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Epoxide hydratase Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
AudaIC506.5 [1]
trans-AUCBIC501.5 [1]
trans-AUCBKi1.5 [1]
t-TUCBIC500.4 [1], 0.8 [2], 0.9 [3], 2.0 [4]
t-TUCBKi156.0 [1]
1,3-DicyclohexylureaIC5025.0 [1]
1-(Adamantane-1-yl)-3-(1-acetylpiperidine-4-yl)ureaIC507.0 [1], 8.0 [2], 15.0 [3], 57.0 [4]
1-(1-Adamantyl)-3-[4-(4-fluorophenoxy)cyclohexyl]ureaIC500.4 [1], 0.5 [2], 0.8 [3], 1.0 [4]
12-(3-Adamantan-1-yl-ureido)-dodecanoic acid butyl esterIC500.8 [1], 7.8 [2], 100.0 [3]
1-Adamantan-1-yl-3-{5-[2-(2-ethoxyethoxy)ethoxy]pentyl}ureaIC5014.0 [1], 14.1 [2]
1-(1-Propanoylpiperidin-4-yl)-3-[4-(trifluoromethoxy)phenyl]ureaIC503.7 [1]
1-(1-Propanoylpiperidin-4-yl)-3-[4-(trifluoromethoxy)phenyl]ureaKi0.91 [1]
1-(1-(Cyclopropanecarbonyl)piperidin-4-yl)-3-(4-(trifluoromethoxy)phenyl)ureaIC500.4 [1]
1-(1-(Cyclopropanecarbonyl)piperidin-4-yl)-3-(4-(trifluoromethoxy)phenyl)ureaKi0.55 [1]
1-Adamantan-1-yl-3-[4-(2,6-difluoro-benzyloxy)-cyclohexyl]-ureaIC500.5 [1], 1.1 [2], 1.4 [3], 1.7 [4]
cis-1-Adamantan-1-yl-3-[4-(4-methoxyphenoxy)cyclohexyl]-ureaIC500.5 [1], 0.55 [2], 0.8 [3], 0.87 [4]
N-(2,4-Dichlorobenzyl)-4-(pyrimidin-2-yloxy)piperidine-1-carboxamideIC5015.0 [1], 18.0 [2], 63.0 [3]
trans-1-Adamantan-1-yl-3-(4-methoxycyclohexyl)ureaIC502.6 [1], 2.7 [2], 4.0 [3], 5.1 [4]
N-1-Adamantyl-N'-cyclohexylureaIC501.6 [1], 2.0 [2]
1-(1-(Methylsulfonyl)piperidin-4-yl)-3-(4-(trifluoromethoxy)phenyl)ureaIC502.9 [1]
Methyl 4-(1-adamantylcarbamoylamino)-2-hydroxy-benzoateIC501.2 [1], 2.8 [2]
4-(3-Adamantan-1-yl-ureido)-butyric acid pentyl esterIC5010.0 [1], 170.0 [2]
cis-4-(3-(4-(4-Fluorophenoxy)cyclohexyl)ureido)benzoic acidIC50142.0 [1], 220.0 [2]
1-Adamantan-1-yl-3-{4-[2-(2-ethoxyethoxy)ethoxy]phenyl}ureaIC501.1 [1], 1.8 [2]
1-(1-Adamantyl)-3-[4-(3-morpholinopropoxy)phenyl]ureaIC501.3 [1], 9.4 [2]
1-Adamantan-1-yl-3-{3-[2-(2-ethoxyethoxy)ethoxy]phenyl}ureaIC501.1 [1], 1.8 [2]
4-Pyrrol-1-yl-N-[4-(trifluoromethoxy)phenyl]piperidine-1-carboxamideIC5011.0 [1], 12.0 [2], 126.0 [3]
1-Adamantan-1-yl-3-(1-propionyl-piperidin-4-yl)-ureaIC502.8 [1], 3.2 [2]
1,3-Bis(1-adamantyl)ureaIC501.2 [1], 1.3 [2]
N-Methyl-4-{[trans-4-({[4-(trifluoromethoxy)phenyl]carbamoyl}amino)cyclohexyl]oxy}benzamideIC500.5 [1], 2.0 [2]
cis-1-Adamantan-1-yl-3-(4-benzyloxycyclohexyl)ureaIC500.9 [1], 1.1 [2], 1.7 [3]
cis-1-Adamantan-1-yl-3-[4-(4-bromobenzyloxy)cyclohexyl]-ureaIC501.7 [1], 2.1 [2], 12.3 [3]
cis-1-Adamantan-1-yl-3-(4-hydroxycyclohexyl)ureaIC5012.6 [1], 14.0 [2], 76.0 [3]
