxopentan-3-yl]carbamoyl]pyrrolidin-1-yl]hexyl]amino]-4-oxobutanoate	Ki	0.58 ^[1]
	Ethyl (4S)-2,2-difluoro-4-[[(2S)-1-[(2S)-2-[[(2S)-2-[(4-methoxy-4-oxobutanoyl)amino]propanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-methyl-3-oxohexanoate	Ki	4300.0 ^[1]
	Tert-butyl N-[(2S)-1-oxo-1-[[(2S)-1-oxo-1-[(2S)-2-[[(3S)-1,1,1-trifluoro-4-methyl-2-oxopentan-3-yl]carbamoyl]pyrrolidin-1-yl]propan-2-yl]amino]propan-2-yl]carbamate	Ki	44.0 ^[1]
	2-[4-[Amino-[2-[(4R)-4-cyano-1,3-thiazolidin-3-yl]-2-oxoethyl]amino]piperidin-1-yl]-N-(5-chloropyridin-2-yl)acetamide;trihydrochloride	IC50	10000.0 ^[1]
	(2S)-1-[(2S)-2-[[(2S)-2-[[5-(Dimethylamino)naphthalen-1-yl]sulfonylamino]propanoyl]amino]propanoyl]-N-[(3S)-1,1,1-trifluoro-4-methyl-2-oxopentan-3-yl]pyrrolidine-2-carboxamide	Ki	1000000.0 ^[1]

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MLA	"Quest Database™ Elastase 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/elastase-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Elastase 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/elastase-1-inhibitors-ic50-ki.
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Elastase 1 Inhibitors (IC50, Ki)

References

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