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GABA-A receptor; alpha-2/beta-3/gamma-2 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
DiazepamKi6.6 [1]
Methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylateKi13.0 [1]
ZolpidemKi103.0 [1]
3-Methyl-6-[3-(trifluoromethyl)phenyl]-[1,2,4]triazolo[4,3-b]pyridazineKi720.0 [1], 1960.0 [2], 1964.0 [3], 2000.0 [4]
Ethyl 8-ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylateKi21.4 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseGABA-A receptor; alpha-2/beta-3/gamma-2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.17 Dec2025https://www.aatbio.com/data-sets/gaba-a-receptor-alpha-2-beta-3-gamma-2-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 17). Quest DatabaseGABA-A receptor; alpha-2/beta-3/gamma-2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/gaba-a-receptor-alpha-2-beta-3-gamma-2-inhibitors-ic50-ki.
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