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Ephrin type-A receptor 3 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
StaurosporineIC5019.72 [1], 48.0 [2]
DoramapimodIC501200.0 [1]
Bms-777607IC50500.0 [1]
3-[[2-[3-(Morpholin-4-ylmethyl)phenyl]thieno[3,2-b]pyridin-7-yl]amino]phenolIC505.1 [1]
4-Tert-Butyl-N-[6-(1h-Imidazol-1-Yl)imidazo[1,2-A]pyridin-2-Yl]benzamideIC5019952.62 [1]
CID 44478401IC5040.0 [1]
5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamideIC5010000.0 [1]
CID 46864270IC501.2 [1]
1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)ureaIC5030000.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
2-Anilino-7-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5,5-dimethylpyrrolo[2,3-d]pyrimidin-6-oneIC502094.0 [1]
CID 71718651IC502500.0 [1]
3-Amino-6-(4-aminopiperidin-1-yl)-4-propylthieno[2,3-b]pyridine-2-carboxamideIC507000.0 [1]
3-Amino-6-(piperazin-1-yl)-4-propylthieno[2,3-b]pyridine-2-carboxamideIC508000.0 [1]
N-[1-(2-Methoxyethyl)pyrazol-4-yl]-2-(4-propan-2-yl-1,2,4-triazol-3-yl)-1,3-thiazole-4-carboxamideIC5019952.62 [1]
3-Amino-6-(3-hydroxypiperidin-1-yl)-4-propylthieno[2,3-b]pyridine-2-carboxamideIC507000.0 [1]
3-Amino-6-(4-hydroxypiperidin-1-yl)-4-propylthieno[2,3-b]pyridine-2-carboxamideIC509000.0 [1]
3-(6-Ethoxynaphthalen-2-yl)-1-propan-2-ylpyrazolo[3,4-d]pyrimidin-4-amine;hydrochlorideIC503700.0 [1]
3-(6-Methoxynaphthalen-2-yl)-1-propan-2-ylpyrazolo[3,4-d]pyrimidin-4-amine;hydrochlorideIC501600.0 [1]
3-(2-Ethoxyquinolin-6-yl)-1-(piperidin-4-ylmethyl)pyrazolo[3,4-d]pyrimidin-4-amine;hydrochlorideIC5010000.0 [1]
3-(6-Methoxynaphthalen-2-yl)-1-(piperidin-4-ylmethyl)pyrazolo[3,4-d]pyrimidin-4-amine;hydrochlorideIC5010000.0 [1]
3-(6-Ethoxynaphthalen-2-yl)-1-(piperidin-4-ylmethyl)pyrazolo[3,4-d]pyrimidin-4-amine;hydrochlorideIC5010000.0 [1]
3-(6-Ethoxynaphthalen-2-yl)-1-(1-methylpiperidin-4-yl)pyrazolo[3,4-d]pyrimidin-4-amine;hydrochlorideIC5010000.0 [1]
3-(6-Ethoxynaphthalen-2-yl)-1-[(1-methylpiperidin-4-yl)methyl]pyrazolo[3,4-d]pyrimidin-4-amine;hydrochlorideIC5010000.0 [1]
1-[5-Tert-butyl-3-(methanesulfonamido)-2-methoxyphenyl]-3-[4-[6-(morpholin-4-ylmethyl)pyridin-3-yl]naphthalen-1-yl]ureaIC503200.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Ephrin type-A receptor 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/ephrin-type-a-receptor-3-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Ephrin type-A receptor 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/ephrin-type-a-receptor-3-inhibitors-ic50-ki.
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