 | Zolpidem | IC50 | 14.0 [1], 130.0 [2] |
| Zolpidem | Ki | 61.9 [1] |
 | Pentobarbital | IC50 | 1000000.0 [1] |
 | Flumazenil | Ki | 3.3 [1] |
 | Alisertib | IC50 | 490.0 [1] |
 | Eszopiclone | Ki | 50.1 [1] |
 | Ethyl (7S)-15-methoxy-12-oxo-2,4,11-triazatetracyclo[11.4.0.02,6.07,11]heptadeca-1(17),3,5,13,15-pentaene-5-carboxylate | Ki | 49.0 [1] |
 | 4-[[9-Chloro-7-(2,6-difluorophenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]benzoic acid | IC50 | 330.0 [1] |
 | 2-(4-Chlorophenyl)-3aH-pyrazolo[4,3-c]quinolin-3-one | IC50 | 1.0 [1] |
 | 3-[3-Tert-butyl-2-[(2-methyl-1,2,4-triazol-3-yl)methoxy]pyrazolo[1,5-d][1,2,4]triazin-7-yl]-5-methyl-1,2-oxazole | Ki | 0.8 [1] |
 | 1-Methyl-5-phenyl-1,3-dihydro-benzo[e][1,4]diazepin-2-one | IC50 | 10000.0 [1] |
 | N-(2-Oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-acetamide | IC50 | 10000.0 [1] |
 | 13-(4-Methyl-1,3-thiazol-2-yl)-15-pyridin-4-yl-4,11-diazatricyclo[9.4.0.02,7]pentadeca-1(15),2(7),3,5,13-pentaen-12-one | Ki | 1.3 [1] |
 | 4-Bromo-3,5-dimethyl-1-((4-(3-nitrophenyl)thiazol-2-yl)methyl)-1H-pyrazole | IC50 | 10000.0 [1] |
 | 4-[[9-Chloro-7-(2-fluoro-6-methoxyphenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]benzoic acid | IC50 | 150.0 [1] |
 | 8-Methyl-5-[4-(trifluoromethyl)-1-benzothiophen-2-yl]-1,9-dihydro-[1,3]oxazolo[4,5-h][2,3]benzodiazepin-2-one | IC50 | 479.0 [1] |
 | 3-(2-Chlorobenzyloxy)-2-(4-chlorophenyl)-6,7,8,9-tetrahydro-2H-pyrazolo[4,3-c]quinoline | IC50 | 46.0 [1] |
 | 2-(4-Chlorophenyl)-3-[(4-fluorophenyl)methoxy]-6,7,8,9-tetrahydropyrazolo[4,3-c]quinoline | IC50 | 50.0 [1] |
 | 2-(1,3-Benzodioxol-5-yl)-3-[(2-chlorophenyl)methoxy]pyrazolo[4,3-c]quinoline | IC50 | 50.0 [1] |
 | N-(4-Chlorophenyl)-5-(2-(methylthio)pyrimidin-4-yl)thiophene-2-sulfonamide | IC50 | 470.0 [1] |
 | 1-(4-Chlorobenzoyl)-6,6-dimethyl-3-methylsulfanyl-1,3,3a,5,7,7a-hexahydro-2-benzothiophen-4-one | IC50 | 580.0 [1] |
 | 1-(4-Chlorobenzoyl)-3-(methylthio)-hexahydrobenzo[c]thiophen-4(1H)-one | IC50 | 580.0 [1] |
 | 6,6-Dimethyl-3-methylsulfanyl-1-(3-nitrobenzoyl)-1,3,3a,5,7,7a-hexahydro-2-benzothiophen-4-one | IC50 | 10000.0 [1] |
 | (3-Aminobenzo[b]thiophen-2-yl)(4-chlorophenyl)methanone | IC50 | 1000.0 [1] |
 | 2-(4-Chlorophenyl)-3-(cyclopropylmethoxy)-8-imidazol-1-ylpyrazolo[4,3-c]quinoline | IC50 | 134.0 [1] |
 | 3-(2-Chlorobenzyloxy)-2-(4-chlorophenyl)-2H-pyrazolo[4,3-c]quinoline | IC50 | 64.0 [1] |
 | 2-(4-Chlorophenyl)-3-(cyclopropylmethoxy)-2H-pyrazolo[4,3-c]quinoline | IC50 | 74.0 [1] |
 | 4-(4-Chlorophenyl)-5-[(2-chlorophenyl)methoxy]-3,4,8-triazatricyclo[7.5.0.02,6]tetradeca-1(9),2,5,7-tetraene | IC50 | 242.0 [1] |
 | 2-(4-Chlorophenyl)-3-[(2-chlorophenyl)methoxy]-8,8-dimethyl-7,9-dihydro-6H-pyrazolo[4,3-c]quinoline | IC50 | 67.0 [1] |
 | 2-(4-Chlorophenyl)-3-[(4-chlorophenyl)methoxy]-6,7,8,9-tetrahydropyrazolo[4,3-c]quinoline | IC50 | 157.0 [1] |
 | 3-(2-Chlorophenoxy)-2-(4-chlorophenyl)-6,7,8,9-tetrahydropyrazolo[4,3-c]quinoline | IC50 | 3000.0 [1] |
 | 3-(2-Chlorobenzyloxy)-2-(2-fluorophenyl)-2H-pyrazolo[4,3-c]quinoline | IC50 | 1.0 [1] |
 | 2-(4-Chlorophenyl)-3-(cyclopropylmethoxy)-6,7,8,9-tetrahydropyrazolo[4,3-c]quinoline | IC50 | 94.0 [1] |
 | 2-(4-Chlorophenyl)-3-[(2-fluorophenyl)methoxy]-6,7,8,9-tetrahydropyrazolo[4,3-c]quinoline | IC50 | 64.0 [1] |
 | (5S)-1-Methyl-5-prop-2-enyl-5-[3-[3-(trifluoromethyl)diazirin-3-yl]phenyl]-1,3-diazinane-2,4,6-trione | IC50 | 120000.0 [1] |
 | (5R)-1-Methyl-5-prop-2-enyl-5-[3-[3-(trifluoromethyl)diazirin-3-yl]phenyl]-1,3-diazinane-2,4,6-trione | IC50 | 3800.0 [1] |
 | 2-[1-[2-(2-Methoxypyridin-3-yl)pyridin-4-yl]benzimidazol-5-yl]propan-2-ol | IC50 | 1.2 [1] |
 | 4-[4-[5-(2-Hydroxypropan-2-yl)benzimidazol-1-yl]pyridin-2-yl]pyridine-3-carbonitrile | IC50 | 26.0 [1] |
 | 2-[1-[2-(2-Chloropyridin-3-yl)pyridin-4-yl]benzimidazol-5-yl]propan-2-ol | IC50 | 38.0 [1] |
 | 2-[1-[2-(3-Fluoropyridin-4-yl)pyridin-4-yl]benzimidazol-5-yl]propan-2-ol | IC50 | 7.5 [1] |
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