Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Imatinib | IC50 | 43.0 [1], 90.0 [2], 337.0 [3], 31000.0 [4] | |
| Nilotinib | IC50 | 3.7 [1], 32.6 [2], 43.0 [3], 100.0 [4] | |
| Dasatinib | IC50 | 0.5 [1], 4.8 [2] | |
| Ddr1-IN-2 | IC50 | 6.81 [1], 9.7 [2] | |
| 3-[[2-[3-(Morpholin-4-ylmethyl)phenyl]thieno[3,2-b]pyridin-7-yl]amino]phenol | IC50 | 164.0 [1] | |
MLA | "Quest Database™ Epithelial discoidin domain-containing receptor 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 15 Dec. 2025, https://www.aatbio.com/data-sets/epithelial-discoidin-domain-containing-receptor-1-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 15). Quest Database™ Epithelial discoidin domain-containing receptor 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/epithelial-discoidin-domain-containing-receptor-1-inhibitors-ic50-ki. | |
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