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GABA A receptor alpha-4/beta-3/gamma-2 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
Ethyl 8-ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylateKi5.3 [1], 53.0 [2]
CID 5255267Ki1550.0 [1]
CID 9971547Ki38.8 [1], 300.0 [2]
Tert-Butyl beta-carboline-3-carboxylateKi1000.0 [1]
Ethyl 4-methyl-5-(1-methylethoxy)-9H-pyrido(3,4-b)indole-3-carboxylateKi137.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseGABA A receptor alpha-4/beta-3/gamma-2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.4 Dec2025https://www.aatbio.com/data-sets/gaba-a-receptor-alpha-4-beta-3-gamma-2-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 4). Quest DatabaseGABA A receptor alpha-4/beta-3/gamma-2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/gaba-a-receptor-alpha-4-beta-3-gamma-2-inhibitors-ic50-ki.
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