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Fibroblast growth factor receptor Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
▲
▼
Standard Values (in nM)
▲
▼
PD173074IC507.0 [1], 15.0 [2], 13000.0 [3]
Unii-NA856793UTIC5060.0 [1]
1,6-Naphthyridine deriv. 20IC501.0 [1], 85.0 [2], 1900.0 [3]
1,6-Naphthyridine 16IC503.6 [1], 15.0 [2], 4800.0 [3]
1,6-Naphthyridine 17IC501.0 [1], 1.9 [2], 330.0 [3]
1,6-Naphthyridine 18IC502.0 [1], 12.0 [2], 1700.0 [3]
1,6-Naphthyridine 19IC503.0 [1], 4.4 [2], 350.0 [3]
1,6-Naphthyridine 20IC500.4 [1], 2.7 [2], 200.0 [3]
1,6-Naphthyridine 22IC502.6 [1], 14.0 [2], 4500.0 [3]
1,6-Naphthyridine 23IC500.5 [1], 2.7 [2], 560.0 [3]
1,6-Naphthyridine 24IC500.5 [1], 2.0 [2], 340.0 [3]
1,6-Naphthyridine 26IC502.0 [1], 200.0 [2]
1,6-Naphthyridine 75IC502.7 [1], 6.0 [2], 56.0 [3]
1,6-Naphthyridine 76IC504.7 [1], 6.0 [2], 42.0 [3]
1,6-Naphthyridine 77IC503.0 [1], 4.0 [2], 630.0 [3]
Pyrido[2,3-d]pyrimidine 102IC5015.0 [1], 88.0 [2], 6800.0 [3]
Pyrido[2,3-d]pyrimidine 103IC506.0 [1], 28.0 [2], 4600.0 [3]
Pyrido[2,3-d]pyrimidine 104IC5033.0 [1], 430.0 [2], 25000.0 [3]
Pyrido[2,3-d]pyrimidine 105IC5020.0 [1], 37.0 [2], 6800.0 [3]
6-(2,6-Dichlorophenyl)-2-[4-[2-(diethylamino)ethoxy]anilino]-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5044.0 [1], 43000.0 [2]
1-Tert-butyl-3-[6-(2,6-dichlorophenyl)-2-[4-(diethylamino)butylamino]pyrido[2,3-d]pyrimidin-7-yl]ureaIC5048.0 [1]
1-[2-Amino-6-(2,6-dichlorophenyl)pyrido[2,3-d]pyrimidin-7-yl]-3-tert-butylureaIC50130.0 [1]
3-(3,5-Dimethoxyphenyl)-7-N-[3-(4-methylpiperazin-1-yl)propyl]-1,6-naphthyridine-2,7-diamineIC50150.0 [1], 6400.0 [2]
7-N-[4-(Diethylamino)butyl]-3-(3,5-dimethoxyphenyl)-1,6-naphthyridine-2,7-diamineIC50130.0 [1], 12000.0 [2]
1,6-Naphthyridine 25IC503.0 [1], 170.0 [2]
StaurosporineIC50420.0 [1]
SemaxanibIC505000.0 [1]
CanertinibIC5050000.0 [1]
TandutinibIC5030000.0 [1]
LinifanibIC5012500.0 [1]
Pyridone 6IC501480.0 [1]
Azd-1152hqpaKi10000.0 [1]
CID 6918852Ki5000.0 [1]
9-Hydroxy-4-phenyl-6H-pyrrolo[3,4-C]carbazole-1,3-dioneIC5050000.0 [1]
N-(4-Bromo-2-fluorophenyl)-6-methoxy-7-[2-(triazol-1-yl)ethoxy]quinazolin-4-amineIC501500.0 [1]
JNK Inhibitor VIIIKi4700.0 [1]
PDGF Receptor Tyrosine Kinase Inhibitor IIIIC5029700.0 [1]
2-Aminopyrido[2,3-d]pyrimidin-7(8H)-one 38IC50510.0 [1]
1-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-3-(3-methylphenyl)ureaIC504200.0 [1]
N-(3-Bromophenyl)-1H-imidazo[4,5-g]quinazolin-8-amineIC5050000.0 [1]
2-Aminopyrido[2,3-d]pyrimidin-7(8H)-one 2IC501320.0 [1]
CID 9916282IC508000.0 [1]
2-Aminopyrido[2,3-d]pyrimidin-7(8H)-one 19IC5050000.0 [1]
