Name: GABA-A receptor; alpha-5/beta-3/gamma-2 Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

GABA-A receptor; alpha-5/beta-3/gamma-2 Inhibitors (IC50, Ki)

Structure	Compound Name	Standard Type	Standard Values (in nM)
	Methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate	Ki	1.0 ^[1], 2.2 ^[2]
	Diazepam	IC50	17.0 ^[1]
	Diazepam	Ki	11.0 ^[1], 11.2 ^[2]
	Zolpidem	Ki	3333.0 ^[1]
	3-Methyl-6-[3-(trifluoromethyl)phenyl]-[1,2,4]triazolo[4,3-b]pyridazine	Ki	460.0 ^[1], 560.0 ^[2], 561.0 ^[3]
Rows per page: 1–5 of 99

References

This online resource may be cited as follows

MLA	"Quest Database™ GABA-A receptor; alpha-5/beta-3/gamma-2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 12 Jun. 2026, https://www.aatbio.com/data-sets/gaba-a-receptor-alpha-5-beta-3-gamma-2-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2026, June 12). Quest Database™ GABA-A receptor; alpha-5/beta-3/gamma-2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/gaba-a-receptor-alpha-5-beta-3-gamma-2-inhibitors-ic50-ki.
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