cis-1-Adamantan-1-yl-3-[4-(2,6-difluoro-4-isopropoxybenzyloxy)cyclohexyl]ureaIC503.5 [1], 4.8 [2]
cis-1-Adamantan-1-yl-3-[4-(4-bromophenoxy)cyclohexyl]ureaIC501.1 [1], 1.3 [2], 2.0 [3]
cis-1-Adamantan-1-yl-3-(4-methoxycyclohexyl)ureaIC502.5 [1], 4.0 [2], 4.8 [3]
1-(1-(Isopropylsulfonyl)piperidin-4-yl)-3-(4-(trifluoromethyl)phenyl)ureaIC502.9 [1], 13.0 [2]
1-(1-(Isopropylsulfonyl)piperidin-4-yl)-3-(4-(trifluoromethyl)phenyl)ureaKi1.17 [1]
1-(1-(Methylsulfonyl)piperidin-4-yl)-3-(4-(trifluoromethyl)phenyl)ureaIC503.7 [1], 26.0 [2]
1-(1-(Methylsulfonyl)piperidin-4-yl)-3-(4-(trifluoromethyl)phenyl)ureaKi7.16 [1]
1-(1-Acetylpiperidin-4-yl)-3-(4-(trifluoromethyl)phenyl)ureaIC5011.0 [1], 98.0 [2]
1-(1-Acetylpiperidin-4-yl)-3-(4-(trifluoromethyl)phenyl)ureaKi14.6 [1]
1-(1-Propionylpiperidin-4-yl)-3-(4-(trifluoromethyl)phenyl)ureaIC500.7 [1]
1-(1-Propionylpiperidin-4-yl)-3-(4-(trifluoromethyl)phenyl)ureaKi2.96 [1]
4-[3-(1-Methylethyl)-1,2,4-Oxadiazol-5-Yl]-N-[(1s,2r)-2-Phenylcyclopropyl]piperidine-1-CarboxamideIC506.1 [1], 8.5 [2], 13.0 [3]
4-[4-[[4-Chloro-3-(trifluoromethyl)phenyl]carbamoylamino]cyclohexyl]oxy-N-methylpyridine-2-carboxamideIC500.5 [1]
1-[1-(1-Adamantyl)ethyl]-3-[4-[1-(1-adamantyl)ethylcarbamoylamino]butyl]ureaIC501.2 [1], 2.5 [2]
1-[1-(1-Adamantyl)ethyl]-3-[4-[1-(1-adamantyl)ethylcarbamoylamino]butyl]ureaKi2.7 [1]
1-[1-(1-Adamantyl)ethyl]-3-[8-[1-(1-adamantyl)ethylcarbamoylamino]octyl]ureaIC500.5 [1], 0.8 [2]
1-[1-(1-Adamantyl)ethyl]-3-[8-[1-(1-adamantyl)ethylcarbamoylamino]octyl]ureaKi3.1 [1]
1-(2-Adamantyl)-3-[8-(2-adamantylcarbamoylamino)octyl]ureaIC502.6 [1], 4.1 [2]
1-(2-Adamantyl)-3-[8-(2-adamantylcarbamoylamino)octyl]ureaKi2.4 [1]
1-[(Z)-12-(5-Oxo-4H-1,2,4-oxadiazol-3-yl)dodec-5-enyl]-3-pentylureaIC5065.0 [1]
1-[(Z)-12-(5-Oxo-4H-1,2,4-thiadiazol-3-yl)dodec-5-enyl]-3-pentylureaIC50231.0 [1]
2-[2-(2-Hydroxyethoxy)ethoxy]ethyl (Z)-13-[[2-(butylamino)-2-oxoacetyl]amino]tridec-8-enoateIC50500.0 [1]
2-[2-(2-Hydroxyethoxy)ethoxy]ethyl (Z)-13-(pentylcarbamoylamino)tridec-8-enoateIC50255.0 [1]
2-[[(Z)-13-[Methyl-[methyl(pentyl)carbamoyl]amino]tridec-8-enoyl]amino]acetic acidIC50500.0 [1]
(Z)-N-Methylsulfonyl-13-(pentylcarbamoylamino)tridec-8-enamideIC5071.0 [1]
1-Pentyl-3-[(Z)-11-(1H-1,2,4-triazol-5-ylsulfinyl)undec-5-enyl]ureaIC5096.0 [1]
1-Pentyl-3-[(Z)-11-(1H-1,2,4-triazol-5-ylsulfanyl)undec-5-enyl]ureaIC5032.0 [1]
1-Pentyl-3-[(Z)-11-(2H-tetrazol-5-ylsulfanyl)undec-5-enyl]ureaIC5022.0 [1]
1-[(Z)-11-(2-Hydroxyphenyl)sulfonylundec-5-enyl]-3-pentylureaIC5011.0 [1]
1-[(Z)-11-(2-Hydroxyphenyl)sulfanylundec-5-enyl]-3-pentylureaIC506.0 [1]
