Fatty acid binding protein epidermal Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Palmitic acid	IC50	1200.0 [1]
	Palmitic acid	Ki	802.0 [1]
	(2S,4S)-3-(6-Acetamidonaphthalen-1-yl)oxycarbonyl-2,4-diphenylcyclobutane-1-carboxylic acid	Ki	970.0 [1], 7080.0 [2]
	(2R,4R)-2,4-Diphenyl-3-[[4-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3-thiazol-2-yl]carbamoyl]cyclobutane-1-carboxylic acid	Ki	10000.0 [1]
	3-(Naphthyloxycarbonyl)-2,4-diphenylcyclobutanecarboxylic acid	Ki	810.0 [1], 900.0 [2]
	Oleic acid	Ki	248.0 [1]
	2-((2'-(5-Ethyl-3,4-diphenyl-1H-pyrazol-1-yl)-[1,1'-biphenyl]-3-yl)oxy)acetic acid	Ki	350.0 [1]
	Truxillic acid	Ki	10000.0 [1]
	2,4,6-Triisopropylbenzoic acid	IC50	50000.0 [1]
	(E)-4-[(2-Methoxycarbonyl-5-thiophen-2-ylthiophen-3-yl)amino]-4-oxobut-2-enoic acid	Ki	3400.0 [1]
	3-Carbazol-9-yl-propionic acid	IC50	30000.0 [1]
	5-(2-(4,5-Diphenyloxazol-2-yl)phenoxy)pentanoic acid	Ki	2000.0 [1]
	6-Chloro-4-Phenyl-2-(Piperidin-1-Yl)-3-(1h-Tetrazol-5-Yl)quinoline	Ki	86.0 [1]
	[[2'-(4,5-Diphenyl-2-oxazolyl)-1,1'-biphenyl-3-yl]oxy]acetic acid	Ki	2000.0 [1]
	(2R,4R)-3-Naphthalen-1-yloxycarbonyl-2,4-diphenylcyclobutane-1-carboxylic acid	Ki	710.0 [1]
	(1s,2s,3s,4s)-3-{[(Naphthalen-1-Yl)oxy]carbonyl}-2,4-Diphenylcyclobutane-1-Carboxylic Acid	Ki	790.0 [1]
	2,4,6-Triisopropylbenzenesulfonic acid	IC50	16000.0 [1]
	2-(2,3-Bis(2-chlorobenzyloxy)phenyl)acetic acid	Ki	3.0 [1]
	1,3-Cyclobutanedicarboxylic acid, 2,4-bis(4-hydroxy-3-methoxyphenyl)-	Ki	10000.0 [1]
	2-((2'-(1-Ethyl-4,5-diphenyl-1H-imidazol-2-yl)(1,1'-biphenyl)-3-yl)oxy)-acetic acid	Ki	830.0 [1]
	2-[3-[2-(1-Ethyl-4,5-diphenylimidazol-2-yl)phenyl]anilino]acetic acid	Ki	2000.0 [1]
	(2S,4S)-3-[(4-Methoxyphenyl)methoxycarbonyl]-2,4-diphenylcyclobutane-1-carboxylic acid	Ki	2150.0 [1]
	(2S,4S)-3-(9H-Fluoren-9-ylmethoxycarbonyl)-2,4-diphenylcyclobutane-1-carboxylic acid	Ki	2560.0 [1]
	(2S,4S)-3-[3-[1-[2-[2-(2-Ethoxyethoxy)ethoxy]ethyl]triazol-4-yl]phenoxy]carbonyl-2,4-diphenylcyclobutane-1-carboxylic acid	Ki	10000.0 [1]
	(2S,4S)-3-[2-(2-Hydroxyphenyl)phenoxy]carbonyl-2,4-diphenylcyclobutane-1-carboxylic acid	Ki	1590.0 [1]
	(2S,4S)-3-(3-Ethynylphenoxy)carbonyl-2,4-diphenylcyclobutane-1-carboxylic acid	Ki	890.0 [1]
	(2S,4S)-2,4-Diphenyl-3-(2-phenylphenoxy)carbonylcyclobutane-1-carboxylic acid	Ki	770.0 [1]
	(2S,4S)-3-(2-Iodophenoxy)carbonyl-2,4-diphenylcyclobutane-1-carboxylic acid	Ki	1340.0 [1]
	(2S,4S)-3-(5-Ethynylnaphthalen-1-yl)oxycarbonyl-2,4-diphenylcyclobutane-1-carboxylic acid	Ki	3920.0 [1]
