Name: GABA-A receptor; anion channel Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

GABA-A receptor; anion channel Inhibitors (IC50, Ki)

Structure	Compound Name	Standard Type	Standard Values (in nM)
	Diazepam	IC50	12.0 ^[1]
	Diazepam	Ki	10.0 ^[1]
	4-Butyl-3-[(3-chlorophenyl)methyl]-1H-1,2,4-triazole-5-thione	IC50	370.0 ^[1], 467.0 ^[2], 567.0 ^[3]
	4-Butyl-3-[(3-chlorophenyl)methyl]-1H-1,2,4-triazole-5-thione	Ki	88.0 ^[1], 93.3 ^[2], 113.0 ^[3]
	3-[(3-Chlorophenyl)methyl]-4-hexyl-1H-1,2,4-triazole-5-thione	IC50	361.0 ^[1], 535.0 ^[2], 626.0 ^[3]
Rows per page: 1–5 of 100

References

This online resource may be cited as follows

MLA	"Quest Database™ GABA-A receptor; anion channel Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 6 Dec. 2025, https://www.aatbio.com/data-sets/gaba-a-receptor-anion-channel-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, December 6). Quest Database™ GABA-A receptor; anion channel Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/gaba-a-receptor-anion-channel-inhibitors-ic50-ki.
BibTeX	EndNote	RefMan