Name: GABA-A receptor; alpha-6/beta-3/gamma-2 Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

GABA-A receptor; alpha-6/beta-3/gamma-2 Inhibitors (IC50, Ki)

Structure	Compound Name	Standard Type	Standard Values (in nM)
	Ethyl 8-ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	28.8 ^[1]
	Ethyl (7S)-15-methoxy-12-oxo-2,4,11-triazatetracyclo[11.4.0.02,6.07,11]heptadeca-1(17),3,5,13,15-pentaene-5-carboxylate	Ki	83.0 ^[1], 83.2 ^[2]
	Tert-butyl 8-ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	5.1 ^[1]
	Zolpidem	Ki	10000.0 ^[1]
	Ethyl-8-azido-5,6-dihydro-5-methyl-6-oxo-4H-imidazo-1,4-benzodiazepine-3-carboxylate	Ki	3.8 ^[1]
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References

This online resource may be cited as follows

MLA	"Quest Database™ GABA-A receptor; alpha-6/beta-3/gamma-2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 12 Dec. 2025, https://www.aatbio.com/data-sets/gaba-a-receptor-alpha-6-beta-3-gamma-2-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, December 12). Quest Database™ GABA-A receptor; alpha-6/beta-3/gamma-2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/gaba-a-receptor-alpha-6-beta-3-gamma-2-inhibitors-ic50-ki.
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