2-Aminopyrido[2,3-d]pyrimidin-7(8H)-one 29IC501970.0 [1]
2-Aminopyrido[2,3-d]pyrimidin-7(8H)-one 30IC501260.0 [1]
2-Aminopyrido[2,3-d]pyrimidin-7(8H)-one 68IC5051.0 [1]
8-(2-Bicyclo[2.2.1]heptanyl)-2-[4-[4-(3-hydroxypropyl)piperidin-1-yl]anilino]pyrido[2,3-d]pyrimidin-7-oneIC508620.0 [1]
4-(6,7-Dimethoxy-4-quinazolinyl)-N-(4-nitrophenyl)-1-piperazinecarboxamideIC50200000.0 [1]
N-(2-Chloro-6-methylphenyl)-2-[(cyclopropylcarbonyl)amino]-1,3-thiazole-5-carboxamideIC5025000.0 [1]
2,4-Difluoro-N-methoxy-5-[[6-(5-methyl-1,3,4-oxadiazol-2-yl)-5-propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]benzamideIC506.5 [1]
N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)acetamideKi4700.0 [1]
N-Benzyl-4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1-carbothioamideIC50200000.0 [1]
4-Amino-5-chloro-6-ethoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamideKi4700.0 [1]
1-Oxo-3-phenyl-1h-indene-2-carboxamideIC504700.0 [1]
(2S)-2-Amino-N-hydroxy-3-(4-hydroxyphenyl)propanamideKi23000.0 [1]
1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acidIC5010000.0 [1]
2-Aminopyrido[2,3-d]pyrimidin-7(8H)-one 28IC5050000.0 [1]
2-Aminopyrido[2,3-d]pyrimidin-7(8H)-one 31IC50348.0 [1]
2-Aminopyrido[2,3-d]pyrimidin-7(8H)-one 62IC5048.0 [1]
2-Aminopyrido[2,3-d]pyrimidin-7(8H)-one 71IC5061.0 [1]
6-Arylpyrido[2,3-d]pyrimidine deriv. 55IC50125.0 [1]
6-Arylpyrido[2,3-d]pyrimidine deriv. 56IC5040.0 [1]
6-Arylpyrido[2,3-d]pyrimidine deriv. 69IC50139.0 [1]
8-Ethyl-2-phenylamino-8H-pyrido[2,3-d]pyrimidin-7-oneIC503295.0 [1]
N8 Pyrido[2,3-d]pyrimidin-7-one deriv. 45IC502980.0 [1]
Pyrido-[2,3-d]-pyrimidin-7-one 35IC501740.0 [1]
6-Acetyl-8-cyclopentyl-5-methyl-2-(4-piperazin-1-yl-phenylamino)-8H-pyrido[2,3-d]pyrimidin-7-oneIC501860.0 [1]
Thienopyrimidine deriv. 28IC501500.0 [1]
N-(1,3-Benzodioxol-5-ylmethyl)-4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1-carbothioamideIC50160000.0 [1]
5-[[6-[5-(Difluoromethyl)-1,3,4-oxadiazol-2-yl]-5-propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]-2,4-difluoro-N-methoxybenzamideIC5021.0 [1]
2,4-Difluoro-N-methoxy-5-[[6-(5-methyl-1,3-oxazol-2-yl)-5-propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]benzamideIC504.0 [1]
2,4-Difluoro-N-methoxy-5-[[6-[5-(methylsulfonylmethyl)-1,3,4-oxadiazol-2-yl]-5-propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]benzamideIC504.6 [1]
N-(4-Bromophenyl)-4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1-carboxamideIC50200000.0 [1]
1-[2-Amino-6-(2,6-dichlorophenyl)pyrido[2,3-d]pyrimidin-7-yl]-3-ethylureaIC50130.0 [1]
