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Folate receptor alpha Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
PemetrexedIC5042.0 [1], 388.0 [2], 894.0 [3]
MethotrexateIC50114.0 [1], 216.0 [2], 461.0 [3]
RaltitrexedIC5015.0 [1], 1000.0 [2]
(2S)-2-[[5-[3-(2-Amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)propyl]thiophene-2-carbonyl]amino]pentanedioic acidIC500.31 [1], 0.38 [2], 173.0 [3], 1000.0 [4]
PralatrexateIC50168.0 [1], 1000.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseFolate receptor alpha Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2026https://www.aatbio.com/data-sets/folate-receptor-alpha-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2026May 9). Quest DatabaseFolate receptor alpha Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/folate-receptor-alpha-inhibitors-ic50-ki.
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