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Endoplasmin Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
Methyl 2-[2-(1-benzyl-1H-imidazol-2-yl)ethyl]-3-chloro-4,6-dihydroxybenzoateIC5032.0 [1], 1140.0 [2], 1150.0 [3], 1200.0 [4]
LuminespibIC5085.0 [1]
LuminespibKi4.0 [1]
Snx-2112Ki484.0 [1]
PU-H71IC5026.0 [1]
6-Chloro-9-((4-methoxy-3,5-dimethylpyridin-2-yl)methyl)-9H-purin-2-amineKi176.0 [1]
CID 67495834Ki375.0 [1]
5-[2-Amino-4-chloro-7-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]pyrrolo[2,3-d]pyrimidin-5-yl]-2-methylpent-4-yn-2-olKi61.0 [1]
8-((3,5-Dichlorophenyl)thio)-9-(3-(isopropylamino)propyl)-9H-purin-6-amineIC50220.0 [1]
9-(Pent-4-yn-1-yl)-8-((2,4,5-trichlorophenyl)thio)-9H-purin-6-amineIC50170.0 [1]
8-((2,4-Dimethylphenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amineIC501630.0 [1]
8-((2,5-Dichlorophenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amineIC50530.0 [1]
8-((3,5-Dimethylphenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amineIC5011450.0 [1]
8-((2,4-Dichlorophenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amineIC50120.0 [1]
8-((3,5-Dichlorophenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amineIC50260.0 [1]
8-((2,5-Dimethylphenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amineIC501140.0 [1]
8-(2-Chloro-phenylsulfanyl)-9-pent-4-ynyl-9H-purin-6-ylamineIC50350.0 [1]
8-(4-Methoxy-phenylsulfanyl)-9-pent-4-ynyl-9H-purin-6-ylamineIC501130.0 [1]
[2-(6-Amino-9-pent-4-ynyl-9H-purin-8-ylsulfanyl)-phenyl]-methanolIC5029400.0 [1]
8-[2-Chloro-5-(trifluoromethyl)phenyl]sulfanyl-9-pent-4-ynylpurin-6-amineIC50500.0 [1]
8-(4-Chloro-phenylsulfanyl)-9-pent-4-ynyl-9H-purin-6-ylamineIC501500.0 [1]
9-Pent-4-ynyl-8-(2-trifluoromethoxy-phenylsulfanyl)-9H-purin-6-ylamineIC501400.0 [1]
8-(2-Methoxy-phenylsulfanyl)-9-pent-4-ynyl-9H-purin-6-ylamineIC506200.0 [1]
8-(2,4-Dimethoxy-phenylsulfanyl)-9-pent-4-ynyl-9H-purin-6-ylamineIC5034500.0 [1]
8-[(2,4-Dimethylphenyl)sulfanyl]-3-Pent-4-Yn-1-Yl-3h-Purin-6-AmineIC5011770.0 [1]
8-(Mesitylthio)-9-(pent-4-yn-1-yl)-9H-purin-6-amineIC502100.0 [1]
8-(2,4-Dichlorophenyl)sulfonyl-9-pent-4-ynylpurin-6-amineIC504700.0 [1]
9-But-3-ynyl-8-(3,5-dichlorophenyl)sulfanylpurin-6-amineIC50287.0 [1]
8-(2,4-Dichlorophenoxy)-9-pent-4-ynylpurin-6-amineIC50500.0 [1]