	(2S,4S)-2,4-Diphenyl-3-(4-phenylphenoxy)carbonylcyclobutane-1-carboxylic acid	Ki	2520.0 [1]
	(2S,4S)-2,4-Diphenyl-3-(3-phenylphenoxy)carbonylcyclobutane-1-carboxylic acid	Ki	850.0 [1]
	(2S,4S)-2,4-Diphenyl-3-[(1R,2S)-2-phenylcyclohexyl]oxycarbonylcyclobutane-1-carboxylic acid	Ki	180.0 [1]
	(2S,4S)-3-Naphthalen-1-yloxycarbonyl-2,4-bis(2-nitrophenyl)cyclobutane-1-carboxylic acid	Ki	10000.0 [1]
	(2S,4S)-2,4-Bis(2-chlorophenyl)-3-(9H-fluoren-9-ylmethoxycarbonyl)cyclobutane-1-carboxylic acid	Ki	890.0 [1]
	(2S,4S)-2,4-Bis(2-methoxyphenyl)-3-quinolin-5-yloxycarbonylcyclobutane-1-carboxylic acid	Ki	3930.0 [1]
	Fabp-IN-1	Ki	550.0 [1]
	(2S,4S)-2,4-Bis(2-chlorophenyl)-3-[(1R,2S)-2-phenylcyclohexyl]oxycarbonylcyclobutane-1-carboxylic acid	Ki	1700.0 [1]
	(2S,4S)-2,4-Bis(2-methoxyphenyl)-3-[(1R,2S)-2-phenylcyclohexyl]oxycarbonylcyclobutane-1-carboxylic acid	Ki	680.0 [1]
	Fabp5-IN-1	Ki	1720.0 [1]
	(2S,4S)-2,4-Bis(4-hydroxy-3-methoxyphenyl)-3-naphthalen-1-yloxycarbonylcyclobutane-1-carboxylic acid	Ki	10000.0 [1]
	(2S,4S)-3-[(4-Fluorophenyl)methoxycarbonyl]-2,4-diphenylcyclobutane-1-carboxylic acid	Ki	2420.0 [1]
	(2S,4S)-3-(2,3-Dihydro-1H-inden-2-yloxycarbonyl)-2,4-diphenylcyclobutane-1-carboxylic acid	Ki	1570.0 [1]
	(2S,4S)-3-[(4-Bromophenyl)methoxycarbonyl]-2,4-diphenylcyclobutane-1-carboxylic acid	Ki	1580.0 [1]
	(2S,4S)-2,4-Diphenyl-3-[(1S,2R)-2-phenylcyclohexyl]oxycarbonylcyclobutane-1-carboxylic acid	Ki	200.0 [1]
	Bis(oxan-4-ylmethyl) 2,4-diphenylcyclobutane-1,3-dicarboxylate	Ki	10000.0 [1]
	(2S,4S)-2,4-Bis(4-hydroxyphenyl)-3-naphthalen-1-yloxycarbonylcyclobutane-1-carboxylic acid	Ki	10000.0 [1]
	Bis[(4-methoxyphenyl)methyl] 2,4-diphenylcyclobutane-1,3-dicarboxylate	Ki	10000.0 [1]
	(2S,4S)-2,4-Bis(2-nitrophenyl)-3-[(1R,2S)-2-phenylcyclohexyl]oxycarbonylcyclobutane-1-carboxylic acid	Ki	10000.0 [1]
	(2S,4S)-2,4-Diphenyl-3-(2,2,2-trifluoroethoxycarbonyl)cyclobutane-1-carboxylic acid	Ki	10000.0 [1]
	(2S,4S)-2,4-Bis(2-bromophenyl)-3-[(1R,2S)-2-phenylcyclohexyl]oxycarbonylcyclobutane-1-carboxylic acid	Ki	2760.0 [1]
	Dibenzyl 2,4-diphenylcyclobutane-1,3-dicarboxylate	Ki	10000.0 [1]
	Bis[(4-fluorophenyl)methyl] 2,4-diphenylcyclobutane-1,3-dicarboxylate	Ki	10000.0 [1]
	(2R,4R)-2,4-Diphenyl-3-[(3-phenylphenyl)carbamoyl]cyclobutane-1-carboxylic acid	Ki	10000.0 [1]
	(2S,4S)-2,4-Diphenyl-3-(2,4,5-trichlorophenoxy)carbonylcyclobutane-1-carboxylic acid	Ki	800.0 [1]
