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Fibroblast growth factor receptor 2 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
Azd4547IC502.5 [1]
StaurosporineIC501.77 [1], 3.36 [2], 5.8 [3], 34.0 [4]
Debio-1347IC507.6 [1]
N-[3-[[3-(2,6-Dichloro-3,5-dimethoxyphenyl)-7-[4-(diethylamino)butylamino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-1-yl]methyl]phenyl]prop-2-enamideIC502.29 [1], 2.3 [2], 6.2 [3]
7-(1,3,4,6,7,8,9,9a-Octahydropyrido[1,2-a]pyrazin-2-yl)-N-[5-[2-(3,5-dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]quinazolin-4-amineIC500.2 [1], 0.4 [2], 0.8 [3]

References
This online resource may be cited as follows
MLA
"Quest DatabaseFibroblast growth factor receptor 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.15 Dec2025https://www.aatbio.com/data-sets/fibroblast-growth-factor-receptor-2-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 15). Quest DatabaseFibroblast growth factor receptor 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/fibroblast-growth-factor-receptor-2-inhibitors-ic50-ki.
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