8-(2,4-Dichlorophenyl)sulfanyl-9-pentan-2-ylpurin-6-amineIC502480.0 [1]
8-(2,4-Dichlorophenyl)sulfinyl-9-pent-4-ynylpurin-6-amineIC505400.0 [1]
8-[(2,4-Dichlorophenyl)methyl]-9-pent-4-ynylpurin-6-amineIC50700.0 [1]
9-Benzyl-8-(3,5-dichlorophenyl)sulfanylpurin-6-amineIC505000.0 [1]
8-(3,5-Dichlorophenyl)sulfanyl-9-(6,6,6-trifluorohexyl)purin-6-amineIC501648.0 [1]
9-Pent-4-ynyl-8-(2,3,4-trichlorophenyl)sulfanylpurin-6-amineIC50430.0 [1]
8-(3,5-Dichlorophenyl)sulfanyl-9-(2-phenylethyl)purin-6-amineIC502500.0 [1]
8-(3,5-Dichlorophenyl)sulfanyl-9-(4,4,4-trifluorobutyl)purin-6-amineIC50502.0 [1]
8-(3,5-Dichlorophenyl)sulfanyl-9-hex-5-yn-3-ylpurin-6-amineIC505000.0 [1]
8-(2,6-Dichloropyridin-4-yl)sulfanyl-9-pent-4-ynylpurin-6-amineIC501900.0 [1]
8-(3,5-Dichlorophenyl)sulfanyl-9-(3,3,3-trifluoropropyl)purin-6-amineIC50560.0 [1]
8-(3,5-Dibromophenyl)sulfanyl-9-pent-4-ynylpurin-6-amineIC50290.0 [1]
8-(2,4-Dichlorophenyl)sulfanyl-9-[3-(propan-2-ylamino)propyl]purin-6-amineIC50410.0 [1]
(6-Amino-9-pent-4-ynylpurin-8-yl)-(2,4-dichlorophenyl)methanoneIC50340.0 [1]
8-(3,5-Dichlorophenyl)sulfanyl-9-hex-5-ynylpurin-6-amineIC50665.0 [1]
8-(3,5-Dichlorophenyl)sulfanyl-9-(5,5,5-trifluoropentyl)purin-6-amineIC502740.0 [1]
5-(6-Amino-9-pent-4-ynylpurin-8-yl)sulfanylbenzene-1,3-dicarbonitrileIC507730.0 [1]
8-(3,5-Dichlorophenyl)sulfanyl-9-pentan-2-ylpurin-6-amineIC5014300.0 [1]
8-(4-Bromo-2-chlorophenyl)sulfanyl-9-pent-4-ynylpurin-6-amineIC50390.0 [1]
9-But-2-ynyl-8-(3,5-dichlorophenyl)sulfanylpurin-6-amineIC505100.0 [1]
4-[6-Amino-8-(3,5-dichlorophenyl)sulfanylpurin-9-yl]butanenitrileIC50429.0 [1]
8-(3,4-Dichlorophenyl)sulfanyl-9-pent-4-ynylpurin-6-amineIC50695.0 [1]
8-(2,4-Dichlorophenyl)sulfanyl-9-hex-5-yn-3-ylpurin-6-amineIC50920.0 [1]
2-(2,4-Dichlorophenyl)sulfanyl-1-[3-(propan-2-ylamino)propyl]imidazo[4,5-c]pyridin-4-amineIC503440.0 [1]
8-(3-Bromo-5-chlorophenyl)sulfanyl-9-pent-4-ynylpurin-6-amineIC50240.0 [1]
2-(3,5-Dichlorophenyl)sulfanyl-1-[3-(propan-2-ylamino)propyl]imidazo[4,5-c]pyridin-4-amineIC501080.0 [1]
8-(3,5-Dichlorophenyl)sulfanyl-9-pent-4-yn-2-ylpurin-6-amineIC505800.0 [1]
9-Butyl-8-(3,5-dichlorophenyl)sulfanylpurin-6-amineIC50800.0 [1]
9-But-3-ynyl-8-(2,4-dichlorophenyl)sulfanylpurin-6-amineIC50390.0 [1]
8-(2,4-Dichlorophenyl)sulfanyl-9-pent-4-yn-2-ylpurin-6-amineIC505000.0 [1]