	(2S,4S)-2,4-Bis(2,6-dichlorophenyl)-3-[(1R,2S)-2-phenylcyclohexyl]oxycarbonylcyclobutane-1-carboxylic acid	Ki	1230.0 [1]
	2,4-Bis(3,4-dimethoxyphenyl)cyclobutane-1,3-dicarboxylic acid	Ki	10000.0 [1]
	Benzeneacetic acid, 2,3-bis((2-chlorophenyl)methoxy)-alpha-hydroxy-, (alphaS)-	Ki	33.0 [1]
	2-[3-[2-(1-Methyl-4,5-diphenylimidazol-2-yl)phenyl]phenoxy]acetic acid	Ki	830.0 [1]
	2-[3-[2-[1-(2-Fluoroethyl)-4,5-diphenylimidazol-2-yl]phenyl]phenoxy]acetic acid	Ki	2000.0 [1]
	2-[3-[2-[1-(Carboxymethyl)-4,5-diphenylimidazol-2-yl]phenyl]anilino]acetic acid	Ki	2000.0 [1]
	2-[3-[2-[1-(2-Methylpropyl)-4,5-diphenylimidazol-2-yl]phenyl]anilino]acetic acid	Ki	2000.0 [1]
	2-[3-[2-(1-Methyl-4,5-diphenylimidazol-2-yl)phenyl]anilino]acetic acid	Ki	2000.0 [1]
	2-[3-[2-(3-Ethyl-4,5-diphenylfuran-2-yl)phenyl]phenoxy]acetic acid	Ki	290.0 [1]
	2-[3-[2-(4,5-Diphenyl-1H-imidazol-2-yl)phenyl]phenoxy]acetic acid	Ki	2000.0 [1]
	2-[3-[2-(4,5-Diphenyl-1H-imidazol-2-yl)phenyl]anilino]acetic acid	Ki	2000.0 [1]
	2-[3-[2-(4,5-Diphenylfuran-2-yl)phenyl]phenoxy]acetic acid	Ki	2000.0 [1]
	2-(2,3-Bis(2-chlorobenzyloxy)phenyl)-2-methoxyacetic acid	Ki	9.0 [1]
	2-[2,3-Bis[(2-chlorophenyl)methoxy]phenyl]-2-oxoacetic acid	Ki	2.0 [1]
	(2S,4S)-2,4-Diphenyl-3-phenylmethoxycarbonylcyclobutane-1-carboxylic acid	Ki	3810.0 [1]
	5-Carbazol-9-yl-pentanoic acid	IC50	3000.0 [1]
	3-(5-Bromo-indole-1-sulfonyl)-thiophene-2-carboxylic acid	IC50	14000.0 [1]
	2-(Carbazole-9-sulfonyl)-benzoic acid	IC50	17000.0 [1]
	3-(Carbazole-9-sulfonyl)-thiophene-2-carboxylic acid	IC50	9100.0 [1]
	1-(2,3-Bis(2-chlorobenzyloxy)phenyl)ethane-1,2-diol	Ki	2000.0 [1]
	2-[3-[2-(5-Ethyl-3,4-diphenylpyrazol-1-yl)phenyl]phenyl]-2-hydroxyacetic acid	Ki	550.0 [1]
	3-[2-(5-Ethyl-3,4-diphenylpyrazol-1-yl)phenyl]benzoic acid	Ki	240.0 [1]
	2,3-Bis[(2,4-dichloro-3-tritiophenyl)methoxy]benzoic acid	Ki	2.0 [1]
	Carbazole butanoic acid	IC50	6700.0 [1]
	(2S,4S)-3-Cyclohexyloxycarbonyl-2,4-diphenylcyclobutane-1-carboxylic acid	Ki	2170.0 [1]
	6-Chloranyl-2-Methyl-4-Phenyl-Quinoline-3-Carboxylic Acid	Ki	23200.0 [1]
	5-(6-Chloro-4-phenyl-2-piperidin-1-yl-quinolin-3-yl)-3H-[1,3,4]oxadiazole-2-thione	Ki	133.0 [1]
	6-Chloro-4-phenyl-2-propan-2-ylquinoline-3-carboxylic acid	Ki	1200.0 [1]
	6-Chloranyl-4-Phenyl-2-Piperidin-1-Yl-Quinoline-3-Carboxylic Acid	Ki	500.0 [1]
	6,8-Dichloro-4-Phenyl-2-(Piperidin-1-Yl)quinoline-3-Carboxylic Acid	Ki	120.0 [1]
	6-Chloro-8-methyl-4-phenyl-2-piperidin-1-yl-quinoline-3-carboxylic acid	Ki	100.0 [1]
