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GABA-A receptor; alpha-1/beta-2/gamma-2 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
DiazepamKi12.0 [1], 13.0 [2]
GabazineIC50240.0 [1], 349.0 [2]
Ethyl-8-azido-5,6-dihydro-5-methyl-6-oxo-4H-imidazo-1,4-benzodiazepine-3-carboxylateKi3.3 [1], 15.0 [2]
FlunitrazepamKi3.9 [1]
ZolpidemIC5010000.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseGABA-A receptor; alpha-1/beta-2/gamma-2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.13 Dec2025https://www.aatbio.com/data-sets/gaba-a-receptor-alpha-1-beta-2-gamma-2-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 13). Quest DatabaseGABA-A receptor; alpha-1/beta-2/gamma-2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/gaba-a-receptor-alpha-1-beta-2-gamma-2-inhibitors-ic50-ki.
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