4-[8-[2-Chloro-5-(trifluoromethyl)phenyl]sulfanyl-6-imino-7H-purin-3-yl]butanenitrileIC50100000.0 [1]
4-[8-(3,5-Dichlorophenyl)sulfanyl-6-imino-7H-purin-3-yl]butanenitrileIC50100000.0 [1]
4-[8-(3,5-Dimethylphenyl)sulfanyl-6-imino-7H-purin-3-yl]butanenitrileIC50100000.0 [1]
4-[6-Imino-8-(2,4,5-trichlorophenyl)sulfanyl-7H-purin-3-yl]butanenitrileIC502080.0 [1]
4-[6-Imino-8-(2,4,6-trimethylphenyl)sulfanyl-7H-purin-3-yl]butanenitrileIC5020000.0 [1]
3-[8-(2,4-Dimethylphenyl)sulfanyl-6-imino-7H-purin-3-yl]-N-propan-2-ylpropan-1-amineIC5025000.0 [1]
3-[8-(3,5-Dichlorophenyl)sulfanyl-6-imino-7H-purin-3-yl]-N-propan-2-ylpropan-1-amineIC502430.0 [1]
4-[8-(2-Chlorophenyl)sulfanyl-6-imino-7H-purin-3-yl]butanenitrileIC50100000.0 [1]
4-[6-Imino-8-(2-methoxyphenyl)sulfanyl-7H-purin-3-yl]butanenitrileIC50100000.0 [1]
4-[8-[2-(Hydroxymethyl)phenyl]sulfanyl-6-imino-7H-purin-3-yl]butanenitrileIC50100000.0 [1]
4-[6-Imino-8-[2-(trifluoromethoxy)phenyl]sulfanyl-7H-purin-3-yl]butanenitrileIC50100000.0 [1]
4-[8-(2,4-Dichlorophenyl)sulfanyl-6-imino-7H-purin-3-yl]butanenitrileIC502370.0 [1]
4-[8-(2,4-Dimethylphenyl)sulfanyl-6-imino-7H-purin-3-yl]butanenitrileIC5011770.0 [1]
4-[8-(2,4-Dimethoxyphenyl)sulfanyl-6-imino-7H-purin-3-yl]butanenitrileIC50100000.0 [1]
4-[8-(2,5-Dichlorophenyl)sulfanyl-6-imino-7H-purin-3-yl]butanenitrileIC5035300.0 [1]
4-[8-(2,5-Dimethylphenyl)sulfanyl-6-imino-7H-purin-3-yl]butanenitrileIC50100000.0 [1]
2-[(6-Iodo-1,3-benzodioxol-5-yl)sulfanyl]-1-[3-(propan-2-ylamino)propyl]imidazo[4,5-c]pyridin-4-amineIC50101.0 [1]
8-[[6-(Dimethylamino)-1,3-benzodioxol-5-yl]sulfanyl]-9-[3-(propan-2-ylamino)propyl]purin-6-amineIC50265.0 [1]
[(4E,6Z,8R,9S,10E,12S,13R,14S,16R)-19-[2-(Dimethylamino)ethylamino]-13-hydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl] carbamateKi5.0 [1]
8-(2-Methylpropyl)-6-(3,6,6-trimethyl-4-oxo-5,7-dihydroindol-1-yl)-3,4-dihydro-2H-isoquinolin-1-oneKi10000.0 [1]
8-Cyclopentyl-6-(3,6,6-trimethyl-4-oxo-5,7-dihydroindol-1-yl)-3,4-dihydro-2H-isoquinolin-1-oneKi10000.0 [1]
4-(6,6-Dimethyl-4-oxo-5,7-dihydroindol-1-yl)-2-fluoro-6-[[(3S)-oxolan-3-yl]amino]benzamideKi2650.0 [1]
8-Cyclohexyl-6-(3,6,6-trimethyl-4-oxo-5,7-dihydroindol-1-yl)-3,4-dihydro-2H-isoquinolin-1-oneKi10000.0 [1]
8-(Oxan-4-yl)-6-(3,6,6-trimethyl-4-oxo-5,7-dihydroindol-1-yl)-3,4-dihydro-2H-isoquinolin-1-oneKi2400.0 [1]