	5-(6-Chloro-4-phenyl-2-piperidin-1-yl-quinolin-3-yl)-3H-[1,3,4]oxadiazol-2-one	Ki	167.0 [1]
	6-Chloro-2-dimethylamino-4-(3-isopropyl-phenyl)-quinoline-3-carboxylic acid	Ki	4300.0 [1]
	2-[3-[2-(4,5-Diphenyl-1H-pyrrol-2-yl)phenyl]phenoxy]acetic acid	Ki	2000.0 [1]
	2-[[5-Cyclopropyl-3-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-4-methylthiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid	IC50	30.0 [1]
	2-[[3-(3-Cyclopropyl-1,2,4-oxadiazol-5-yl)-4,5-dimethylthiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid	IC50	30.0 [1]
	2-[[4-Cyclopropyl-5-methyl-3-[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]thiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid	IC50	30.0 [1]
	3-[[4-Cyclopropyl-3-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-5-methylthiophen-2-yl]carbamoyl]bicyclo[2.2.2]oct-2-ene-2-carboxylic acid	IC50	40.0 [1]
	2-[[3-(3-Cyclopropyl-1,2,4-oxadiazol-5-yl)thiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid	IC50	890.0 [1]
	2-[[3-(3-Cyclopropyl-1,2,4-oxadiazol-5-yl)-4-methyl-5-(oxetan-3-yl)thiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid	IC50	60.0 [1]
	2-[[3-(3-Cyclopropyl-1,2,4-oxadiazol-5-yl)-4-methyl-5-(oxetan-3-yl)thiophen-2-yl]carbamoyl]cyclohexene-1-carboxylic acid	IC50	227.0 [1]
	2-[[3-(3-Cyclopropyl-1,2,4-oxadiazol-5-yl)-5-methyl-4-(trifluoromethyl)thiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid	IC50	60.0 [1]
	2-[[3-(3-Cyclopropyl-1,2,4-oxadiazol-5-yl)-5-ethoxycarbonyl-4-methylthiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid	IC50	130.0 [1]
	2-[[3-(3-Cyclopropyl-1,2,4-oxadiazol-5-yl)-5-(dimethylcarbamoyl)-4-methylthiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid	IC50	2709.7 [1]
	2-[[5-Cyclopropyl-3-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)thiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid	IC50	125.8 [1]
	2-[[4-Cyclopropyl-3-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)thiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid	IC50	38.8 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 100 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Fatty acid binding protein epidermal Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/fatty-acid-binding-protein-epidermal-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Fatty acid binding protein epidermal Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/fatty-acid-binding-protein-epidermal-inhibitors-ic50-ki.
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