N-(4-Cyanophenyl)-4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1-carboxamideIC50200000.0 [1]
4-(6,7-Dimethoxyquinazolin-4-yl)-N-(4-propan-2-ylphenyl)piperazine-1-carboxamideIC5030000.0 [1]
3-[[5-Cyano-6-(cyclopentylamino)pyrimidin-4-yl]amino]-4-methyl-N-(1,2-oxazol-3-yl)benzamideIC5050000.0 [1]
5-[[6-[5-[Difluoro(methylsulfonyl)methyl]-1,3,4-oxadiazol-2-yl]-5-propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]-2,4-difluoro-N-methoxybenzamideIC50130.0 [1]
N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethoxy-4-methylsulfonylphenyl)acetamideKi4700.0 [1]
N-(4-Amino-5-chloro-6-ethoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamideKi4700.0 [1]
N-(4-Amino-5-cyano-6-isopropoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamideKi4700.0 [1]
N-(4-Amino-5-cyano-6-phenylpyridin-2-yl)acetamideKi4700.0 [1]
VegfrecineIC50730.0 [1]
2-Amino-6-(3,5-dimethoxyphenyl)-8-methylpyrido[2,3-d]pyrimidine-7(8H)-oneIC50126.0 [1]
1-Tert-butyl-3-[6-(2,6-dichlorophenyl)-2-[4-[2-(diethylamino)ethoxy]anilino]pyrido[2,3-d]pyrimidin-7-yl]ureaIC5051.0 [1]
6-(2,6-Dichlorophenyl)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-oneIC5050000.0 [1]
6-Bromo-8-cyclopentyl-2-(4-piperazin-1-ylanilino)pyrido[2,3-d]pyrimidin-7-oneIC5080.0 [1]
7-((1H-Imidazol-1-yl)methyl)-3-(thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazoleIC5034355.0 [1]
7-[(4-Methylpiperazin-1-yl)methyl]-3-thiophen-3-yl-1,4-dihydroindeno[1,2-c]pyrazoleIC5050000.0 [1]
6-Arylpyrido[2,3-d]pyrimidine deriv. 13IC5082.0 [1]
1-[2-Amino-6-(2,6-dimethylphenyl)pyrido[2,3-d]pyrimidin-7-yl]-3-tert-butylureaIC50400.0 [1]
1-[2-Amino-6-(2,3,5,6-tetramethylphenyl)pyrido[2,3-d]pyrimidin-7-yl]-3-tert-butylureaIC50780.0 [1]
6-Arylpyrido[2,3-d]pyrimidine deriv. 32IC5033.0 [1]
6-Arylpyrido[2,3-d]pyrimidine deriv. 47IC5051.0 [1]
1-(2-Amino-6-phenylpyrido[2,3-d]pyrimidin-7-yl)-3-tert-butylureaIC503710.0 [1]
PD089828 analog 12IC5050000.0 [1]
1-[2-Amino-6-(3,5-diethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]-3-tert-butylureaIC501650.0 [1]
PD089828 analog 31IC5016000.0 [1]
C2 Pyrido[2,3-d]pyrimidin-7-one deriv. 23IC5044200.0 [1]
N8 Pyrido[2,3-d]pyrimidin-7-one deriv. 40IC506600.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Fibroblast growth factor receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/fibroblast-growth-factor-receptor-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Fibroblast growth factor receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/fibroblast-growth-factor-receptor-inhibitors-ic50-ki.
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