1-[(Z)-11-(Benzenesulfonamido)undec-5-enyl]-3-pentylureaIC5032.0 [1]
1-Pentyl-3-[(Z)-11-(1H-1,2,4-triazol-5-ylsulfonyl)undec-5-enyl]ureaIC5023.0 [1]
1-[(5Z)-12-(1H-Tetrazole-5-yl)-5-dodecenyl]-3-pentylureaIC5011.0 [1]
N-Butyl-N'-[(Z)-12-(2H-tetrazol-5-yl)dodec-5-enyl]oxamideIC50500.0 [1]
1-Pentyl-3-[(Z)-13-(2H-tetrazol-5-yl)tridec-5-enyl]ureaIC5032.0 [1]
1-[(Z)-11-(2,4-Dioxo-1,3-thiazolidin-5-yl)undec-5-enyl]-3-pentylureaIC5057.0 [1]
1-[(Z)-12-(2-Oxo-5H-1,2,3,5-oxathiadiazol-4-yl)dodec-5-enyl]-3-pentylureaIC5010.0 [1]
N-[(Z)-12-(2-Oxo-5H-1,2,3,5-oxathiadiazol-4-yl)dodec-5-enyl]-N-propan-2-ylheptanamideIC50500.0 [1]
(Z)-N-(Benzenesulfonyl)-13-(pentylcarbamoylamino)tridec-8-enamideIC5041.0 [1]
1-Pentyl-3-[(Z)-12-(5-sulfanylidene-2H-1,2,4-oxadiazol-3-yl)dodec-5-enyl]ureaIC5031.0 [1]
N-[4-[5-(Pentylcarbamoylamino)pentoxy]-1,3-benzothiazol-2-yl]acetamideIC50500.0 [1]
N'-[5-[(2-Acetamido-1,3-benzothiazol-4-yl)oxy]pentyl]-N-butyloxamideIC50500.0 [1]
1-(1-Adamantylmethyl)-3-[6-(1-adamantylmethylcarbamoylamino)hexyl]ureaIC500.4 [1], 0.7 [2]
1-(1-Adamantylmethyl)-3-[6-(1-adamantylmethylcarbamoylamino)hexyl]ureaKi3.4 [1]
[(Z)-12-(Pentylcarbamoylamino)dodec-7-enyl]phosphonic acidIC50500.0 [1]
(Z)-12-(Pentylcarbamoylamino)dodec-7-ene-1-sulfonic acidIC5057.0 [1]
SorafenibIC5012.0 [1]
FulvestrantIC506.0 [1]
FulvestrantKi26.0 [1]
Aloe-emodinIC5026800.0 [1]
Aloe-emodinKi52200.0 [1]
Aloin AIC5037400.0 [1]
Aloin AKi57300.0 [1]
AloinIC5041100.0 [1]
AloinKi27800.0 [1]
1,3-DiphenylureaIC50390.0 [1], 400.0 [2]
Unii-L33EX3XR0TIC500.03 [1], 110.0 [2]
1-(2-Adamantyl)-3-(2,3,4-trifluorophenyl)ureaIC500.4 [1]
N-Cyclohexyl-N'-phenylureaIC50760.0 [1], 1390.0 [2]
Methyl 3-(1-adamantylcarbamoylamino)benzoateIC5013.5 [1], 14.0 [2]
1-(1-Adamantyl)-3-(4-pentoxycyclohexyl)ureaIC501.2 [1]
4-(3-Adamantan-1-yl-ureido)butyric acidIC50684.0 [1], 37000.0 [2]
1-Adamantan-1-yl-3-[4-(4-fluorophenoxy)butyl]ureaIC503.9 [1], 11.1 [2]
1-Adamantyl-3-(3-(3-morpholinopropoxy)phenyl)ureaIC500.8 [1]
1-[4-(4-Fluorophenoxy)cyclohexyl]-3-[4-(trifluoromethoxy)phenyl]ureaIC500.9 [1]
3-(1-Acetylpiperidin-4-yl)-1-[4-(trifluoromethoxy)phenyl]ureaIC5012.0 [1], 59.0 [2]
N-(3,3-Diphenylpropyl)pyridine-3-carboxamideIC507.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Epoxide hydratase Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/epoxide-hydratase-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Epoxide hydratase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/epoxide-hydratase-inhibitors-ic50-ki.
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