8-Cyclobutyl-6-(3,6,6-trimethyl-4-oxo-5,7-dihydroindol-1-yl)-3,4-dihydro-2H-isoquinolin-1-oneKi10000.0 [1]
8-Butyl-6-(3,6,6-trimethyl-4-oxo-5,7-dihydroindol-1-yl)-3,4-dihydro-2H-isoquinolin-1-oneKi10000.0 [1]
8-Tert-butyl-6-(3,6,6-trimethyl-4-oxo-5,7-dihydroindol-1-yl)-3,4-dihydro-2H-isoquinolin-1-oneKi10000.0 [1]
8-Benzyl-6-(3,6,6-trimethyl-4-oxo-5,7-dihydroindol-1-yl)-3,4-dihydro-2H-isoquinolin-1-oneKi10000.0 [1]
8-Phenyl-6-(3,6,6-trimethyl-4-oxo-5,7-dihydroindol-1-yl)-3,4-dihydro-2H-isoquinolin-1-oneKi10000.0 [1]
8-(4-Fluorophenyl)-6-(3,6,6-trimethyl-4-oxo-5,7-dihydroindol-1-yl)-3,4-dihydro-2H-isoquinolin-1-oneKi10000.0 [1]
8-(3-Fluorophenyl)-6-(3,6,6-trimethyl-4-oxo-5,7-dihydroindol-1-yl)-3,4-dihydro-2H-isoquinolin-1-oneKi10000.0 [1]
8-(4-Methoxyphenyl)-6-(3,6,6-trimethyl-4-oxo-5,7-dihydroindol-1-yl)-3,4-dihydro-2H-isoquinolin-1-oneKi10000.0 [1]
2-Fluoro-6-[[(3S)-oxolan-3-yl]amino]-4-(2,7,7-trimethyl-5-oxo-3,4,6,8-tetrahydro-1H-pyrido[3,4-b]indol-9-yl)benzamideKi4400.0 [1]
2-[[(3S)-Oxolan-3-yl]amino]-4-(2,7,7-trimethyl-5-oxo-3,4,6,8-tetrahydro-1H-pyrido[3,4-b]indol-9-yl)benzamideKi1100.0 [1]
2-(Cyclopentylamino)-4-(2,7,7-trimethyl-5-oxo-3,4,6,8-tetrahydro-1H-pyrido[3,4-b]indol-9-yl)benzamideKi580.0 [1]
2-(Cyclopropylmethylamino)-4-(2,7,7-trimethyl-5-oxo-3,4,6,8-tetrahydro-1H-pyrido[3,4-b]indol-9-yl)benzamideKi2800.0 [1]
2-(2-Methoxyethylamino)-4-(2,7,7-trimethyl-5-oxo-3,4,6,8-tetrahydro-1H-pyrido[3,4-b]indol-9-yl)benzamideKi10000.0 [1]
2-(Thian-4-ylamino)-4-(2,7,7-trimethyl-5-oxo-3,4,6,8-tetrahydro-1H-pyrido[3,4-b]indol-9-yl)benzamideKi420.0 [1]
2-(Propylamino)-4-(2,7,7-trimethyl-5-oxo-3,4,6,8-tetrahydro-1H-pyrido[3,4-b]indol-9-yl)benzamideKi3200.0 [1]
2-(Cyclopropylamino)-4-(2,7,7-trimethyl-5-oxo-3,4,6,8-tetrahydro-1H-pyrido[3,4-b]indol-9-yl)benzamideKi10000.0 [1]
2-(2,2-Difluoroethylamino)-4-(2,7,7-trimethyl-5-oxo-3,4,6,8-tetrahydro-1H-pyrido[3,4-b]indol-9-yl)benzamideKi3700.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Endoplasmin Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/endoplasmin-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Endoplasmin Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/endoplasmin-inhibitors-ic50-ki.
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